Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0197 | 1 | 1 |
Plasmodium vivax | tubulin epsilon chain, putative | 0.0115 | 0.4715 | 0.4411 |
Brugia malayi | Tubulin beta chain | 0.005 | 0.0543 | 0.0333 |
Brugia malayi | Tubulin alpha-2 chain | 0.0168 | 0.8153 | 0.8113 |
Trichomonas vaginalis | tubulin, putative | 0.0197 | 1 | 1 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0168 | 0.8153 | 0.8047 |
Plasmodium falciparum | tubulin gamma chain | 0.0115 | 0.4715 | 0.4411 |
Trypanosoma brucei | epsilon tubulin | 0.0115 | 0.4715 | 0.4411 |
Brugia malayi | tubulin alpha-2 chain | 0.0168 | 0.8153 | 0.8113 |
Trichomonas vaginalis | tubulin, putative | 0.0065 | 0.1513 | 0.1026 |
Loa Loa (eye worm) | tubulin gamma chain | 0.0115 | 0.4715 | 0.4427 |
Giardia lamblia | Beta tubulin | 0.0197 | 1 | 1 |
Echinococcus granulosus | metabotropic glutamate receptor 5 | 0.0061 | 0.1249 | 0.1249 |
Trypanosoma brucei | epsilon tubulin | 0.0115 | 0.4715 | 0.4411 |
Wolbachia endosymbiont of Brugia malayi | cell division protein FtsZ | 0.005 | 0.0543 | 0.5 |
Trypanosoma brucei | beta tubulin | 0.0197 | 1 | 1 |
Plasmodium falciparum | alpha tubulin 1 | 0.0168 | 0.8153 | 0.8047 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0197 | 1 | 1 |
Brugia malayi | Tubulin alpha chain | 0.005 | 0.0543 | 0.0333 |
Echinococcus multilocularis | tubulin alpha chain | 0.0168 | 0.8153 | 0.8153 |
Echinococcus granulosus | tubulin alpha chain | 0.0168 | 0.8153 | 0.8153 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0065 | 0.1513 | 0.1026 |
Brugia malayi | Cell division protein ftsZ | 0.005 | 0.0543 | 0.0333 |
Entamoeba histolytica | tubulin family protein | 0.0197 | 1 | 1 |
Echinococcus granulosus | alpha tubulin | 0.0168 | 0.8153 | 0.8153 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0168 | 0.8153 | 0.8047 |
Echinococcus multilocularis | tubulin alpha chain | 0.0168 | 0.8153 | 0.8153 |
Echinococcus granulosus | tubulin alpha chain | 0.0168 | 0.8153 | 0.8153 |
Plasmodium vivax | tubulin gamma chain, putative | 0.0115 | 0.4715 | 0.4411 |
Loa Loa (eye worm) | hypothetical protein | 0.0168 | 0.8153 | 0.8053 |
Giardia lamblia | Beta tubulin | 0.0197 | 1 | 1 |
Trypanosoma brucei | alpha tubulin | 0.0168 | 0.8153 | 0.8047 |
Toxoplasma gondii | alpha tubulin TUBA1 | 0.0168 | 0.8153 | 0.8047 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0197 | 1 | 1 |
Leishmania major | beta tubulin | 0.0197 | 1 | 1 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0168 | 0.8153 | 0.8153 |
Echinococcus granulosus | tubulin gamma 1 chain | 0.0115 | 0.4715 | 0.4715 |
Brugia malayi | alpha-tubulin | 0.0168 | 0.8153 | 0.8113 |
Entamoeba histolytica | tubulin alpha chain, putative | 0.0168 | 0.8153 | 0.6506 |
Leishmania major | gamma-tubulin | 0.0115 | 0.4715 | 0.4411 |
Loa Loa (eye worm) | tubulin beta-1 chain | 0.0197 | 1 | 1 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0115 | 0.4715 | 0.4411 |
Echinococcus multilocularis | tubulin beta 1 chain | 0.0197 | 1 | 1 |
Trypanosoma cruzi | beta tubulin, putative | 0.0197 | 1 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0197 | 1 | 1 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0168 | 0.8153 | 0.8153 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0168 | 0.8153 | 0.8047 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0168 | 0.8153 | 0.8153 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0168 | 0.8153 | 0.8047 |
Schistosoma mansoni | tubulin subunit beta | 0.005 | 0.0543 | 0.0543 |
Echinococcus multilocularis | tubulin subunit TubB | 0.0168 | 0.8153 | 0.8153 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0168 | 0.8153 | 0.8047 |
Loa Loa (eye worm) | alpha-tubulin | 0.0168 | 0.8153 | 0.8053 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0115 | 0.4715 | 0.4411 |
Schistosoma mansoni | alpha tubulin | 0.0168 | 0.8153 | 0.8153 |
Giardia lamblia | Alpha-tubulin | 0.0168 | 0.8153 | 0.8047 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0168 | 0.8153 | 0.8153 |
Loa Loa (eye worm) | tubulin beta chain | 0.005 | 0.0543 | 0.0029 |
Echinococcus multilocularis | tubulin, beta 4A class IVa | 0.0197 | 1 | 1 |
Mycobacterium leprae | cell division protein FtsZ | 0.005 | 0.0543 | 0.5 |
Trypanosoma brucei | beta tubulin | 0.0197 | 1 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0168 | 0.8153 | 0.8047 |
Brugia malayi | Tubulin alpha-2 chain | 0.0168 | 0.8153 | 0.8113 |
Echinococcus multilocularis | hypothetical protein | 0.0168 | 0.8153 | 0.8153 |
Echinococcus granulosus | tubulin epsilon chain | 0.0115 | 0.4715 | 0.4715 |
Brugia malayi | beta-tubulin, identical | 0.0197 | 1 | 1 |
Schistosoma mansoni | tubulin subunit gamma | 0.0115 | 0.4715 | 0.4715 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0115 | 0.4715 | 0.4411 |
Trypanosoma cruzi | tubulin gamma chain | 0.0115 | 0.4715 | 0.4411 |
Loa Loa (eye worm) | hypothetical protein | 0.0061 | 0.1249 | 0.0773 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0168 | 0.8153 | 0.8047 |
Echinococcus multilocularis | tubulin alpha chain | 0.0168 | 0.8153 | 0.8153 |
Plasmodium falciparum | tubulin beta chain | 0.0197 | 1 | 1 |
Trypanosoma brucei | beta tubulin | 0.0115 | 0.4715 | 0.4411 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0168 | 0.8153 | 0.8153 |
Toxoplasma gondii | beta tubulin | 0.0197 | 1 | 1 |
Echinococcus granulosus | tubulin beta 1 chain | 0.0197 | 1 | 1 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0168 | 0.8153 | 0.8153 |
Echinococcus granulosus | tubulin beta 4A class IVa | 0.0197 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0168 | 0.8153 | 0.8047 |
Giardia lamblia | Alpha-tubulin | 0.0168 | 0.8153 | 0.8047 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0168 | 0.8153 | 0.8153 |
Trypanosoma cruzi | epsilon tubulin, putative | 0.0115 | 0.4715 | 0.4411 |
Schistosoma mansoni | tubulin subunit alpha | 0.005 | 0.0543 | 0.0543 |
Schistosoma mansoni | alpha tubulin | 0.0168 | 0.8153 | 0.8153 |
Echinococcus multilocularis | beta tubulin | 0.0197 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0168 | 0.8153 | 0.8047 |
Leishmania major | alpha tubulin | 0.0168 | 0.8153 | 0.8047 |
Echinococcus granulosus | tubulin subunit TubB | 0.0168 | 0.8153 | 0.8153 |
Toxoplasma gondii | alpha-tubulin I, putative | 0.0168 | 0.8153 | 0.8047 |
Echinococcus granulosus | tubulin alpha chain | 0.0168 | 0.8153 | 0.8153 |
Loa Loa (eye worm) | tubulin alpha-3 chain | 0.0103 | 0.3982 | 0.3655 |
Echinococcus multilocularis | metabotropic glutamate receptor 5 | 0.0061 | 0.1249 | 0.1249 |
Trypanosoma brucei | epsilon tubulin | 0.0115 | 0.4715 | 0.4411 |
Loa Loa (eye worm) | BEN-1 protein | 0.0197 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0168 | 0.8153 | 0.8047 |
Brugia malayi | Tubulin beta chain | 0.0065 | 0.1513 | 0.1325 |
Loa Loa (eye worm) | alpha-tubulin | 0.0168 | 0.8153 | 0.8053 |
Echinococcus granulosus | beta tubulin | 0.0197 | 1 | 1 |
Leishmania major | beta tubulin | 0.0197 | 1 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0197 | 1 | 1 |
Leishmania major | beta tubulin | 0.0197 | 1 | 1 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0197 | 1 | 1 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0168 | 0.8153 | 0.8153 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.0118 | 0.4952 | 0.4678 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0168 | 0.8153 | 0.8047 |
Treponema pallidum | cell division protein FtsZ | 0.005 | 0.0543 | 0.5 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0103 | 0.3982 | 0.3636 |
Entamoeba histolytica | tubulin family protein | 0.0197 | 1 | 1 |
Plasmodium falciparum | alpha tubulin 2 | 0.0168 | 0.8153 | 0.8047 |
Brugia malayi | Metabotropic glutamate receptor precursor. | 0.0049 | 0.0515 | 0.0305 |
Echinococcus granulosus | beta tubulin | 0.0197 | 1 | 1 |
Trypanosoma brucei | alpha tubulin | 0.0168 | 0.8153 | 0.8047 |
Trypanosoma brucei | beta tubulin | 0.0197 | 1 | 1 |
Leishmania major | epsilon tubulin, putative | 0.0115 | 0.4715 | 0.4411 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0065 | 0.1513 | 0.1026 |
Loa Loa (eye worm) | hypothetical protein | 0.0103 | 0.3982 | 0.3655 |
Toxoplasma gondii | beta-tubulin, putative | 0.0197 | 1 | 1 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0197 | 1 | 1 |
Toxoplasma gondii | beta-1 tubulin, putative | 0.0197 | 1 | 1 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0197 | 1 | 1 |
Onchocerca volvulus | 0.0065 | 0.1513 | 0.5 | |
Leishmania major | alpha tubulin | 0.0168 | 0.8153 | 0.8047 |
Echinococcus multilocularis | tubulin alpha | 0.0115 | 0.4715 | 0.4715 |
Trypanosoma cruzi | alpha tubulin, putative | 0.0168 | 0.8153 | 0.8047 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0168 | 0.8153 | 0.8047 |
Loa Loa (eye worm) | BEN-1 protein | 0.0197 | 1 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0168 | 0.8153 | 0.8047 |
Leishmania major | beta tubulin | 0.0197 | 1 | 1 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0168 | 0.8153 | 0.8053 |
Brugia malayi | Tubulin gamma chain | 0.0115 | 0.4715 | 0.4597 |
Leishmania major | beta tubulin | 0.0197 | 1 | 1 |
Schistosoma mansoni | tubulin subunit alpha | 0.0168 | 0.8153 | 0.8153 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0197 | 1 | 1 |
Mycobacterium tuberculosis | Cell division protein FtsZ | 0.005 | 0.0543 | 0.5 |
Echinococcus multilocularis | tubulin alpha chain | 0.0168 | 0.8153 | 0.8153 |
Leishmania major | beta tubulin | 0.0197 | 1 | 1 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0168 | 0.8153 | 0.8053 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.0118 | 0.4952 | 0.4678 |
Entamoeba histolytica | tubulin alpha-1 chain | 0.0168 | 0.8153 | 0.6506 |
Echinococcus multilocularis | tubulin epsilon chain | 0.0115 | 0.4715 | 0.4715 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0168 | 0.8153 | 0.8153 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0065 | 0.1513 | 0.1026 |
Leishmania major | alpha tubulin | 0.0168 | 0.8153 | 0.8047 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0197 | 1 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0197 | 1 | 1 |
Schistosoma mansoni | tubulin subunit alpha | 0.0168 | 0.8153 | 0.8153 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0197 | 1 | 1 |
Echinococcus multilocularis | tubulin alpha chain | 0.0168 | 0.8153 | 0.8153 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0168 | 0.8153 | 0.8153 |
Trypanosoma brucei | alpha tubulin | 0.0168 | 0.8153 | 0.8047 |
Plasmodium vivax | tubulin beta chain, putative | 0.0197 | 1 | 1 |
Schistosoma mansoni | alpha tubulin | 0.0168 | 0.8153 | 0.8153 |
Schistosoma mansoni | metabotropic glutamate receptor 2 3 (mglur group 2) | 0.0056 | 0.095 | 0.095 |
Echinococcus multilocularis | peroxisome assembly protein 26 | 0.0168 | 0.8153 | 0.8153 |
Trypanosoma brucei | alpha tubulin, putative | 0.0065 | 0.1513 | 0.1026 |
Echinococcus granulosus | tubulin alpha chain | 0.0168 | 0.8153 | 0.8153 |
Echinococcus multilocularis | tubulin gamma 1 chain | 0.0115 | 0.4715 | 0.4715 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0065 | 0.1513 | 0.1026 |
Leishmania major | alpha tubulin | 0.0168 | 0.8153 | 0.8047 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0197 | 1 | 1 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0118 | 0.4952 | 0.4662 |
Echinococcus granulosus | tubulin delta chain | 0.005 | 0.0543 | 0.0543 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0197 | 1 | 1 |
Leishmania major | beta tubulin | 0.0197 | 1 | 1 |
Trichomonas vaginalis | tubulin, putative | 0.0065 | 0.1513 | 0.1026 |
Schistosoma mansoni | tubulin subunit epsilon | 0.0115 | 0.4715 | 0.4715 |
Echinococcus multilocularis | tubulin delta chain | 0.005 | 0.0543 | 0.0543 |
Leishmania major | beta tubulin | 0.0197 | 1 | 1 |
Loa Loa (eye worm) | alpha-tubulin isotype 2 | 0.0118 | 0.4952 | 0.4678 |
Trypanosoma brucei | beta tubulin | 0.0197 | 1 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0197 | 1 | 1 |
Giardia lamblia | Beta tubulin | 0.0197 | 1 | 1 |
Schistosoma mansoni | tubulin subunit alpha | 0.0168 | 0.8153 | 0.8153 |
Leishmania major | beta tubulin | 0.0197 | 1 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0197 | 1 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0197 | 1 | 1 |
Leishmania major | beta tubulin | 0.0197 | 1 | 1 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0168 | 0.8153 | 0.8153 |
Leishmania major | alpha tubulin | 0.0168 | 0.8153 | 0.8047 |
Echinococcus multilocularis | beta tubulin | 0.0197 | 1 | 1 |
Loa Loa (eye worm) | tubulin alpha-2 chain | 0.0168 | 0.8153 | 0.8053 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0197 | 1 | 1 |
Loa Loa (eye worm) | tubulin beta-2A chain | 0.0197 | 1 | 1 |
Leishmania major | beta tubulin | 0.0197 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0168 | 0.8153 | 0.8047 |
Leishmania major | alpha tubulin | 0.0168 | 0.8153 | 0.8047 |
Loa Loa (eye worm) | tubulin beta chain | 0.0197 | 1 | 1 |
Echinococcus granulosus | tubulin alpha chain | 0.0168 | 0.8153 | 0.8153 |
Loa Loa (eye worm) | beta-tubulin | 0.0197 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0168 | 0.8153 | 0.8047 |
Leishmania major | beta tubulin | 0.0197 | 1 | 1 |
Echinococcus granulosus | tubulin subunit beta | 0.0197 | 1 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0197 | 1 | 1 |
Trypanosoma cruzi | epsilon tubulin, putative | 0.0115 | 0.4715 | 0.4411 |
Leishmania major | beta tubulin | 0.0197 | 1 | 1 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0065 | 0.1513 | 0.1026 |
Trypanosoma brucei | alpha tubulin | 0.0168 | 0.8153 | 0.8047 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0168 | 0.8153 | 0.8153 |
Echinococcus granulosus | tubulin alpha | 0.0115 | 0.4715 | 0.4715 |
Leishmania major | beta tubulin | 0.0197 | 1 | 1 |
Leishmania major | beta tubulin | 0.0197 | 1 | 1 |
Leishmania major | beta tubulin | 0.0197 | 1 | 1 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0168 | 0.8153 | 0.8153 |
Brugia malayi | Tubulin alpha chain | 0.0168 | 0.8153 | 0.8113 |
Loa Loa (eye worm) | tubulin beta-4 chain | 0.0197 | 1 | 1 |
Plasmodium falciparum | tubulin epsilon chain, putative | 0.0115 | 0.4715 | 0.4411 |
Leishmania major | beta tubulin | 0.0197 | 1 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0197 | 1 | 1 |
Leishmania major | beta tubulin | 0.0197 | 1 | 1 |
Toxoplasma gondii | tubulin/FtsZ family, GTPase domain-containing protein | 0.0115 | 0.4715 | 0.4411 |
Mycobacterium ulcerans | cell division protein FtsZ | 0.005 | 0.0543 | 0.5 |
Trypanosoma brucei | tubulin gamma chain | 0.0115 | 0.4715 | 0.4411 |
Echinococcus multilocularis | tubulin subunit beta | 0.0197 | 1 | 1 |
Schistosoma mansoni | tubulin subunit delta | 0.005 | 0.0543 | 0.0543 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.0053 | 0.078 | 0.028 |
Leishmania major | alpha tubulin | 0.0168 | 0.8153 | 0.8047 |
Schistosoma mansoni | tubulin subunit beta | 0.0197 | 1 | 1 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0168 | 0.8153 | 0.8153 |
Loa Loa (eye worm) | hypothetical protein | 0.0118 | 0.4952 | 0.4678 |
Giardia lamblia | Gamma tubulin | 0.0115 | 0.4715 | 0.4411 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0168 | 0.8153 | 0.8047 |
Echinococcus granulosus | peroxisome assembly protein 26 | 0.0168 | 0.8153 | 0.8153 |
Brugia malayi | tubulin alpha chain - mouse | 0.0168 | 0.8153 | 0.8113 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
Inhibition (binding) | = 8 % | Inhibition of pig kidney microsomal APN at 10 uM | ChEMBL. | 17326615 |
Inhibition (binding) | = 8 % | Inhibition of pig kidney microsomal APN at 10 uM | ChEMBL. | 17326615 |
Inhibition (binding) | = 64 % | Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidase at 10 uM | ChEMBL. | 17326615 |
Inhibition (binding) | = 64 % | Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidase at 10 uM | ChEMBL. | 17326615 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.