Drug uptake (ADMET)
|
= 0.11 % ID/g
|
Biodistribution in muscle of iv dosed testis-intact Sprague-Dawley rat after 18 hrs block
|
ChEMBL.
|
17328524
|
Drug uptake (ADMET)
|
= 0.12 % ID/g
|
Biodistribution in bone of iv dosed testis-intact Sprague-Dawley rat after 18 hrs block
|
ChEMBL.
|
17328524
|
Drug uptake (ADMET)
|
= 0.13 % ID/g
|
Biodistribution in bone of iv dosed Sprague-Dawley rat after 18 hrs
|
ChEMBL.
|
17328524
|
Drug uptake (ADMET)
|
= 0.15 % ID/g
|
Biodistribution in muscle of iv dosed Sprague-Dawley rat after 18 hrs
|
ChEMBL.
|
17328524
|
Drug uptake (ADMET)
|
= 0.22 % ID/g
|
Biodistribution in prostate of iv dosed testis-intact Sprague-Dawley rat after 18 hrs block
|
ChEMBL.
|
17328524
|
Drug uptake (ADMET)
|
= 0.26 % ID/g
|
Biodistribution in kidney of iv dosed testis-intact Sprague-Dawley rat after 18 hrs block
|
ChEMBL.
|
17328524
|
Drug uptake (ADMET)
|
= 0.27 % ID/g
|
Biodistribution in prostate of iv dosed Sprague-Dawley rat after 18 hrs
|
ChEMBL.
|
17328524
|
Drug uptake (ADMET)
|
= 0.28 % ID/g
|
Biodistribution in bone of iv dosed Sprague-Dawley rat after 1 hr
|
ChEMBL.
|
17328524
|
Drug uptake (ADMET)
|
= 0.29 % ID/g
|
Biodistribution in blood of iv dosed testis-intact Sprague-Dawley rat after 18 hrs block
|
ChEMBL.
|
17328524
|
Drug uptake (ADMET)
|
= 0.31 % ID/g
|
Biodistribution in bone of iv dosed testis-intact Sprague-Dawley rat after 1 hr block
|
ChEMBL.
|
17328524
|
Drug uptake (ADMET)
|
= 0.34 % ID/g
|
Biodistribution in blood of iv dosed Sprague-Dawley rat after 18 hrs
|
ChEMBL.
|
17328524
|
Drug uptake (ADMET)
|
= 0.34 % ID/g
|
Biodistribution in muscle of iv dosed Sprague-Dawley rat after 1 hr
|
ChEMBL.
|
17328524
|
Drug uptake (ADMET)
|
= 0.36 % ID/g
|
Biodistribution in liver of iv dosed testis-intact Sprague-Dawley rat after 18 hrs block
|
ChEMBL.
|
17328524
|
Drug uptake (ADMET)
|
= 0.36 % ID/g
|
Biodistribution in kidney of iv dosed Sprague-Dawley rat after 18 hrs
|
ChEMBL.
|
17328524
|
Drug uptake (ADMET)
|
= 0.38 % ID/g
|
Biodistribution in muscle of iv dosed testis-intact Sprague-Dawley rat after 1 hr block
|
ChEMBL.
|
17328524
|
Drug uptake (ADMET)
|
= 0.56 % ID/g
|
Biodistribution in blood of iv dosed Sprague-Dawley rat after 1 hr
|
ChEMBL.
|
17328524
|
Drug uptake (ADMET)
|
= 0.56 % ID/g
|
Biodistribution in liver of iv dosed Sprague-Dawley rat after 18 hrs
|
ChEMBL.
|
17328524
|
Drug uptake (ADMET)
|
= 0.62 % ID/g
|
Biodistribution in blood of iv dosed testis-intact Sprague-Dawley rat after 1 hr block
|
ChEMBL.
|
17328524
|
Drug uptake (ADMET)
|
= 0.68 % ID/g
|
Biodistribution in prostate of iv dosed testis-intact Sprague-Dawley rat after 1 hr block
|
ChEMBL.
|
17328524
|
Drug uptake (ADMET)
|
= 1 % ID/g
|
Biodistribution in kidney of iv dosed Sprague-Dawley rat after 1 hr
|
ChEMBL.
|
17328524
|
Drug uptake (ADMET)
|
= 1 % ID/g
|
Biodistribution in kidney of iv dosed testis-intact Sprague-Dawley rat after 1 hr block
|
ChEMBL.
|
17328524
|
Drug uptake (ADMET)
|
= 1 % ID/g
|
Biodistribution in prostate of iv dosed Sprague-Dawley rat after 1 hr
|
ChEMBL.
|
17328524
|
Drug uptake (ADMET)
|
= 2.1 % ID/g
|
Biodistribution in liver of iv dosed Sprague-Dawley rat after 1 hr
|
ChEMBL.
|
17328524
|
Drug uptake (ADMET)
|
= 2.2 % ID/g
|
Biodistribution in prostate of iv dosed CWR22 tumor bearing mouse after 30 min
|
ChEMBL.
|
17328524
|
Drug uptake (ADMET)
|
= 2.5 % ID/g
|
Biodistribution in liver of iv dosed testis-intact Sprague-Dawley rat after 1 hr block
|
ChEMBL.
|
17328524
|
Drug uptake (ADMET)
|
= 2.5 % ID/g
|
Biodistribution in muscle of iv dosed CWR22 tumor bearing mouse after 30 min
|
ChEMBL.
|
17328524
|
Drug uptake (ADMET)
|
= 2.5 % ID/g
|
Biodistribution in tumor of iv dosed CWR22 tumor bearing mouse after 30 min
|
ChEMBL.
|
17328524
|
Drug uptake (ADMET)
|
= 2.7 % ID/g
|
Biodistribution in blood of iv dosed CWR22 tumor bearing mouse after 30 min
|
ChEMBL.
|
17328524
|
Drug uptake (ADMET)
|
= 2.8 % ID/g
|
Biodistribution in muscle of iv dosed CWR22 tumor bearing mouse with 17alpha-methyltestosterone-induced androgen block after 90 min
|
ChEMBL.
|
17328524
|
Drug uptake (ADMET)
|
= 2.8 % ID/g
|
Biodistribution in prostate of iv dosed CWR22 tumor bearing mouse after 60 min
|
ChEMBL.
|
17328524
|
Drug uptake (ADMET)
|
= 2.9 % ID/g
|
Biodistribution in muscle of iv dosed CWR22 tumor bearing mouse after 60 min
|
ChEMBL.
|
17328524
|
Drug uptake (ADMET)
|
= 3 % ID/g
|
Biodistribution in blood of iv dosed CWR22 tumor bearing mouse with 17alpha-methyltestosterone-induced androgen block after 90 min
|
ChEMBL.
|
17328524
|
Drug uptake (ADMET)
|
= 3.4 % ID/g
|
Biodistribution in prostate of iv dosed CWR22 tumor bearing mouse with 17alpha-methyltestosterone-induced androgen block after 90 min
|
ChEMBL.
|
17328524
|
Drug uptake (ADMET)
|
= 3.5 % ID/g
|
Biodistribution in blood of iv dosed CWR22 tumor bearing mouse after 60 min
|
ChEMBL.
|
17328524
|
Drug uptake (ADMET)
|
= 3.8 % ID/g
|
Biodistribution in tumor of iv dosed CWR22 tumor bearing mouse after 60 min
|
ChEMBL.
|
17328524
|
Drug uptake (ADMET)
|
= 4.5 % ID/g
|
Biodistribution in tumor of iv dosed CWR22 tumor bearing mouse with 17alpha-methyltestosterone-induced androgen block after 90 min
|
ChEMBL.
|
17328524
|
Drug uptake (ADMET)
|
= 7.2 % ID/g
|
Biodistribution in kidney of iv dosed CWR22 tumor bearing mouse after 30 min
|
ChEMBL.
|
17328524
|
Drug uptake (ADMET)
|
= 7.6 % ID/g
|
Biodistribution in kidney of iv dosed CWR22 tumor bearing mouse with 17alpha-methyltestosterone-induced androgen block after 90 min
|
ChEMBL.
|
17328524
|
Drug uptake (ADMET)
|
= 7.8 % ID/g
|
Biodistribution in kidney of iv dosed CWR22 tumor bearing mouse after 60 min
|
ChEMBL.
|
17328524
|
Drug uptake (ADMET)
|
= 14 % ID/g
|
Biodistribution in liver of iv dosed CWR22 tumor bearing mouse with 17alpha-methyltestosterone-induced androgen block after 90 min
|
ChEMBL.
|
17328524
|
Drug uptake (ADMET)
|
= 15 % ID/g
|
Biodistribution in liver of iv dosed CWR22 tumor bearing mouse after 30 min
|
ChEMBL.
|
17328524
|
Drug uptake (ADMET)
|
= 18 % ID/g
|
Biodistribution in liver of iv dosed CWR22 tumor bearing mouse after 60 min
|
ChEMBL.
|
17328524
|
Ratio (ADMET)
|
= 1.8
|
Ratio of drug uptake in prostate to blood in iv dosed Sprague-Dawley rat after 1 hr
|
ChEMBL.
|
17328524
|
Ratio (ADMET)
|
= 2.9
|
Ratio of drug uptake in prostate to muscle in iv dosed Sprague-Dawley rat after 1 hr
|
ChEMBL.
|
17328524
|