Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Mycobacterium tuberculosis | 3-dehydroquinate dehydratase AroD (AROQ) (3-dehydroquinase) (type II dhqase) | 0.2577 | 1 | 0.5 |
Entamoeba histolytica | tubulin family protein | 0.0027 | 0.0064 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0027 | 0.0064 | 1 |
Leishmania major | beta tubulin | 0.0027 | 0.0064 | 1 |
Loa Loa (eye worm) | beta-tubulin | 0.0027 | 0.0064 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0027 | 0.0064 | 1 |
Echinococcus granulosus | tubulin beta 4A class IVa | 0.0027 | 0.0064 | 1 |
Giardia lamblia | Beta tubulin | 0.0027 | 0.0064 | 1 |
Loa Loa (eye worm) | BEN-1 protein | 0.0027 | 0.0064 | 1 |
Leishmania major | beta tubulin | 0.0027 | 0.0064 | 1 |
Leishmania major | beta tubulin | 0.0027 | 0.0064 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0027 | 0.0064 | 1 |
Trypanosoma brucei | beta tubulin | 0.0027 | 0.0064 | 1 |
Leishmania major | beta tubulin | 0.0027 | 0.0064 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0027 | 0.0064 | 1 |
Toxoplasma gondii | beta-1 tubulin, putative | 0.0027 | 0.0064 | 1 |
Loa Loa (eye worm) | tubulin beta-2A chain | 0.0027 | 0.0064 | 1 |
Giardia lamblia | Beta tubulin | 0.0027 | 0.0064 | 1 |
Echinococcus multilocularis | tubulin subunit beta | 0.0027 | 0.0064 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0027 | 0.0064 | 1 |
Echinococcus multilocularis | tubulin beta 1 chain | 0.0027 | 0.0064 | 1 |
Leishmania major | beta tubulin | 0.0027 | 0.0064 | 1 |
Loa Loa (eye worm) | BEN-1 protein | 0.0027 | 0.0064 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0027 | 0.0064 | 1 |
Leishmania major | beta tubulin | 0.0027 | 0.0064 | 1 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0027 | 0.0064 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0027 | 0.0064 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0027 | 0.0064 | 1 |
Toxoplasma gondii | beta-tubulin, putative | 0.0027 | 0.0064 | 1 |
Entamoeba histolytica | tubulin family protein | 0.0027 | 0.0064 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0027 | 0.0064 | 1 |
Echinococcus multilocularis | beta tubulin | 0.0027 | 0.0064 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0027 | 0.0064 | 1 |
Giardia lamblia | Beta tubulin | 0.0027 | 0.0064 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0027 | 0.0064 | 1 |
Leishmania major | beta tubulin | 0.0027 | 0.0064 | 1 |
Leishmania major | beta tubulin | 0.0027 | 0.0064 | 1 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0027 | 0.0064 | 1 |
Leishmania major | beta tubulin | 0.0027 | 0.0064 | 1 |
Echinococcus granulosus | tubulin beta 1 chain | 0.0027 | 0.0064 | 1 |
Leishmania major | beta tubulin | 0.0027 | 0.0064 | 1 |
Leishmania major | beta tubulin | 0.0027 | 0.0064 | 1 |
Leishmania major | beta tubulin | 0.0027 | 0.0064 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0027 | 0.0064 | 1 |
Leishmania major | beta tubulin | 0.0027 | 0.0064 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0027 | 0.0064 | 1 |
Loa Loa (eye worm) | tubulin beta-1 chain | 0.0027 | 0.0064 | 1 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0027 | 0.0064 | 1 |
Leishmania major | beta tubulin | 0.0027 | 0.0064 | 1 |
Toxoplasma gondii | beta tubulin | 0.0027 | 0.0064 | 1 |
Trypanosoma cruzi | beta tubulin, putative | 0.0027 | 0.0064 | 1 |
Echinococcus granulosus | beta tubulin | 0.0027 | 0.0064 | 1 |
Trichomonas vaginalis | tubulin, putative | 0.0027 | 0.0064 | 1 |
Leishmania major | beta tubulin | 0.0027 | 0.0064 | 1 |
Echinococcus granulosus | beta tubulin | 0.0027 | 0.0064 | 1 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0027 | 0.0064 | 1 |
Trypanosoma brucei | beta tubulin | 0.0027 | 0.0064 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0027 | 0.0064 | 1 |
Mycobacterium ulcerans | 3-dehydroquinate dehydratase | 0.2577 | 1 | 0.5 |
Echinococcus multilocularis | tubulin, beta 4A class IVa | 0.0027 | 0.0064 | 1 |
Echinococcus granulosus | tubulin subunit beta | 0.0027 | 0.0064 | 1 |
Plasmodium falciparum | tubulin beta chain | 0.0027 | 0.0064 | 1 |
Trypanosoma brucei | beta tubulin | 0.0027 | 0.0064 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0027 | 0.0064 | 1 |
Brugia malayi | beta-tubulin, identical | 0.0027 | 0.0064 | 1 |
Leishmania major | beta tubulin | 0.0027 | 0.0064 | 1 |
Trypanosoma brucei | beta tubulin | 0.0027 | 0.0064 | 1 |
Plasmodium vivax | tubulin beta chain, putative | 0.0027 | 0.0064 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0027 | 0.0064 | 1 |
Echinococcus multilocularis | beta tubulin | 0.0027 | 0.0064 | 1 |
Leishmania major | beta tubulin | 0.0027 | 0.0064 | 1 |
Brugia malayi | Tubulin beta-1 chain | 0.0027 | 0.0064 | 1 |
Leishmania major | beta tubulin | 0.0027 | 0.0064 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0027 | 0.0064 | 1 |
Loa Loa (eye worm) | tubulin beta chain | 0.0027 | 0.0064 | 1 |
Loa Loa (eye worm) | tubulin beta-4 chain | 0.0027 | 0.0064 | 1 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
IC50 (binding) | = 1 nM | Inhibition of FTase by SPA | ChEMBL. | 17316920 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.