Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0026 | 0.0067 | 1 |
Leishmania major | beta tubulin | 0.0026 | 0.0067 | 1 |
Leishmania major | beta tubulin | 0.0026 | 0.0067 | 1 |
Leishmania major | beta tubulin | 0.0026 | 0.0067 | 1 |
Leishmania major | beta tubulin | 0.0026 | 0.0067 | 1 |
Loa Loa (eye worm) | tubulin beta-4 chain | 0.0026 | 0.0067 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0026 | 0.0067 | 1 |
Loa Loa (eye worm) | BEN-1 protein | 0.0026 | 0.0067 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0026 | 0.0067 | 1 |
Echinococcus granulosus | beta tubulin | 0.0026 | 0.0067 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0026 | 0.0067 | 1 |
Echinococcus granulosus | beta tubulin | 0.0026 | 0.0067 | 1 |
Leishmania major | beta tubulin | 0.0026 | 0.0067 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0026 | 0.0067 | 1 |
Leishmania major | beta tubulin | 0.0026 | 0.0067 | 1 |
Leishmania major | beta tubulin | 0.0026 | 0.0067 | 1 |
Loa Loa (eye worm) | BEN-1 protein | 0.0026 | 0.0067 | 1 |
Leishmania major | beta tubulin | 0.0026 | 0.0067 | 1 |
Echinococcus multilocularis | beta tubulin | 0.0026 | 0.0067 | 1 |
Echinococcus multilocularis | beta tubulin | 0.0026 | 0.0067 | 1 |
Brugia malayi | beta-tubulin, identical | 0.0026 | 0.0067 | 1 |
Brugia malayi | Tubulin beta-1 chain | 0.0026 | 0.0067 | 1 |
Leishmania major | beta tubulin | 0.0026 | 0.0067 | 1 |
Giardia lamblia | Beta tubulin | 0.0026 | 0.0067 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0026 | 0.0067 | 1 |
Echinococcus multilocularis | tubulin beta 1 chain | 0.0026 | 0.0067 | 1 |
Loa Loa (eye worm) | tubulin beta-1 chain | 0.0026 | 0.0067 | 1 |
Leishmania major | beta tubulin | 0.0026 | 0.0067 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0026 | 0.0067 | 1 |
Leishmania major | beta tubulin | 0.0026 | 0.0067 | 1 |
Echinococcus granulosus | tubulin beta 1 chain | 0.0026 | 0.0067 | 1 |
Toxoplasma gondii | beta-tubulin, putative | 0.0026 | 0.0067 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0026 | 0.0067 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0026 | 0.0067 | 1 |
Plasmodium falciparum | tubulin beta chain | 0.0026 | 0.0067 | 1 |
Entamoeba histolytica | tubulin family protein | 0.0026 | 0.0067 | 1 |
Trypanosoma brucei | beta tubulin | 0.0026 | 0.0067 | 1 |
Echinococcus granulosus | tubulin subunit beta | 0.0026 | 0.0067 | 1 |
Leishmania major | beta tubulin | 0.0026 | 0.0067 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0026 | 0.0067 | 1 |
Trypanosoma brucei | beta tubulin | 0.0026 | 0.0067 | 1 |
Mycobacterium tuberculosis | 3-dehydroquinate dehydratase AroD (AROQ) (3-dehydroquinase) (type II dhqase) | 0.2391 | 1 | 0.5 |
Plasmodium vivax | tubulin beta chain, putative | 0.0026 | 0.0067 | 1 |
Giardia lamblia | Beta tubulin | 0.0026 | 0.0067 | 1 |
Leishmania major | beta tubulin | 0.0026 | 0.0067 | 1 |
Leishmania major | beta tubulin | 0.0026 | 0.0067 | 1 |
Toxoplasma gondii | beta tubulin | 0.0026 | 0.0067 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0026 | 0.0067 | 1 |
Echinococcus multilocularis | tubulin subunit beta | 0.0026 | 0.0067 | 1 |
Mycobacterium ulcerans | 3-dehydroquinate dehydratase | 0.2391 | 1 | 0.5 |
Leishmania major | beta tubulin | 0.0026 | 0.0067 | 1 |
Loa Loa (eye worm) | tubulin beta chain | 0.0026 | 0.0067 | 1 |
Leishmania major | beta tubulin | 0.0026 | 0.0067 | 1 |
Echinococcus granulosus | tubulin beta 4A class IVa | 0.0026 | 0.0067 | 1 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0026 | 0.0067 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0026 | 0.0067 | 1 |
Echinococcus multilocularis | tubulin, beta 4A class IVa | 0.0026 | 0.0067 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0026 | 0.0067 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0026 | 0.0067 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0026 | 0.0067 | 1 |
Toxoplasma gondii | beta-1 tubulin, putative | 0.0026 | 0.0067 | 1 |
Trypanosoma cruzi | beta tubulin, putative | 0.0026 | 0.0067 | 1 |
Trypanosoma brucei | beta tubulin | 0.0026 | 0.0067 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0026 | 0.0067 | 1 |
Entamoeba histolytica | tubulin family protein | 0.0026 | 0.0067 | 1 |
Leishmania major | beta tubulin | 0.0026 | 0.0067 | 1 |
Loa Loa (eye worm) | beta-tubulin | 0.0026 | 0.0067 | 1 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0026 | 0.0067 | 1 |
Giardia lamblia | Beta tubulin | 0.0026 | 0.0067 | 1 |
Trichomonas vaginalis | tubulin, putative | 0.0026 | 0.0067 | 1 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0026 | 0.0067 | 1 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0026 | 0.0067 | 1 |
Trypanosoma brucei | beta tubulin | 0.0026 | 0.0067 | 1 |
Leishmania major | beta tubulin | 0.0026 | 0.0067 | 1 |
Loa Loa (eye worm) | tubulin beta-2A chain | 0.0026 | 0.0067 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0026 | 0.0067 | 1 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
log(1/ID50) (functional) | = -2.152 | Antiproliferative activity against human HCV29T cells by SRB method | ChEMBL. | 17320247 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.