Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0028 | 0.0067 | 1 |
Trypanosoma brucei | beta tubulin | 0.0028 | 0.0067 | 1 |
Echinococcus multilocularis | beta tubulin | 0.0028 | 0.0067 | 1 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0028 | 0.0067 | 1 |
Leishmania major | beta tubulin | 0.0028 | 0.0067 | 1 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0028 | 0.0067 | 1 |
Entamoeba histolytica | tubulin family protein | 0.0028 | 0.0067 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0028 | 0.0067 | 1 |
Leishmania major | beta tubulin | 0.0028 | 0.0067 | 1 |
Mycobacterium tuberculosis | 3-dehydroquinate dehydratase AroD (AROQ) (3-dehydroquinase) (type II dhqase) | 0.2542 | 1 | 0.5 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0028 | 0.0067 | 1 |
Leishmania major | beta tubulin | 0.0028 | 0.0067 | 1 |
Leishmania major | beta tubulin | 0.0028 | 0.0067 | 1 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0028 | 0.0067 | 1 |
Trypanosoma brucei | beta tubulin | 0.0028 | 0.0067 | 1 |
Leishmania major | beta tubulin | 0.0028 | 0.0067 | 1 |
Plasmodium vivax | tubulin beta chain, putative | 0.0028 | 0.0067 | 1 |
Leishmania major | beta tubulin | 0.0028 | 0.0067 | 1 |
Echinococcus granulosus | beta tubulin | 0.0028 | 0.0067 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0028 | 0.0067 | 1 |
Loa Loa (eye worm) | beta-tubulin | 0.0028 | 0.0067 | 1 |
Loa Loa (eye worm) | tubulin beta-1 chain | 0.0028 | 0.0067 | 1 |
Leishmania major | beta tubulin | 0.0028 | 0.0067 | 1 |
Entamoeba histolytica | tubulin family protein | 0.0028 | 0.0067 | 1 |
Loa Loa (eye worm) | tubulin beta chain | 0.0028 | 0.0067 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0028 | 0.0067 | 1 |
Giardia lamblia | Beta tubulin | 0.0028 | 0.0067 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0028 | 0.0067 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0028 | 0.0067 | 1 |
Leishmania major | beta tubulin | 0.0028 | 0.0067 | 1 |
Leishmania major | beta tubulin | 0.0028 | 0.0067 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0028 | 0.0067 | 1 |
Leishmania major | beta tubulin | 0.0028 | 0.0067 | 1 |
Echinococcus multilocularis | beta tubulin | 0.0028 | 0.0067 | 1 |
Echinococcus multilocularis | tubulin, beta 4A class IVa | 0.0028 | 0.0067 | 1 |
Leishmania major | beta tubulin | 0.0028 | 0.0067 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0028 | 0.0067 | 1 |
Echinococcus granulosus | tubulin beta 1 chain | 0.0028 | 0.0067 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0028 | 0.0067 | 1 |
Echinococcus granulosus | tubulin subunit beta | 0.0028 | 0.0067 | 1 |
Trypanosoma brucei | beta tubulin | 0.0028 | 0.0067 | 1 |
Brugia malayi | beta-tubulin, identical | 0.0028 | 0.0067 | 1 |
Toxoplasma gondii | beta tubulin | 0.0028 | 0.0067 | 1 |
Giardia lamblia | Beta tubulin | 0.0028 | 0.0067 | 1 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0028 | 0.0067 | 1 |
Toxoplasma gondii | beta-1 tubulin, putative | 0.0028 | 0.0067 | 1 |
Leishmania major | beta tubulin | 0.0028 | 0.0067 | 1 |
Plasmodium falciparum | tubulin beta chain | 0.0028 | 0.0067 | 1 |
Brugia malayi | Tubulin beta-1 chain | 0.0028 | 0.0067 | 1 |
Leishmania major | beta tubulin | 0.0028 | 0.0067 | 1 |
Toxoplasma gondii | beta-tubulin, putative | 0.0028 | 0.0067 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0028 | 0.0067 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0028 | 0.0067 | 1 |
Leishmania major | beta tubulin | 0.0028 | 0.0067 | 1 |
Leishmania major | beta tubulin | 0.0028 | 0.0067 | 1 |
Giardia lamblia | Beta tubulin | 0.0028 | 0.0067 | 1 |
Echinococcus multilocularis | tubulin beta 1 chain | 0.0028 | 0.0067 | 1 |
Loa Loa (eye worm) | tubulin beta-4 chain | 0.0028 | 0.0067 | 1 |
Trichomonas vaginalis | tubulin, putative | 0.0028 | 0.0067 | 1 |
Echinococcus multilocularis | tubulin subunit beta | 0.0028 | 0.0067 | 1 |
Leishmania major | beta tubulin | 0.0028 | 0.0067 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0028 | 0.0067 | 1 |
Trypanosoma cruzi | beta tubulin, putative | 0.0028 | 0.0067 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0028 | 0.0067 | 1 |
Echinococcus granulosus | tubulin beta 4A class IVa | 0.0028 | 0.0067 | 1 |
Loa Loa (eye worm) | BEN-1 protein | 0.0028 | 0.0067 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0028 | 0.0067 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0028 | 0.0067 | 1 |
Leishmania major | beta tubulin | 0.0028 | 0.0067 | 1 |
Echinococcus granulosus | beta tubulin | 0.0028 | 0.0067 | 1 |
Loa Loa (eye worm) | BEN-1 protein | 0.0028 | 0.0067 | 1 |
Mycobacterium ulcerans | 3-dehydroquinate dehydratase | 0.2542 | 1 | 0.5 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0028 | 0.0067 | 1 |
Trypanosoma brucei | beta tubulin | 0.0028 | 0.0067 | 1 |
Loa Loa (eye worm) | tubulin beta-2A chain | 0.0028 | 0.0067 | 1 |
Leishmania major | beta tubulin | 0.0028 | 0.0067 | 1 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
log(1/ID50) (functional) | < -2.567 | Antiproliferative activity against human HCV29T cells by SRB method | ChEMBL. | 17320247 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.