Species | Target name | Source | Bibliographic reference |
---|---|---|---|
Homo sapiens | arginine vasopressin receptor 1A | Starlite/ChEMBL | References |
Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Loa Loa (eye worm) | tubulin beta-1 chain | 0.0176 | 1 | 1 |
Leishmania major | beta tubulin | 0.0176 | 1 | 1 |
Echinococcus multilocularis | tubulin, beta 4A class IVa | 0.0176 | 1 | 1 |
Plasmodium vivax | tubulin beta chain, putative | 0.0176 | 1 | 1 |
Leishmania major | beta tubulin | 0.0176 | 1 | 1 |
Leishmania major | beta tubulin | 0.0176 | 1 | 1 |
Loa Loa (eye worm) | tubulin beta-2A chain | 0.0176 | 1 | 1 |
Echinococcus multilocularis | tubulin beta 1 chain | 0.0176 | 1 | 1 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0176 | 1 | 1 |
Trypanosoma brucei | beta tubulin | 0.0176 | 1 | 1 |
Echinococcus granulosus | tubulin beta 4A class IVa | 0.0176 | 1 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0176 | 1 | 1 |
Brugia malayi | beta-tubulin, identical | 0.0176 | 1 | 1 |
Leishmania major | beta tubulin | 0.0176 | 1 | 1 |
Leishmania major | beta tubulin | 0.0176 | 1 | 1 |
Leishmania major | beta tubulin | 0.0176 | 1 | 1 |
Echinococcus multilocularis | beta tubulin | 0.0176 | 1 | 1 |
Toxoplasma gondii | beta tubulin | 0.0176 | 1 | 1 |
Entamoeba histolytica | tubulin family protein | 0.0176 | 1 | 1 |
Leishmania major | beta tubulin | 0.0176 | 1 | 1 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0176 | 1 | 1 |
Loa Loa (eye worm) | tubulin beta chain | 0.0176 | 1 | 1 |
Giardia lamblia | Beta tubulin | 0.0176 | 1 | 1 |
Loa Loa (eye worm) | beta-tubulin | 0.0176 | 1 | 1 |
Leishmania major | beta tubulin | 0.0176 | 1 | 1 |
Toxoplasma gondii | beta-tubulin, putative | 0.0176 | 1 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0176 | 1 | 1 |
Leishmania major | beta tubulin | 0.0176 | 1 | 1 |
Echinococcus granulosus | tubulin subunit beta | 0.0176 | 1 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0176 | 1 | 1 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0176 | 1 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0176 | 1 | 1 |
Loa Loa (eye worm) | BEN-1 protein | 0.0176 | 1 | 1 |
Leishmania major | beta tubulin | 0.0176 | 1 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0176 | 1 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0176 | 1 | 1 |
Trypanosoma brucei | beta tubulin | 0.0176 | 1 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0176 | 1 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0176 | 1 | 1 |
Leishmania major | beta tubulin | 0.0176 | 1 | 1 |
Loa Loa (eye worm) | BEN-1 protein | 0.0176 | 1 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0176 | 1 | 1 |
Leishmania major | beta tubulin | 0.0176 | 1 | 1 |
Echinococcus granulosus | beta tubulin | 0.0176 | 1 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0176 | 1 | 1 |
Echinococcus granulosus | beta tubulin | 0.0176 | 1 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0176 | 1 | 1 |
Leishmania major | beta tubulin | 0.0176 | 1 | 1 |
Leishmania major | beta tubulin | 0.0176 | 1 | 1 |
Trypanosoma cruzi | beta tubulin, putative | 0.0176 | 1 | 1 |
Leishmania major | beta tubulin | 0.0176 | 1 | 1 |
Trichomonas vaginalis | tubulin, putative | 0.0176 | 1 | 1 |
Entamoeba histolytica | tubulin family protein | 0.0176 | 1 | 1 |
Echinococcus multilocularis | beta tubulin | 0.0176 | 1 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0176 | 1 | 1 |
Leishmania major | beta tubulin | 0.0176 | 1 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0176 | 1 | 1 |
Giardia lamblia | Beta tubulin | 0.0176 | 1 | 1 |
Echinococcus multilocularis | tubulin subunit beta | 0.0176 | 1 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0176 | 1 | 1 |
Echinococcus granulosus | tubulin beta 1 chain | 0.0176 | 1 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0176 | 1 | 1 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0176 | 1 | 1 |
Leishmania major | beta tubulin | 0.0176 | 1 | 1 |
Giardia lamblia | Beta tubulin | 0.0176 | 1 | 1 |
Plasmodium falciparum | tubulin beta chain | 0.0176 | 1 | 1 |
Trypanosoma brucei | beta tubulin | 0.0176 | 1 | 1 |
Trypanosoma brucei | beta tubulin | 0.0176 | 1 | 1 |
Leishmania major | beta tubulin | 0.0176 | 1 | 1 |
Toxoplasma gondii | beta-1 tubulin, putative | 0.0176 | 1 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0176 | 1 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0176 | 1 | 1 |
Loa Loa (eye worm) | tubulin beta-4 chain | 0.0176 | 1 | 1 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
Ki (binding) | = 30 nM | Binding affinity for human cloned vasopressin V1a receptor expressed in CHO cells | ChEMBL. | 17234419 |
Ki (binding) | = 30 nM | Binding affinity for human cloned vasopressin V1a receptor expressed in CHO cells | ChEMBL. | 17234419 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.