Species | Target name | Source | Bibliographic reference |
---|---|---|---|
Homo sapiens | transient receptor potential cation channel, subfamily V, member 1 | Starlite/ChEMBL | References |
Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Echinococcus multilocularis | tubulin beta 1 chain | 0.0051 | 1 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0051 | 1 | 1 |
Leishmania major | beta tubulin | 0.0051 | 1 | 1 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.002 | 0.2166 | 0.2166 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.002 | 0.2166 | 0.2166 |
Leishmania major | beta tubulin | 0.0051 | 1 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0051 | 1 | 1 |
Toxoplasma gondii | beta tubulin | 0.0051 | 1 | 1 |
Brugia malayi | Tubulin alpha-2 chain | 0.002 | 0.2166 | 0.2166 |
Brugia malayi | Tubulin alpha-2 chain | 0.002 | 0.2166 | 0.2166 |
Loa Loa (eye worm) | hypothetical protein | 0.002 | 0.2166 | 0.2166 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.002 | 0.2166 | 0.2166 |
Loa Loa (eye worm) | beta-tubulin | 0.0051 | 1 | 1 |
Loa Loa (eye worm) | tubulin alpha-2 chain | 0.002 | 0.2166 | 0.2166 |
Echinococcus granulosus | tubulin beta 1 chain | 0.0051 | 1 | 1 |
Plasmodium falciparum | tubulin beta chain | 0.0051 | 1 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0051 | 1 | 1 |
Leishmania major | beta tubulin | 0.0051 | 1 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0051 | 1 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.002 | 0.2166 | 0.2166 |
Giardia lamblia | Beta tubulin | 0.0051 | 1 | 1 |
Trypanosoma brucei | beta tubulin | 0.0051 | 1 | 1 |
Plasmodium vivax | tubulin beta chain, putative | 0.0051 | 1 | 1 |
Leishmania major | beta tubulin | 0.0051 | 1 | 1 |
Brugia malayi | Tubulin alpha chain | 0.002 | 0.2166 | 0.2166 |
Loa Loa (eye worm) | alpha-tubulin | 0.002 | 0.2166 | 0.2166 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0051 | 1 | 1 |
Echinococcus multilocularis | tubulin, beta 4A class IVa | 0.0051 | 1 | 1 |
Loa Loa (eye worm) | tubulin alpha chain | 0.002 | 0.2166 | 0.2166 |
Loa Loa (eye worm) | tubulin beta-2A chain | 0.0051 | 1 | 1 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.002 | 0.2166 | 0.2166 |
Trypanosoma brucei | alpha tubulin | 0.002 | 0.2166 | 0.2166 |
Leishmania major | beta tubulin | 0.0051 | 1 | 1 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0051 | 1 | 1 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.002 | 0.2166 | 0.2166 |
Loa Loa (eye worm) | alpha-tubulin | 0.002 | 0.2166 | 0.2166 |
Leishmania major | beta tubulin | 0.0051 | 1 | 1 |
Loa Loa (eye worm) | tubulin beta chain | 0.0051 | 1 | 1 |
Brugia malayi | alpha-tubulin | 0.002 | 0.2166 | 0.2166 |
Leishmania major | beta tubulin | 0.0051 | 1 | 1 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0051 | 1 | 1 |
Leishmania major | beta tubulin | 0.0051 | 1 | 1 |
Echinococcus granulosus | tubulin subunit beta | 0.0051 | 1 | 1 |
Trypanosoma brucei | alpha tubulin | 0.002 | 0.2166 | 0.2166 |
Loa Loa (eye worm) | tubulin gamma chain | 0.002 | 0.2166 | 0.2166 |
Schistosoma mansoni | tubulin subunit beta | 0.0051 | 1 | 1 |
Echinococcus multilocularis | beta tubulin | 0.0051 | 1 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0051 | 1 | 1 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0051 | 1 | 1 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.002 | 0.2166 | 0.2166 |
Trypanosoma brucei | epsilon tubulin | 0.002 | 0.2166 | 0.2166 |
Giardia lamblia | Beta tubulin | 0.0051 | 1 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0051 | 1 | 1 |
Leishmania major | beta tubulin | 0.0051 | 1 | 1 |
Trichomonas vaginalis | tubulin, putative | 0.0051 | 1 | 1 |
Leishmania major | beta tubulin | 0.0051 | 1 | 1 |
Leishmania major | beta tubulin | 0.0051 | 1 | 1 |
Brugia malayi | Tubulin gamma chain | 0.002 | 0.2166 | 0.2166 |
Trypanosoma brucei | alpha tubulin | 0.002 | 0.2166 | 0.2166 |
Leishmania major | beta tubulin | 0.0051 | 1 | 1 |
Leishmania major | beta tubulin | 0.0051 | 1 | 1 |
Entamoeba histolytica | tubulin family protein | 0.0051 | 1 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0051 | 1 | 1 |
Leishmania major | beta tubulin | 0.0051 | 1 | 1 |
Echinococcus granulosus | beta tubulin | 0.0051 | 1 | 1 |
Brugia malayi | tubulin alpha chain - mouse | 0.002 | 0.2166 | 0.2166 |
Schistosoma mansoni | tubulin subunit beta | 0.0051 | 1 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.002 | 0.2166 | 0.2166 |
Leishmania major | beta tubulin | 0.0051 | 1 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.002 | 0.2166 | 0.2166 |
Toxoplasma gondii | beta-1 tubulin, putative | 0.0051 | 1 | 1 |
Echinococcus multilocularis | tubulin subunit beta | 0.0051 | 1 | 1 |
Trypanosoma brucei | epsilon tubulin | 0.002 | 0.2166 | 0.2166 |
Brugia malayi | tubulin alpha-2 chain | 0.002 | 0.2166 | 0.2166 |
Echinococcus granulosus | beta tubulin | 0.0051 | 1 | 1 |
Echinococcus multilocularis | beta tubulin | 0.0051 | 1 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0051 | 1 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.002 | 0.2166 | 0.2166 |
Onchocerca volvulus | 0.0011 | 0 | 0.5 | |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0051 | 1 | 1 |
Echinococcus granulosus | tubulin beta 4A class IVa | 0.0051 | 1 | 1 |
Entamoeba histolytica | tubulin family protein | 0.0051 | 1 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0051 | 1 | 1 |
Loa Loa (eye worm) | tubulin beta-4 chain | 0.0051 | 1 | 1 |
Loa Loa (eye worm) | BEN-1 protein | 0.0051 | 1 | 1 |
Leishmania major | beta tubulin | 0.0051 | 1 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0051 | 1 | 1 |
Trypanosoma brucei | tubulin gamma chain | 0.002 | 0.2166 | 0.2166 |
Leishmania major | beta tubulin | 0.0051 | 1 | 1 |
Trypanosoma brucei | alpha tubulin | 0.002 | 0.2166 | 0.2166 |
Trypanosoma brucei | beta tubulin | 0.0051 | 1 | 1 |
Trypanosoma brucei | beta tubulin | 0.0051 | 1 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0051 | 1 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0051 | 1 | 1 |
Loa Loa (eye worm) | BEN-1 protein | 0.0051 | 1 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.002 | 0.2166 | 0.2166 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0051 | 1 | 1 |
Trypanosoma brucei | epsilon tubulin | 0.002 | 0.2166 | 0.2166 |
Loa Loa (eye worm) | tubulin alpha chain | 0.002 | 0.2166 | 0.2166 |
Toxoplasma gondii | beta-tubulin, putative | 0.0051 | 1 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0051 | 1 | 1 |
Giardia lamblia | Beta tubulin | 0.0051 | 1 | 1 |
Brugia malayi | beta-tubulin, identical | 0.0051 | 1 | 1 |
Trypanosoma cruzi | beta tubulin, putative | 0.0051 | 1 | 1 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.002 | 0.2166 | 0.2166 |
Trypanosoma brucei | beta tubulin | 0.002 | 0.2166 | 0.2166 |
Leishmania major | beta tubulin | 0.0051 | 1 | 1 |
Loa Loa (eye worm) | tubulin beta-1 chain | 0.0051 | 1 | 1 |
Trypanosoma brucei | beta tubulin | 0.0051 | 1 | 1 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
EC50 (functional) | = 15.2 nM | Agonist activity at human recombinant TRPV1 expressed in human HEK293 cells | ChEMBL. | 17046253 |
EC50 (functional) | = 15.2 nM | Agonist activity at human recombinant TRPV1 expressed in human HEK293 cells | ChEMBL. | 17046253 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.