Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Trichomonas vaginalis | fructose-bisphosphate aldolase, putative | 0.0282 | 0.3766 | 0.481 |
Trichomonas vaginalis | fructose-bisphosphate aldolase, putative | 0.0282 | 0.3766 | 0.481 |
Plasmodium falciparum | histone deacetylase, putative | 0.0634 | 0.9315 | 1 |
Loa Loa (eye worm) | histone deacetylase 3 | 0.054 | 0.7829 | 0.8405 |
Brugia malayi | Histone deacetylase family protein | 0.0634 | 0.9315 | 1 |
Trypanosoma brucei | histone deacetylase 1 | 0.054 | 0.7829 | 0.8405 |
Trypanosoma cruzi | histone deacetylase 1, putative | 0.054 | 0.7829 | 0.8405 |
Trichomonas vaginalis | fructose-bisphosphate aldolase, putative | 0.0282 | 0.3766 | 0.481 |
Toxoplasma gondii | histone deacetylase HDAC2 | 0.054 | 0.7829 | 0.8405 |
Trichomonas vaginalis | fructose-bisphosphate aldolase, putative | 0.0282 | 0.3766 | 0.481 |
Giardia lamblia | Histone deacetylase | 0.054 | 0.7829 | 1 |
Plasmodium falciparum | fructose-bisphosphate aldolase | 0.0263 | 0.3465 | 0.372 |
Trichomonas vaginalis | fructose-bisphosphate aldolase, putative | 0.0282 | 0.3766 | 0.481 |
Toxoplasma gondii | histone deacetylase HDAC1 | 0.0634 | 0.9315 | 1 |
Loa Loa (eye worm) | fructose-bisphosphate aldolase 1 | 0.0263 | 0.3465 | 0.372 |
Trichomonas vaginalis | histone deacetylase, putative | 0.054 | 0.7829 | 1 |
Echinococcus multilocularis | fructose 1,6 bisphosphate aldolase | 0.0263 | 0.3465 | 0.3465 |
Entamoeba histolytica | histone deacetylase, putative | 0.054 | 0.7829 | 1 |
Entamoeba histolytica | fructose-1,6-bisphosphate aldolase, putative | 0.0282 | 0.3766 | 0.481 |
Echinococcus multilocularis | histone deacetylase 7 | 0.0634 | 0.9315 | 0.9315 |
Loa Loa (eye worm) | hypothetical protein | 0.0267 | 0.3523 | 0.3782 |
Mycobacterium leprae | Probable fructose bisphosphate aldolase Fba | 0.0138 | 0.1489 | 0.5 |
Schistosoma mansoni | histone deacetylase | 0.054 | 0.7829 | 0.7829 |
Brugia malayi | histone deacetylase 11 | 0.0267 | 0.3523 | 0.3782 |
Entamoeba histolytica | fructose-1,6-bisphosphate aldolase, putative | 0.0282 | 0.3766 | 0.481 |
Echinococcus granulosus | fructose 16 bisphosphate aldolase | 0.0263 | 0.3465 | 0.3465 |
Loa Loa (eye worm) | histone deacetylase | 0.0634 | 0.9315 | 1 |
Trypanosoma cruzi | histone deacetylase, putative | 0.0634 | 0.9315 | 1 |
Trypanosoma brucei | histone deacetylase 3 | 0.0634 | 0.9315 | 1 |
Trichomonas vaginalis | histone deacetylase, putative | 0.054 | 0.7829 | 1 |
Toxoplasma gondii | histone deacetylase HDAC5 | 0.0267 | 0.3523 | 0.3782 |
Trichomonas vaginalis | fructose-bisphosphate aldolase, putative | 0.0282 | 0.3766 | 0.481 |
Treponema pallidum | fructose-bisphosphate aldolase | 0.0282 | 0.3766 | 0.5 |
Schistosoma mansoni | histone deacetylase 4 5 | 0.0634 | 0.9315 | 0.9315 |
Echinococcus granulosus | fructose 16 bisphosphate aldolase | 0.0263 | 0.3465 | 0.3465 |
Trichomonas vaginalis | histone deacetylase 1, 2 ,3, putative | 0.054 | 0.7829 | 1 |
Trichomonas vaginalis | histone deacetylase 1, 2 ,3, putative | 0.054 | 0.7829 | 1 |
Trichomonas vaginalis | histone deacetylase, putative | 0.054 | 0.7829 | 1 |
Loa Loa (eye worm) | histone deacetylase 11 | 0.0267 | 0.3523 | 0.3782 |
Loa Loa (eye worm) | histone deacetylase 1 | 0.054 | 0.7829 | 0.8405 |
Trypanosoma cruzi | fructose-bisphosphate aldolase, glycosomal, putative | 0.0263 | 0.3465 | 0.372 |
Mycobacterium tuberculosis | Probable fructose-bisphosphate aldolase Fba | 0.0138 | 0.1489 | 0.5 |
Echinococcus multilocularis | fructose 1,6 bisphosphate aldolase | 0.0263 | 0.3465 | 0.3465 |
Echinococcus multilocularis | histone deacetylase 1 | 0.054 | 0.7829 | 0.7829 |
Brugia malayi | Histone deacetylase 1 | 0.054 | 0.7829 | 0.8405 |
Loa Loa (eye worm) | hypothetical protein | 0.0367 | 0.5107 | 0.5482 |
Echinococcus granulosus | fructose 16 bisphosphate aldolase | 0.0263 | 0.3465 | 0.3465 |
Leishmania major | histone deacetylase, putative | 0.054 | 0.7829 | 0.8405 |
Echinococcus multilocularis | histone deacetylase 8 | 0.0267 | 0.3523 | 0.3523 |
Trypanosoma brucei | histone deacetylase, putative | 0.0634 | 0.9315 | 1 |
Echinococcus granulosus | histone deacetylase 6 | 0.0634 | 0.9315 | 0.9315 |
Echinococcus multilocularis | fructose bisphosphate aldolase class I | 0.0263 | 0.3465 | 0.3465 |
Trypanosoma cruzi | fructose-bisphosphate aldolase, glycosomal, putative | 0.0263 | 0.3465 | 0.372 |
Trichomonas vaginalis | fructose-bisphosphate aldolase, putative | 0.0282 | 0.3766 | 0.481 |
Trypanosoma cruzi | histone deacetylase, putative | 0.0267 | 0.3523 | 0.3782 |
Echinococcus multilocularis | histone deacetylase 6 | 0.0634 | 0.9315 | 0.9315 |
Toxoplasma gondii | fructose-bisphosphate aldolase, putative | 0.0263 | 0.3465 | 0.372 |
Trypanosoma cruzi | histone deacetylase, putative | 0.0267 | 0.3523 | 0.3782 |
Trichomonas vaginalis | histone deacetylase 1, 2 ,3, putative | 0.054 | 0.7829 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.054 | 0.7829 | 0.8405 |
Echinococcus granulosus | histone deacetylase 6 | 0.0634 | 0.9315 | 0.9315 |
Trypanosoma brucei | fructose-bisphosphate aldolase, glycosomal, putative | 0.0263 | 0.3465 | 0.372 |
Echinococcus multilocularis | histone deacetylase | 0.0634 | 0.9315 | 0.9315 |
Schistosoma mansoni | fructose 16-bisphosphate aldolase | 0.0263 | 0.3465 | 0.3465 |
Brugia malayi | histone deacetylase 3 (HD3) | 0.054 | 0.7829 | 0.8405 |
Echinococcus multilocularis | histone deacetylase 3 | 0.054 | 0.7829 | 0.7829 |
Echinococcus granulosus | histone deacetylase 1 | 0.054 | 0.7829 | 0.7829 |
Toxoplasma gondii | histone deacetylase HDAC4 | 0.0267 | 0.3523 | 0.3782 |
Loa Loa (eye worm) | hypothetical protein | 0.0411 | 0.5792 | 0.6218 |
Trypanosoma cruzi | fructose-bisphosphate aldolase, glycosomal, putative | 0.0263 | 0.3465 | 0.372 |
Leishmania major | fructose-1,6-bisphosphate aldolase | 0.0263 | 0.3465 | 0.372 |
Schistosoma mansoni | histone deacetylase 4 5 | 0.0634 | 0.9315 | 0.9315 |
Echinococcus granulosus | histone deacetylase 7 | 0.0634 | 0.9315 | 0.9315 |
Trichomonas vaginalis | histone deacetylase, putative | 0.054 | 0.7829 | 1 |
Schistosoma mansoni | histone deacetylase 1 2 3 | 0.0267 | 0.3523 | 0.3523 |
Trichomonas vaginalis | histone deacetylase, putative | 0.054 | 0.7829 | 1 |
Trypanosoma cruzi | fructose-bisphosphate aldolase, glycosomal, putative | 0.0263 | 0.3465 | 0.372 |
Plasmodium vivax | fructose 1,6-bisphosphate aldolase, putative | 0.0263 | 0.3465 | 0.372 |
Toxoplasma gondii | histone deacetylase HDAC3 | 0.054 | 0.7829 | 0.8405 |
Schistosoma mansoni | histone deacetylase hda2 | 0.0267 | 0.3523 | 0.3523 |
Plasmodium vivax | histone deacetylase 2, putative | 0.0634 | 0.9315 | 1 |
Schistosoma mansoni | histone deacetylase hda2 | 0.0678 | 1 | 1 |
Brugia malayi | fructose-bisphosphate aldolase 2 | 0.0263 | 0.3465 | 0.372 |
Trypanosoma cruzi | histone deacetylase, putative | 0.0634 | 0.9315 | 1 |
Schistosoma mansoni | fructose 16-bisphosphate aldolase | 0.0263 | 0.3465 | 0.3465 |
Echinococcus multilocularis | fructose 1,6 bisphosphate aldolase | 0.0263 | 0.3465 | 0.3465 |
Trichomonas vaginalis | fructose-bisphosphate aldolase, putative | 0.0282 | 0.3766 | 0.481 |
Leishmania major | histone deacetylase, putative | 0.0634 | 0.9315 | 1 |
Echinococcus granulosus | fructose bisphosphate aldolase class I | 0.0263 | 0.3465 | 0.3465 |
Trypanosoma brucei | histone deacetylase 4 | 0.0634 | 0.9315 | 1 |
Echinococcus granulosus | histone deacetylase 8 | 0.0267 | 0.3523 | 0.3523 |
Trichomonas vaginalis | histone deacetylase, putative | 0.054 | 0.7829 | 1 |
Echinococcus granulosus | histone deacetylase | 0.0634 | 0.9315 | 0.9315 |
Plasmodium falciparum | histone deacetylase 2 | 0.0634 | 0.9315 | 1 |
Trypanosoma cruzi | histone deacetylase 1, putative | 0.054 | 0.7829 | 0.8405 |
Trypanosoma brucei | histone deacetylase 2 | 0.0267 | 0.3523 | 0.3782 |
Echinococcus granulosus | histone deacetylase 3 | 0.054 | 0.7829 | 0.7829 |
Trypanosoma cruzi | histone deacetylase, putative | 0.0634 | 0.9315 | 1 |
Toxoplasma gondii | fructose-1,6-bisphosphate aldolase | 0.0263 | 0.3465 | 0.372 |
Toxoplasma gondii | fructose-1,6-bisphosphate aldolase | 0.0263 | 0.3465 | 0.372 |
Echinococcus multilocularis | histone deacetylase 6 | 0.0678 | 1 | 1 |
Leishmania major | histone deacetylase, putative | 0.054 | 0.7829 | 0.8405 |
Giardia lamblia | Fructose-bisphosphate aldolase | 0.0282 | 0.3766 | 0.481 |
Plasmodium vivax | histone deacetylase, putative | 0.0634 | 0.9315 | 1 |
Mycobacterium ulcerans | fructose-bisphosphate aldolase | 0.0138 | 0.1489 | 0.5 |
Echinococcus multilocularis | histone deacetylase 6 | 0.0634 | 0.9315 | 0.9315 |
Leishmania major | histone deacetylase, putative | 0.0634 | 0.9315 | 1 |
Plasmodium vivax | histone deacetylase 1, putative | 0.054 | 0.7829 | 0.8405 |
Brugia malayi | fructose-bisphosphate aldolase 1 | 0.0263 | 0.3465 | 0.372 |
Brugia malayi | Histone deacetylase family protein | 0.0634 | 0.9315 | 1 |
Schistosoma mansoni | histone deacetylase | 0.054 | 0.7829 | 0.7829 |
Plasmodium vivax | histone deacetylase, putative | 0.0267 | 0.3523 | 0.3782 |
Onchocerca volvulus | Histone deacetylase 10 homolog | 0.0267 | 0.3523 | 1 |
Brugia malayi | histone deacetylase 1 (HD1) | 0.054 | 0.7829 | 0.8405 |
Plasmodium falciparum | histone deacetylase 1 | 0.054 | 0.7829 | 0.8405 |
Loa Loa (eye worm) | fructose-bisphosphate aldolase 2 | 0.0263 | 0.3465 | 0.372 |
Loa Loa (eye worm) | histone deacetylase 7A | 0.0634 | 0.9315 | 1 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
Activity (functional) | < 50 % | Agonist activity at human cloned GPR109a receptor up to 30 uM by forskolin-stimulated cAMP production test | ChEMBL. | 17588745 |
Activity (functional) | < 50 % | Agonist activity at human cloned GPR109a receptor up to 30 uM by forskolin-stimulated cAMP production test | ChEMBL. | 17588745 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.