Species | Target name | Source | Bibliographic reference |
---|---|---|---|
Homo sapiens | sodium channel, voltage-gated, type IX, alpha subunit | Starlite/ChEMBL | References |
Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Mycobacterium leprae | PROBABLE OXIDOREDUCTASE | 0.0032 | 0.4802 | 1 |
Brugia malayi | oxidoreductase, aldo/keto reductase family protein | 0.0032 | 0.4802 | 0.7688 |
Leishmania major | DNA polymerase kappa, putative | 0.0025 | 0.2481 | 0.2773 |
Mycobacterium ulcerans | DNA polymerase IV | 0.0049 | 1 | 1 |
Trypanosoma brucei | DNA polymerase kappa, putative | 0.0037 | 0.6246 | 0.6246 |
Echinococcus granulosus | aldo keto reductase family 1 member B4 | 0.0032 | 0.4802 | 0.4802 |
Echinococcus multilocularis | aldo keto reductase family 1, member B4 | 0.0032 | 0.4802 | 0.4802 |
Schistosoma mansoni | aldo-keto reductase | 0.0032 | 0.4802 | 1 |
Echinococcus granulosus | hypothetical protein | 0.0032 | 0.4802 | 0.4802 |
Trypanosoma brucei | DNA polymerase kappa, putative | 0.0049 | 1 | 1 |
Echinococcus granulosus | aldo keto reductase | 0.0032 | 0.4802 | 0.4802 |
Onchocerca volvulus | 0.0032 | 0.4802 | 0.5 | |
Echinococcus multilocularis | aldo keto reductase | 0.0032 | 0.4802 | 0.4802 |
Trypanosoma brucei | DNA polymerase kappa, putative | 0.0049 | 1 | 1 |
Giardia lamblia | Aldose reductase | 0.0032 | 0.4802 | 1 |
Trypanosoma brucei | DNA polymerase kappa, putative | 0.0037 | 0.6246 | 0.6246 |
Echinococcus granulosus | aldo keto reductase | 0.0032 | 0.4802 | 0.4802 |
Trypanosoma cruzi | DNA polymerase kappa, putative | 0.0049 | 1 | 1 |
Loa Loa (eye worm) | oxidoreductase | 0.0032 | 0.4802 | 0.7688 |
Brugia malayi | oxidoreductase, aldo/keto reductase family protein | 0.0032 | 0.4802 | 0.7688 |
Trypanosoma brucei | unspecified product | 0.0041 | 0.7519 | 0.7519 |
Trypanosoma brucei | DNA polymerase kappa, putative | 0.002 | 0.0792 | 0.0792 |
Echinococcus multilocularis | aldo keto reductase family 1, member B4 | 0.0032 | 0.4802 | 0.4802 |
Echinococcus multilocularis | aldo keto reductase family 1, member B4 | 0.0032 | 0.4802 | 0.4802 |
Echinococcus multilocularis | aldo keto reductase family 1, member B4 | 0.0032 | 0.4802 | 0.4802 |
Trypanosoma brucei | DNA polymerase kappa, putative | 0.0049 | 1 | 1 |
Onchocerca volvulus | 0.0032 | 0.4802 | 0.5 | |
Loa Loa (eye worm) | oxidoreductase | 0.0032 | 0.4802 | 0.7688 |
Leishmania major | DNA polymerase kappa, putative,DNA polymerase IV, putative | 0.0025 | 0.2481 | 0.2773 |
Echinococcus granulosus | aldo keto reductase family 1 member B4 | 0.0032 | 0.4802 | 0.4802 |
Echinococcus granulosus | aldo keto reductase family 1 member B4 | 0.0032 | 0.4802 | 0.4802 |
Echinococcus granulosus | aldo keto reductase family 1 member B4 | 0.0032 | 0.4802 | 0.4802 |
Loa Loa (eye worm) | oxidoreductase | 0.0032 | 0.4802 | 0.7688 |
Echinococcus multilocularis | dna polymerase kappa | 0.0049 | 1 | 1 |
Echinococcus multilocularis | aldo keto reductase family 1, member B4 | 0.0032 | 0.4802 | 0.4802 |
Echinococcus granulosus | aldo keto reductase family 1 member B4 | 0.0032 | 0.4802 | 0.4802 |
Trypanosoma cruzi | DNA polymerase kappa, putative | 0.0049 | 1 | 1 |
Trypanosoma brucei | DNA polymerase IV, putative | 0.0049 | 1 | 1 |
Leishmania major | aldo-keto reductase-like protein | 0.0032 | 0.4802 | 0.5367 |
Loa Loa (eye worm) | hypothetical protein | 0.0037 | 0.6246 | 1 |
Loa Loa (eye worm) | oxidoreductase | 0.0032 | 0.4802 | 0.7688 |
Loa Loa (eye worm) | oxidoreductase | 0.0032 | 0.4802 | 0.7688 |
Mycobacterium tuberculosis | Probable oxidoreductase | 0.0032 | 0.4802 | 1 |
Echinococcus granulosus | aldehyde reductase | 0.0023 | 0.1835 | 0.1835 |
Toxoplasma gondii | aldose reductase, putative | 0.0032 | 0.4802 | 0.5 |
Onchocerca volvulus | 0.0032 | 0.4802 | 0.5 | |
Trypanosoma cruzi | aldo/keto reductase, putative | 0.0032 | 0.4802 | 0.4802 |
Brugia malayi | polk-prov protein | 0.0037 | 0.6246 | 1 |
Trypanosoma brucei | DNA polymerase kappa, putative | 0.0049 | 1 | 1 |
Trypanosoma brucei | DNA polymerase kappa, putative | 0.002 | 0.0792 | 0.0792 |
Echinococcus multilocularis | aldo keto reductase | 0.0032 | 0.4802 | 0.4802 |
Brugia malayi | oxidoreductase, aldo/keto reductase family protein | 0.0032 | 0.4802 | 0.7688 |
Echinococcus granulosus | aldo keto reductase family 1 member B4 | 0.0032 | 0.4802 | 0.4802 |
Entamoeba histolytica | aldose reductase, putative | 0.0032 | 0.4802 | 1 |
Trypanosoma brucei | aldo-keto reductase, putative | 0.0032 | 0.4802 | 0.4802 |
Trypanosoma brucei | DNA polymerase kappa, putative | 0.0049 | 1 | 1 |
Echinococcus granulosus | aldo keto reductase family 1 member B4 | 0.0032 | 0.4802 | 0.4802 |
Echinococcus multilocularis | aldo keto reductase family 1, member B4 | 0.0032 | 0.4802 | 0.4802 |
Echinococcus granulosus | voltage gated sodium channel Nav1 alpha subunit | 0.0045 | 0.8947 | 0.8947 |
Echinococcus multilocularis | aldo keto reductase family 1, member B4 | 0.0032 | 0.4802 | 0.4802 |
Mycobacterium tuberculosis | Possible DNA-damage-inducible protein P DinP (DNA polymerase V) (pol IV 2) (DNA nucleotidyltransferase (DNA-directed)) | 0.0025 | 0.2481 | 0.5166 |
Echinococcus multilocularis | aldo keto reductase | 0.0032 | 0.4802 | 0.4802 |
Entamoeba histolytica | aldose reductase, putative | 0.0032 | 0.4802 | 1 |
Leishmania major | aldehyde reductase, putative,oxidoreductase, putative | 0.0032 | 0.4802 | 0.5367 |
Schistosoma mansoni | pol-related | 0.0032 | 0.4802 | 1 |
Echinococcus multilocularis | aldo keto reductase family 1, member B4 | 0.0032 | 0.4802 | 0.4802 |
Mycobacterium ulcerans | DNA polymerase IV | 0.0049 | 1 | 1 |
Echinococcus multilocularis | aldehyde reductase | 0.0023 | 0.1835 | 0.1835 |
Trichomonas vaginalis | DNA polymerase eta, putative | 0.0049 | 1 | 1 |
Trypanosoma brucei | DNA polymerase IV, putative | 0.0049 | 1 | 1 |
Onchocerca volvulus | 0.0032 | 0.4802 | 0.5 | |
Trypanosoma brucei | DNA polymerase kappa, putative | 0.0025 | 0.2481 | 0.2481 |
Echinococcus granulosus | aldo keto reductase family 1 member B4 | 0.0032 | 0.4802 | 0.4802 |
Brugia malayi | oxidoreductase, aldo/keto reductase family protein | 0.0032 | 0.4802 | 0.7688 |
Trichomonas vaginalis | DNA polymerase IV / kappa, putative | 0.0049 | 1 | 1 |
Trypanosoma cruzi | aldo-keto reductase | 0.0032 | 0.4802 | 0.4802 |
Echinococcus multilocularis | aldo keto reductase family 1, member B4 | 0.0032 | 0.4802 | 0.4802 |
Loa Loa (eye worm) | hypothetical protein | 0.0032 | 0.4802 | 0.7688 |
Echinococcus granulosus | aldo keto reductase | 0.0032 | 0.4802 | 0.4802 |
Leishmania major | prostaglandin f synthase, putative | 0.0032 | 0.4802 | 0.5367 |
Leishmania major | calcium channel protein, putative,ion transporter, putative | 0.0045 | 0.8947 | 1 |
Trypanosoma cruzi | DNA polymerase kappa, putative | 0.0049 | 1 | 1 |
Giardia lamblia | Aldose reductase | 0.0032 | 0.4802 | 1 |
Echinococcus granulosus | sodium channel protein | 0.0045 | 0.8947 | 0.8947 |
Entamoeba histolytica | aldose reductase, putative | 0.0032 | 0.4802 | 1 |
Trypanosoma brucei | prostaglandin f synthase | 0.0032 | 0.4802 | 0.4802 |
Onchocerca volvulus | 0.0032 | 0.4802 | 0.5 | |
Leishmania major | prostaglandin f2-alpha synthase/D-arabinose dehydrogenase | 0.0032 | 0.4802 | 0.5367 |
Trypanosoma brucei | DNA polymerase kappa, putative | 0.002 | 0.0792 | 0.0792 |
Echinococcus multilocularis | aldo keto reductase | 0.0032 | 0.4802 | 0.4802 |
Echinococcus multilocularis | aldo keto reductase family 1, member B4 | 0.0032 | 0.4802 | 0.4802 |
Trypanosoma brucei | DNA polymerase kappa, putative | 0.0049 | 1 | 1 |
Echinococcus granulosus | aldo keto reductase family 1 member B4 | 0.0032 | 0.4802 | 0.4802 |
Onchocerca volvulus | 0.0032 | 0.4802 | 0.5 | |
Trypanosoma brucei | DNA polymerase kappa, putative | 0.0049 | 1 | 1 |
Echinococcus multilocularis | aldo keto reductase family 1, member B4 | 0.0032 | 0.4802 | 0.4802 |
Schistosoma mansoni | aldo-keto reductase | 0.0032 | 0.4802 | 1 |
Trypanosoma brucei | DNA polymerase kappa, putative | 0.0049 | 1 | 1 |
Trypanosoma brucei | DNA polymerase kappa, putative | 0.0049 | 1 | 1 |
Echinococcus multilocularis | sodium channel protein | 0.0045 | 0.8947 | 0.8947 |
Trypanosoma cruzi | DNA polymerase kappa, putative | 0.0049 | 1 | 1 |
Trypanosoma brucei | DNA polymerase IV, putative | 0.0041 | 0.7519 | 0.7519 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.