Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Onchocerca volvulus | 0.0061 | 0.4861 | 0.5 | |
Giardia lamblia | Aldose reductase | 0.0061 | 0.4861 | 1 |
Toxoplasma gondii | lactate dehydrogenase LDH2 | 0.009 | 1 | 1 |
Trichomonas vaginalis | aldo-keto reductase, putative | 0.0061 | 0.4861 | 1 |
Plasmodium falciparum | L-lactate dehydrogenase | 0.009 | 1 | 1 |
Entamoeba histolytica | aldose reductase, putative | 0.0061 | 0.4861 | 0.4861 |
Entamoeba histolytica | malate dehydrogenase, putative | 0.009 | 1 | 1 |
Echinococcus multilocularis | aldehyde reductase | 0.0044 | 0.1611 | 0.1611 |
Wolbachia endosymbiont of Brugia malayi | malate dehydrogenase | 0.009 | 1 | 0.5 |
Trichomonas vaginalis | dihydrodiol dehydrogenase, putative | 0.0061 | 0.4861 | 1 |
Echinococcus multilocularis | aldo keto reductase family 1, member B4 | 0.0061 | 0.4861 | 0.4861 |
Loa Loa (eye worm) | oxidoreductase | 0.0061 | 0.4861 | 0.4861 |
Echinococcus multilocularis | aldo keto reductase | 0.0061 | 0.4861 | 0.4861 |
Giardia lamblia | Aldose reductase | 0.0061 | 0.4861 | 1 |
Trypanosoma brucei | prostaglandin f synthase | 0.0061 | 0.4861 | 1 |
Echinococcus multilocularis | aldo keto reductase family 1, member B4 | 0.0061 | 0.4861 | 0.4861 |
Trichomonas vaginalis | aldo-keto reductase, putative | 0.0061 | 0.4861 | 1 |
Trichomonas vaginalis | aldo-keto reductase, putative | 0.0061 | 0.4861 | 1 |
Trichomonas vaginalis | dihydrodiol dehydrogenase, putative | 0.0061 | 0.4861 | 1 |
Echinococcus multilocularis | lactate dehydrogenase a | 0.009 | 1 | 1 |
Echinococcus granulosus | lactate dehydrogenase a | 0.009 | 1 | 1 |
Mycobacterium ulcerans | oxidoreductase | 0.0061 | 0.4861 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0061 | 0.4861 | 0.4861 |
Trichomonas vaginalis | aldo-keto reductase, putative | 0.0061 | 0.4861 | 1 |
Toxoplasma gondii | lactate dehydrogenase LDH1 | 0.009 | 1 | 1 |
Echinococcus multilocularis | aldo keto reductase family 1, member B4 | 0.0061 | 0.4861 | 0.4861 |
Echinococcus granulosus | aldehyde reductase | 0.0044 | 0.1611 | 0.1611 |
Echinococcus granulosus | lactate dehydrogenase protein | 0.009 | 1 | 1 |
Trypanosoma cruzi | aldo/keto reductase, putative | 0.0061 | 0.4861 | 1 |
Echinococcus multilocularis | aldo keto reductase family 1, member B4 | 0.0061 | 0.4861 | 0.4861 |
Brugia malayi | oxidoreductase, aldo/keto reductase family protein | 0.0061 | 0.4861 | 0.4861 |
Plasmodium falciparum | malate dehydrogenase | 0.009 | 1 | 1 |
Echinococcus granulosus | aldo keto reductase | 0.0061 | 0.4861 | 0.4861 |
Echinococcus multilocularis | aldo keto reductase family 1, member B4 | 0.0061 | 0.4861 | 0.4861 |
Echinococcus granulosus | L lactate dehydrogenase | 0.0055 | 0.3641 | 0.3641 |
Echinococcus granulosus | aldo keto reductase family 1 member B4 | 0.0061 | 0.4861 | 0.4861 |
Schistosoma mansoni | aldo-keto reductase | 0.0061 | 0.4861 | 0.4861 |
Loa Loa (eye worm) | hypothetical protein | 0.009 | 1 | 1 |
Trichomonas vaginalis | aldo-keto reductase, putative | 0.0061 | 0.4861 | 1 |
Trichomonas vaginalis | aldo-keto reductase, putative | 0.0061 | 0.4861 | 1 |
Echinococcus granulosus | aldo keto reductase family 1 member B4 | 0.0061 | 0.4861 | 0.4861 |
Trichomonas vaginalis | aldo-keto reductase, putative | 0.0061 | 0.4861 | 1 |
Echinococcus multilocularis | aldo keto reductase family 1, member B4 | 0.0061 | 0.4861 | 0.4861 |
Schistosoma mansoni | L-lactate dehydrogenase | 0.009 | 1 | 1 |
Leishmania major | malate dehydrogenase, putative | 0.009 | 1 | 1 |
Echinococcus multilocularis | aldo keto reductase family 1, member B4 | 0.0061 | 0.4861 | 0.4861 |
Trichomonas vaginalis | aldo-keto reductase, putative | 0.0061 | 0.4861 | 1 |
Trichomonas vaginalis | aldo-keto reductase, putative | 0.0061 | 0.4861 | 1 |
Mycobacterium leprae | Conserved hypothetical protein | 0.0044 | 0.1611 | 0.3314 |
Onchocerca volvulus | 0.0061 | 0.4861 | 0.5 | |
Echinococcus granulosus | aldo keto reductase family 1 member B4 | 0.0061 | 0.4861 | 0.4861 |
Toxoplasma gondii | malate dehydrogenase MDH | 0.009 | 1 | 1 |
Loa Loa (eye worm) | oxidoreductase | 0.0061 | 0.4861 | 0.4861 |
Trypanosoma brucei | aldo-keto reductase, putative | 0.0061 | 0.4861 | 1 |
Loa Loa (eye worm) | oxidoreductase | 0.0061 | 0.4861 | 0.4861 |
Trichomonas vaginalis | aldo-keto reductase, putative | 0.0061 | 0.4861 | 1 |
Brugia malayi | oxidoreductase, aldo/keto reductase family protein | 0.0061 | 0.4861 | 0.4861 |
Brugia malayi | oxidoreductase, aldo/keto reductase family protein | 0.0061 | 0.4861 | 0.4861 |
Chlamydia trachomatis | malate dehydrogenase | 0.0035 | 0 | 0.5 |
Trichomonas vaginalis | dihydrodiol dehydrogenase, putative | 0.0061 | 0.4861 | 1 |
Leishmania major | prostaglandin f2-alpha synthase/D-arabinose dehydrogenase | 0.0061 | 0.4861 | 0.4861 |
Schistosoma mansoni | malate dehydrogenase | 0.009 | 1 | 1 |
Leishmania major | aldehyde reductase, putative,oxidoreductase, putative | 0.0061 | 0.4861 | 0.4861 |
Leishmania major | aldo-keto reductase-like protein | 0.0061 | 0.4861 | 0.4861 |
Plasmodium vivax | lactate dehydrogenase | 0.009 | 1 | 1 |
Echinococcus multilocularis | L lactate dehydrogenase B chain | 0.009 | 1 | 1 |
Leishmania major | prostaglandin f synthase, putative | 0.0061 | 0.4861 | 0.4861 |
Echinococcus multilocularis | aldo keto reductase | 0.0061 | 0.4861 | 0.4861 |
Echinococcus multilocularis | lactate dehydrogenase a | 0.009 | 1 | 1 |
Mycobacterium tuberculosis | Probable oxidoreductase | 0.0061 | 0.4861 | 1 |
Echinococcus granulosus | aldo keto reductase family 1 member B4 | 0.0061 | 0.4861 | 0.4861 |
Echinococcus granulosus | aldo keto reductase family 1 member B4 | 0.0061 | 0.4861 | 0.4861 |
Onchocerca volvulus | 0.0061 | 0.4861 | 0.5 | |
Echinococcus multilocularis | lactate dehydrogenase protein | 0.009 | 1 | 1 |
Schistosoma mansoni | pol-related | 0.0061 | 0.4861 | 0.4861 |
Echinococcus multilocularis | aldo keto reductase family 1, member B4 | 0.0061 | 0.4861 | 0.4861 |
Onchocerca volvulus | 0.0061 | 0.4861 | 0.5 | |
Echinococcus granulosus | hypothetical protein | 0.0061 | 0.4861 | 0.4861 |
Echinococcus granulosus | aldo keto reductase family 1 member B4 | 0.0061 | 0.4861 | 0.4861 |
Echinococcus granulosus | L lactate dehydrogenase B chain | 0.009 | 1 | 1 |
Trichomonas vaginalis | aldo-keto reductase, putative | 0.0061 | 0.4861 | 1 |
Entamoeba histolytica | aldose reductase, putative | 0.0061 | 0.4861 | 0.4861 |
Echinococcus granulosus | aldo keto reductase | 0.0061 | 0.4861 | 0.4861 |
Loa Loa (eye worm) | oxidoreductase | 0.0061 | 0.4861 | 0.4861 |
Mycobacterium leprae | PROBABLE OXIDOREDUCTASE | 0.0061 | 0.4861 | 1 |
Echinococcus granulosus | aldo keto reductase family 1 member B4 | 0.0061 | 0.4861 | 0.4861 |
Echinococcus multilocularis | aldo keto reductase family 1, member B4 | 0.0061 | 0.4861 | 0.4861 |
Onchocerca volvulus | 0.0061 | 0.4861 | 0.5 | |
Echinococcus granulosus | aldo keto reductase family 1 member B4 | 0.0061 | 0.4861 | 0.4861 |
Echinococcus multilocularis | aldo keto reductase | 0.0061 | 0.4861 | 0.4861 |
Loa Loa (eye worm) | oxidoreductase | 0.0061 | 0.4861 | 0.4861 |
Echinococcus multilocularis | lactate dehydrogenase a | 0.009 | 1 | 1 |
Echinococcus granulosus | aldo keto reductase | 0.0061 | 0.4861 | 0.4861 |
Schistosoma mansoni | aldo-keto reductase | 0.0061 | 0.4861 | 0.4861 |
Brugia malayi | oxidoreductase, aldo/keto reductase family protein | 0.0061 | 0.4861 | 0.4861 |
Trichomonas vaginalis | aldo-keto reductase, putative | 0.0061 | 0.4861 | 1 |
Echinococcus multilocularis | L lactate dehydrogenase | 0.0055 | 0.3641 | 0.3641 |
Trichomonas vaginalis | aldo/keto reductase, putative | 0.0061 | 0.4861 | 1 |
Plasmodium vivax | malate dehydrogenase, putative | 0.009 | 1 | 1 |
Echinococcus multilocularis | aldo keto reductase family 1, member B4 | 0.0061 | 0.4861 | 0.4861 |
Onchocerca volvulus | 0.0061 | 0.4861 | 0.5 | |
Echinococcus granulosus | aldo keto reductase family 1 member B4 | 0.0061 | 0.4861 | 0.4861 |
Echinococcus granulosus | lactate dehydrogenase a | 0.009 | 1 | 1 |
Trichomonas vaginalis | aldo/keto reductase, putative | 0.0061 | 0.4861 | 1 |
Entamoeba histolytica | aldose reductase, putative | 0.0061 | 0.4861 | 0.4861 |
Trypanosoma cruzi | aldo-keto reductase | 0.0061 | 0.4861 | 1 |
Echinococcus multilocularis | aldo keto reductase | 0.0061 | 0.4861 | 0.4861 |
Trichomonas vaginalis | aldo/keto reductase, putative | 0.0061 | 0.4861 | 1 |
Echinococcus multilocularis | aldo keto reductase family 1, member B4 | 0.0061 | 0.4861 | 0.4861 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
Inhibition (binding) | = 12 % | Inhibition of human Kv1.5 channel expressed in mouse L929 cells assessed as blockade of ultra rapidly activating potassium current at 1 uM by volatge clamp technique | ChEMBL. | 18374568 |
Inhibition (binding) | = 12 % | Inhibition of human Kv1.5 channel expressed in mouse L929 cells assessed as blockade of ultra rapidly activating potassium current at 1 uM by volatge clamp technique | ChEMBL. | 18374568 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.