Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Loa Loa (eye worm) | hypothetical protein | 0.0051 | 0.028 | 0.0451 |
Brugia malayi | RNA binding protein | 0.047 | 0.6203 | 1 |
Echinococcus multilocularis | beta LACTamase domain containing family member | 0.0035 | 0.006 | 0.006 |
Trypanosoma brucei | phosphatidylinositol 4-kinase, putative | 0.0092 | 0.0863 | 1 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0073 | 0.0597 | 0.6922 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0055 | 0.034 | 0.3945 |
Entamoeba histolytica | phosphatidylinositol3-kinaseTor2, putative | 0.0092 | 0.0863 | 0.5 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0055 | 0.034 | 0.3945 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.006 | 0.0407 | 0.4722 |
Trypanosoma brucei | FAT domain/Rapamycin binding domain/Phosphatidylinositol 3- and 4-kinase, putative | 0.0038 | 0.0104 | 0.1204 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0068 | 0.053 | 0.6145 |
Trypanosoma brucei | hypothetical protein, conserved | 0.0035 | 0.006 | 0.0699 |
Trypanosoma cruzi | Phosphatidylinositol 3-kinase tor1 | 0.0092 | 0.0863 | 1 |
Echinococcus multilocularis | tumor protein p63 | 0.0346 | 0.4452 | 0.4452 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.005 | 0.0265 | 0.3066 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0068 | 0.053 | 0.6145 |
Mycobacterium ulcerans | beta-lactamase | 0.0035 | 0.006 | 0.5 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.005 | 0.0266 | 0.3078 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0092 | 0.0863 | 1 |
Brugia malayi | beta-lactamase family protein | 0.0035 | 0.006 | 0.0097 |
Leishmania major | target of rapamycin (TOR) kinase 1, putative | 0.0092 | 0.0863 | 1 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0068 | 0.053 | 0.6145 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.005 | 0.0266 | 0.3078 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0073 | 0.0597 | 0.6922 |
Loa Loa (eye worm) | hypothetical protein | 0.0035 | 0.006 | 0.0097 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0068 | 0.053 | 0.6145 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0092 | 0.0863 | 1 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0092 | 0.0863 | 1 |
Schistosoma mansoni | tar DNA-binding protein | 0.047 | 0.6203 | 0.6203 |
Trypanosoma cruzi | Phosphatidylinositol 3-kinase tor2 | 0.0092 | 0.0863 | 1 |
Toxoplasma gondii | target of rapamycin (TOR), putative | 0.0068 | 0.053 | 1 |
Brugia malayi | Hypothetical 52.5 kDa protein ZK945.1 in chromosome II, putative | 0.0035 | 0.006 | 0.0097 |
Echinococcus multilocularis | microtubule associated protein 2 | 0.0739 | 1 | 1 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0054 | 0.0333 | 0.3855 |
Trypanosoma cruzi | target of rapamycin kinase 3 | 0.0073 | 0.0598 | 0.6934 |
Schistosoma mansoni | family S12 unassigned peptidase (S12 family) | 0.0035 | 0.006 | 0.006 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0068 | 0.053 | 0.6145 |
Loa Loa (eye worm) | hypothetical protein | 0.0051 | 0.0286 | 0.0461 |
Loa Loa (eye worm) | hypothetical protein | 0.0035 | 0.006 | 0.0097 |
Brugia malayi | RNA recognition motif domain containing protein | 0.047 | 0.6203 | 1 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0068 | 0.053 | 0.6145 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0073 | 0.0597 | 0.6922 |
Loa Loa (eye worm) | beta-lactamase | 0.0035 | 0.006 | 0.0097 |
Trypanosoma cruzi | hypothetical protein, conserved | 0.0035 | 0.006 | 0.0699 |
Loa Loa (eye worm) | RNA binding protein | 0.047 | 0.6203 | 1 |
Loa Loa (eye worm) | RNA recognition domain-containing protein domain-containing protein | 0.047 | 0.6203 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0035 | 0.006 | 0.0097 |
Echinococcus granulosus | FKBP12 rapamycin complex associated protein | 0.0092 | 0.0863 | 0.0863 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0073 | 0.0597 | 0.6922 |
Loa Loa (eye worm) | hypothetical protein | 0.0035 | 0.006 | 0.0097 |
Leishmania major | hypothetical protein, conserved | 0.0035 | 0.006 | 0.0699 |
Echinococcus multilocularis | FKBP12 rapamycin complex associated protein | 0.0092 | 0.0863 | 0.0863 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0055 | 0.034 | 0.3945 |
Trypanosoma brucei | target of rapamycin kinase 3, putative | 0.0073 | 0.0598 | 0.6934 |
Loa Loa (eye worm) | beta-LACTamase domain containing family member | 0.0035 | 0.006 | 0.0097 |
Loa Loa (eye worm) | pigment dispersing factor receptor c | 0.0051 | 0.0286 | 0.0461 |
Loa Loa (eye worm) | MH2 domain-containing protein | 0.0379 | 0.4916 | 0.7925 |
Schistosoma mansoni | tar DNA-binding protein | 0.047 | 0.6203 | 0.6203 |
Trypanosoma brucei | Phosphatidylinositol 3-kinase tor1 | 0.0092 | 0.0863 | 1 |
Echinococcus granulosus | tar DNA binding protein | 0.047 | 0.6203 | 0.6203 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.005 | 0.0266 | 0.3078 |
Mycobacterium ulcerans | esterase/lipase LipP | 0.0035 | 0.006 | 0.5 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.005 | 0.0266 | 0.3078 |
Schistosoma mansoni | microtubule-associated protein tau | 0.0739 | 1 | 1 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0073 | 0.0597 | 0.6922 |
Mycobacterium tuberculosis | Possible penicillin-binding protein | 0.0224 | 0.2731 | 1 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0078 | 0.0673 | 0.78 |
Entamoeba histolytica | FKBP-rapamycin associated protein (FRAP), putative | 0.0092 | 0.0863 | 0.5 |
Brugia malayi | Corticotropin releasing factor receptor 2 precursor, putative | 0.0051 | 0.0286 | 0.0461 |
Brugia malayi | MH2 domain containing protein | 0.0379 | 0.4916 | 0.7925 |
Schistosoma mansoni | ataxia telangiectasia mutated (atm)-related | 0.0092 | 0.0863 | 0.0863 |
Onchocerca volvulus | 0.0051 | 0.028 | 1 | |
Schistosoma mansoni | cellular tumor antigen P53 | 0.0051 | 0.028 | 0.028 |
Loa Loa (eye worm) | transcription factor SMAD2 | 0.0379 | 0.4916 | 0.7925 |
Trichomonas vaginalis | penicillin-binding protein, putative | 0.0035 | 0.006 | 0.0699 |
Brugia malayi | latrophilin 2 splice variant baaae | 0.0035 | 0.0058 | 0.0093 |
Plasmodium vivax | hypothetical protein, conserved | 0.0035 | 0.006 | 0.5 |
Loa Loa (eye worm) | hypothetical protein | 0.0035 | 0.006 | 0.0097 |
Trichomonas vaginalis | D-aminoacylase, putative | 0.0035 | 0.006 | 0.0699 |
Schistosoma mansoni | hypothetical protein | 0.0035 | 0.0058 | 0.0058 |
Mycobacterium leprae | conserved hypothetical protein | 0.0035 | 0.006 | 0.5 |
Loa Loa (eye worm) | hypothetical protein | 0.0035 | 0.006 | 0.0097 |
Loa Loa (eye worm) | hypothetical protein | 0.0035 | 0.0058 | 0.0093 |
Trichomonas vaginalis | D-aminoacylase, putative | 0.0035 | 0.006 | 0.0699 |
Schistosoma mansoni | family S12 unassigned peptidase (S12 family) | 0.0035 | 0.006 | 0.006 |
Brugia malayi | Calcitonin receptor-like protein seb-1 | 0.0051 | 0.0286 | 0.0461 |
Giardia lamblia | GTOR | 0.0092 | 0.0863 | 0.5 |
Leishmania major | target of rapamycin (TOR) kinase 2, putative | 0.0092 | 0.0863 | 1 |
Echinococcus multilocularis | tar DNA binding protein | 0.047 | 0.6203 | 0.6203 |
Loa Loa (eye worm) | TAR-binding protein | 0.047 | 0.6203 | 1 |
Schistosoma mansoni | tar DNA-binding protein | 0.047 | 0.6203 | 0.6203 |
Brugia malayi | TAR-binding protein | 0.047 | 0.6203 | 1 |
Schistosoma mansoni | tar DNA-binding protein | 0.047 | 0.6203 | 0.6203 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0062 | 0.0435 | 0.5047 |
Mycobacterium leprae | Probable lipase LipE | 0.0035 | 0.006 | 0.5 |
Trichomonas vaginalis | D-aminoacylase, putative | 0.0035 | 0.006 | 0.0699 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.005 | 0.0265 | 0.3066 |
Loa Loa (eye worm) | phosphatidylinositol 3 | 0.0092 | 0.0863 | 0.1391 |
Trichomonas vaginalis | penicillin-binding protein, putative | 0.0035 | 0.006 | 0.0699 |
Echinococcus granulosus | tumor protein p63 | 0.0346 | 0.4452 | 0.4452 |
Trypanosoma cruzi | hypothetical protein, conserved | 0.0035 | 0.006 | 0.0699 |
Mycobacterium ulcerans | lipase LipD | 0.0035 | 0.006 | 0.5 |
Brugia malayi | beta-lactamase family protein | 0.0035 | 0.006 | 0.0097 |
Trypanosoma brucei | phosphatidylinositol 3-kinase tor, putative | 0.0043 | 0.0179 | 0.207 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.005 | 0.0265 | 0.3066 |
Leishmania major | target of rapamycin kinase (TOR) kinase 3 | 0.0073 | 0.0598 | 0.6934 |
Schistosoma mansoni | tar DNA-binding protein | 0.047 | 0.6203 | 0.6203 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0068 | 0.053 | 0.6145 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0054 | 0.0333 | 0.3855 |
Trichomonas vaginalis | esterase, putative | 0.0035 | 0.006 | 0.0699 |
Brugia malayi | Phosphatidylinositol 3- and 4-kinase family protein | 0.0092 | 0.0863 | 0.1391 |
Mycobacterium ulcerans | fusion of enoyl-CoA hydratase, EchA21 and lipase, LipE | 0.0035 | 0.006 | 0.5 |
Echinococcus granulosus | beta LACTamase domain containing family member | 0.0035 | 0.006 | 0.006 |
Mycobacterium ulcerans | hypothetical protein | 0.0035 | 0.006 | 0.5 |
Brugia malayi | beta-lactamase | 0.0035 | 0.006 | 0.0097 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.