TDR Targets

Basic information

Technical information

Name: Unnamed compound
MW: 581.589 | Formula: C29H30F3N7O3
H donors: 3 H acceptors: 5 LogP: 3.78 Rotable bonds: 11
Rule of 5 violations (Lipinski): 2
SMILES: C[C@@H](CNc1nccc(n1)n1ccnc1Cc1cccc(c1)NC(=O)c1ccc(c(c1)C(F)(F)F)N1CCOCC1)O
InChi: 1S/C29H30F3N7O3/c1-19(40)18-35-28-34-8-7-25(37-28)39-10-9-33-26(39)16-20-3-2-4-22(15-20)36-27(41)21-5-6-24(23(17-21)29(30,31)32)38-11-13-42-14-12-38/h2-10,15,17,19,40H,11-14,16,18H2,1H3,(H,36,41)(H,34,35,37)/t19-/m0/s1
InChiKey: GUYYXXVMTRJERW-IBGZPJMESA-N

Network

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Target Layer

Model Organisms

Species	Viewmode
Arabidopsis thaliana
Caenorhabditis elegans
Dictyostelium discoideum
Drosophila melanogaster
Escherichia coli
Homo sapiens
Mus musculus
Oryza sativa
Saccharomyces cerevisiae
Schmidtea mediterranea
Other organisms

TDR Pathogens:

Species	Viewmode
Brugia malayi
Chlamydia trachomatis
Echinococcus granulosus
Entamoeba histolytica
Echinococcus multilocularis
Giardia lamblia
Leishmania major
Loa Loa (eye worm)
Mycobacterium leprae
Mycobacterium tuberculosis
Mycobacterium ulcerans
Onchocerca volvulus
Plasmodium falciparum
Plasmodium vivax
Schistosoma mansoni
Trypanosoma brucei
Trypanosoma cruzi
Toxoplasma gondii
Treponema pallidum
Trichomonas vaginalis
Wolbachia endosymbiont of Brugia malayi

Other Pathogens:

Species	Viewmode
Babesia bovis
Candida albicans
Cryptosporidium hominis
Cryptosporidium parvum
Leishmania braziliensis
Leishmania donovani
Leishmania infantum
Leishmania mexicana
Neospora caninum
Plasmodium berghei
Plasmodium knowlesi
Plasmodium yoelii
Schistosoma japonicum
Trypanosoma brucei gambiense
Trypanosoma congolense
Theileria parva

Compound Layer

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Clustering layers

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Synonyms

No synonyms found for this compound

Targets

Known targets for this compound

No curated genes were found associated with this compound

Predicted pathogen targets for this compound

By orthology

No druggable targets predicted by orthology data

By sequence similarity to non orthologous known druggable targets

No druggable targets predicted by sequence similarity

Ranking Plot

Putative Targets List

Species	Potential target	Raw	Global	Species
Schistosoma mansoni	DNA topoisomerase type I	0.0364	0.5208	0.5208
Schistosoma mansoni	DNA topoisomerase type I	0.0364	0.5208	0.5208
Schistosoma mansoni	family S9 non-peptidase homologue (S09 family)	0.0045	0.029	0.029
Loa Loa (eye worm)	hypothetical protein	0.0035	0.014	0.0269
Loa Loa (eye worm)	beta-LACTamase domain containing family member	0.0035	0.014	0.0269
Echinococcus multilocularis	bromodomain adjacent to zinc finger domain	0.0058	0.0497	0.0497
Echinococcus multilocularis	DNA topoisomerase 2 alpha	0.0272	0.3792	0.3792
Mycobacterium tuberculosis	POSSIBLE PARA-NITROBENZYL ESTERASE (FRAGMENT)	0.0045	0.029	0.0402
Trypanosoma cruzi	hypothetical protein, conserved	0.0035	0.014	0.0231
Loa Loa (eye worm)	cytochrome P450 family protein	0.0027	0.002	0.0039
Schistosoma mansoni	family S9 non-peptidase homologue (S09 family)	0.0266	0.37	0.37
Echinococcus multilocularis	family S9 non peptidase ue (S09 family)	0.0045	0.029	0.029
Trichomonas vaginalis	fructose-bisphosphate aldolase, putative	0.0569	0.8369	1
Trypanosoma cruzi	hypothetical protein, conserved	0.0035	0.014	0.0231
Echinococcus granulosus	mitogen activated protein kinase 3	0.005	0.0365	0.0365
Schistosoma mansoni	tar DNA-binding protein	0.0062	0.0552	0.0552
Plasmodium falciparum	topoisomerase I	0.0364	0.5208	1
Brugia malayi	MAP kinase sur-1	0.005	0.0365	0.0701
Chlamydia trachomatis	DNA gyrase subunit B	0.0159	0.2043	1
Echinococcus multilocularis	geminin	0.0166	0.2152	0.2152
Trichomonas vaginalis	fructose-bisphosphate aldolase, putative	0.0569	0.8369	1
Loa Loa (eye worm)	hypothetical protein	0.0038	0.0176	0.0337
Onchocerca volvulus	Putative DNA topoisomerase 2, mitochondrial	0.0184	0.2432	1
Mycobacterium ulcerans	putative regulatory protein	0.0035	0.0135	0.0297
Plasmodium falciparum	DNA topoisomerase 2	0.0272	0.3792	0.6994
Echinococcus multilocularis	acetylcholinesterase	0.0266	0.37	0.37
Leishmania major	DNA topoisomerase IB, large subunit	0.0364	0.5208	1
Entamoeba histolytica	fructose-1,6-bisphosphate aldolase, putative	0.0569	0.8369	1
Echinococcus multilocularis	acetylcholinesterase	0.0266	0.37	0.37
Loa Loa (eye worm)	hypothetical protein	0.0045	0.029	0.0558
Echinococcus granulosus	bromodomain adjacent to zinc finger domain	0.0035	0.0139	0.0139
Echinococcus granulosus	acetylcholinesterase	0.0266	0.37	0.37
Chlamydia trachomatis	DNA gyrase subunit B	0.0125	0.153	0.7481
Loa Loa (eye worm)	hypothetical protein	0.0045	0.029	0.0558
Leishmania major	hypothetical protein, conserved	0.0035	0.014	0.0231
Brugia malayi	Carboxylesterase family protein	0.0266	0.37	0.7104
Schistosoma mansoni	microtubule-associated protein tau	0.0675	1	1
Loa Loa (eye worm)	hypothetical protein	0.0035	0.014	0.0269
Echinococcus multilocularis	mitogen activated protein kinase 3	0.005	0.0365	0.0365
Brugia malayi	DNA topoisomerase I	0.0364	0.5208	1
Loa Loa (eye worm)	hypothetical protein	0.0042	0.024	0.0461
Echinococcus multilocularis	tar DNA binding protein	0.0062	0.0552	0.0552
Loa Loa (eye worm)	hypothetical protein	0.0037	0.0174	0.0333
Loa Loa (eye worm)	hypothetical protein	0.0045	0.029	0.0558
Loa Loa (eye worm)	hypothetical protein	0.0035	0.014	0.0269
Plasmodium vivax	DNA topoisomerase II, putative	0.0272	0.3792	0.7207
Giardia lamblia	DNA topoisomerase II	0.0258	0.3574	0.4009
Loa Loa (eye worm)	hypothetical protein	0.0045	0.029	0.0558
Mycobacterium tuberculosis	DNA gyrase (subunit B) GyrB (DNA topoisomerase (ATP-hydrolysing)) (DNA topoisomerase II) (type II DNA topoisomerase)	0.0159	0.2043	0.5086
Loa Loa (eye worm)	hypothetical protein	0.0111	0.1304	0.2503
Toxoplasma gondii	DNA topoisomerase I, putative	0.0364	0.5208	1
Loa Loa (eye worm)	carboxylesterase	0.0045	0.029	0.0558
Mycobacterium ulcerans	esterase/lipase LipP	0.0035	0.014	0.031
Schistosoma mansoni	hypothetical protein	0.0166	0.2152	0.2152
Brugia malayi	RNA binding protein	0.0062	0.0552	0.106
Brugia malayi	bHLH-PAS transcription factor	0.0035	0.0135	0.0259
Brugia malayi	PAS domain containing protein	0.0047	0.0324	0.0622
Onchocerca volvulus		0.0045	0.029	0.1194
Mycobacterium ulcerans	fusion of enoyl-CoA hydratase, EchA21 and lipase, LipE	0.0035	0.014	0.031
Schistosoma mansoni	bromodomain containing protein	0.0062	0.0551	0.0551
Brugia malayi	Carboxylesterase family protein	0.0045	0.029	0.0558
Trypanosoma cruzi	mitogen-activated protein kinase 11, putative	0.005	0.0365	0.0665
Brugia malayi	hypothetical protein	0.0158	0.2035	0.3908
Trichomonas vaginalis	carboxylesterase domain containing protein, putative	0.0045	0.029	0.0183
Leishmania major	DNA topoisomerase ii	0.0258	0.3566	0.6835
Plasmodium vivax	DNA gyrase subunit A, putative	0.0059	0.0499	0.0709
Schistosoma mansoni	gliotactin	0.0045	0.029	0.029
Mycobacterium leprae	Probable fructose bisphosphate aldolase Fba	0.0278	0.3882	1
Brugia malayi	beta-lactamase	0.0035	0.014	0.0269
Loa Loa (eye worm)	hypothetical protein	0.0069	0.0663	0.1274
Mycobacterium ulcerans	DNA gyrase subunit B	0.0159	0.2043	0.5239
Brugia malayi	DNA topoisomerase II, alpha isozyme	0.0272	0.3792	0.7282
Onchocerca volvulus		0.0045	0.029	0.1194
Schistosoma mansoni	serine/threonine protein kinase	0.005	0.0365	0.0365
Brugia malayi	Carboxylesterase family protein	0.0266	0.37	0.7104
Echinococcus granulosus	para nitrobenzyl esterase	0.0045	0.029	0.029
Onchocerca volvulus		0.0035	0.014	0.0575
Echinococcus granulosus	carboxylesterase 5A	0.0266	0.37	0.37
Schistosoma mansoni	tar DNA-binding protein	0.0062	0.0552	0.0552
Toxoplasma gondii	ATPase/histidine kinase/DNA gyrase B/HSP90 domain-containing protein	0.0159	0.2043	0.3756
Onchocerca volvulus		0.0045	0.029	0.1194
Entamoeba histolytica	DNA topoisomerase II, putative	0.0272	0.3792	0.3714
Trypanosoma brucei	DNA topoisomerase II alpha, putative	0.0258	0.3566	0.6835
Loa Loa (eye worm)	RNA recognition domain-containing protein domain-containing protein	0.0062	0.0552	0.106
Trypanosoma brucei	DNA topoisomerase II beta, putative	0.0258	0.3566	0.6835
Schistosoma mansoni	DNA topoisomerase II	0.0272	0.3792	0.3792
Loa Loa (eye worm)	CYP4Cod1	0.0027	0.002	0.0039
Echinococcus granulosus	tar DNA binding protein	0.0062	0.0552	0.0552
Echinococcus granulosus	geminin	0.0166	0.2152	0.2152
Plasmodium vivax	DNA gyrase subunit B, putative	0.0159	0.2043	0.3756
Brugia malayi	hypoxia-induced factor 1	0.0146	0.1846	0.3545
Mycobacterium ulcerans	hypothetical protein	0.0035	0.014	0.031
Entamoeba histolytica	fructose-1,6-bisphosphate aldolase, putative	0.0569	0.8369	1
Trichomonas vaginalis	fructose-bisphosphate aldolase, putative	0.0569	0.8369	1
Loa Loa (eye worm)	TOPoisomerase family member	0.0272	0.3792	0.7282
Loa Loa (eye worm)	acetylcholinesterase 1	0.0266	0.37	0.7104
Echinococcus multilocularis	beta LACTamase domain containing family member	0.0035	0.014	0.014
Trypanosoma brucei	protein kinase, putative	0.005	0.0365	0.0665
Onchocerca volvulus		0.0045	0.029	0.1194
Mycobacterium tuberculosis	Carboxylesterase LipT	0.0045	0.029	0.0402
Trypanosoma cruzi	mitochondrial DNA topoisomerase II, putative	0.0306	0.4306	0.8262
Brugia malayi	Bromodomain containing protein	0.0073	0.0728	0.1397
Trichomonas vaginalis	fructose-bisphosphate aldolase, putative	0.0569	0.8369	1
Brugia malayi	Carboxylesterase family protein	0.0045	0.029	0.0558
Loa Loa (eye worm)	hypothetical protein	0.0035	0.014	0.0269
Loa Loa (eye worm)	hypothetical protein	0.004	0.0211	0.0406
Loa Loa (eye worm)	beta-lactamase	0.0035	0.014	0.0269
Treponema pallidum	DNA gyrase, subunit B (gyrB)	0.0159	0.2043	0.1962
Brugia malayi	TAR-binding protein	0.0062	0.0552	0.106
Brugia malayi	Hypothetical 52.5 kDa protein ZK945.1 in chromosome II, putative	0.0035	0.014	0.0269
Onchocerca volvulus		0.0035	0.014	0.0575
Mycobacterium tuberculosis	Probable fructose-bisphosphate aldolase Fba	0.0278	0.3882	1
Trypanosoma cruzi	DNA topoisomerase IB, large subunit, putative	0.0364	0.5208	1
Trichomonas vaginalis	fructose-bisphosphate aldolase, putative	0.0569	0.8369	1
Trichomonas vaginalis	fructose-bisphosphate aldolase, putative	0.0569	0.8369	1
Mycobacterium ulcerans	carboxylesterase, LipT	0.0045	0.029	0.0699
Trypanosoma cruzi	mitochondrial DNA topoisomerase II, putative	0.0306	0.4306	0.8262
Loa Loa (eye worm)	CMGC/MAPK/ERK1 protein kinase	0.005	0.0365	0.0701
Toxoplasma gondii	DNA topoisomerase 2, putative	0.0272	0.3792	0.7207
Echinococcus granulosus	beta LACTamase domain containing family member	0.0035	0.014	0.014
Trichomonas vaginalis	CMGC family protein kinase	0.005	0.0365	0.0274
Trypanosoma cruzi	mitogen activated protein kinase 4, putative	0.005	0.0365	0.0665
Loa Loa (eye worm)	carboxylesterase	0.0045	0.029	0.0558
Leishmania major	mitogen activated protein kinase, putative,map kinase, putative	0.005	0.0365	0.0665
Giardia lamblia	DNA repair protein RAD52	0.034	0.4838	0.5588
Wolbachia endosymbiont of Brugia malayi	DNA gyrase, topoisomerase II, B subunit, GyrB	0.0159	0.2043	1
Trypanosoma cruzi	DNA topoisomerase II, putative	0.0258	0.3566	0.6835
Plasmodium falciparum	DNA gyrase subunit B	0.0159	0.2043	0.3279
Trichomonas vaginalis	CMGC family protein kinase	0.005	0.0365	0.0274
Loa Loa (eye worm)	carboxylesterase	0.0266	0.37	0.7104
Loa Loa (eye worm)	DNA topoisomerase I	0.0364	0.5208	1
Brugia malayi	Carboxylesterase family protein	0.0045	0.029	0.0558
Echinococcus granulosus	BC026374 protein S09 family	0.0045	0.029	0.029
Schistosoma mansoni	neuroligin 3 (S09 family)	0.0045	0.029	0.029
Schistosoma mansoni	family S9 non-peptidase homologue (S09 family)	0.0045	0.029	0.029
Brugia malayi	DNA gyrase/topoisomerase IV, A subunit family protein	0.0272	0.3792	0.7282
Loa Loa (eye worm)	hypothetical protein	0.0037	0.0174	0.0333
Onchocerca volvulus	DNA topoisomerase 2 homolog	0.0184	0.2432	1
Trichomonas vaginalis	fructose-bisphosphate aldolase, putative	0.0569	0.8369	1
Echinococcus granulosus	mitogen activated protein kinase	0.005	0.0365	0.0365
Schistosoma mansoni	BC026374 protein (S09 family)	0.0045	0.029	0.029
Echinococcus multilocularis	BC026374 protein (S09 family)	0.0045	0.029	0.029
Echinococcus granulosus	family S9 non peptidase ue S09 family	0.0045	0.029	0.029
Mycobacterium tuberculosis	Possible penicillin-binding protein	0.0225	0.3065	0.7815
Loa Loa (eye worm)	hypothetical protein	0.0045	0.029	0.0558
Mycobacterium leprae	Probable DNA gyrase (subunit B) GyrB (DNA topoisomerase (ATP-hydrolysing)) (DNA topoisomerase II) (Type II DNA topoisomerase)	0.0071	0.0687	0.1463
Schistosoma mansoni	tar DNA-binding protein	0.0062	0.0552	0.0552
Echinococcus granulosus	acetylcholinesterase	0.0266	0.37	0.37
Entamoeba histolytica	DNA repair and recombination protein RAD52, putative	0.034	0.4838	0.515
Giardia lamblia	Fructose-bisphosphate aldolase	0.0569	0.8369	1
Mycobacterium tuberculosis	POSSIBLE PARA-NITROBENZYL ESTERASE (FRAGMENT)	0.0045	0.029	0.0402
Schistosoma mansoni	tar DNA-binding protein	0.0062	0.0552	0.0552
Schistosoma mansoni	hypothetical protein	0.0166	0.2152	0.2152
Schistosoma mansoni	family S12 unassigned peptidase (S12 family)	0.0035	0.014	0.014
Onchocerca volvulus		0.0035	0.0135	0.0555
Schistosoma mansoni	DNA topoisomerase type I	0.0364	0.5208	0.5208
Echinococcus multilocularis	para nitrobenzyl esterase	0.0045	0.029	0.029
Echinococcus granulosus	DNA topoisomerase 1	0.0364	0.5208	0.5208
Brugia malayi	Cytochrome P450 family protein	0.0027	0.002	0.0039
Echinococcus multilocularis	bromodomain adjacent to zinc finger domain	0.0035	0.0139	0.0139
Echinococcus multilocularis	carboxylesterase 5A	0.0266	0.37	0.37
Loa Loa (eye worm)	hypothetical protein	0.0035	0.014	0.0269
Loa Loa (eye worm)	hypothetical protein	0.0266	0.37	0.7104
Loa Loa (eye worm)	hypothetical protein	0.0184	0.2436	0.4678
Brugia malayi	Cytochrome P450 family protein	0.0027	0.002	0.0039
Trichomonas vaginalis	fructose-bisphosphate aldolase, putative	0.0569	0.8369	1
Loa Loa (eye worm)	hypothetical protein	0.0158	0.2035	0.3908
Echinococcus multilocularis	transfer RNA-Lys	0.0035	0.0135	0.0135
Schistosoma mansoni	single-minded	0.0047	0.0324	0.0324
Onchocerca volvulus		0.0035	0.014	0.0575
Onchocerca volvulus		0.0045	0.029	0.1194
Treponema pallidum	fructose-bisphosphate aldolase	0.0569	0.8369	1
Schistosoma mansoni	acetylcholinesterase	0.0045	0.029	0.029
Loa Loa (eye worm)	RNA binding protein	0.0062	0.0552	0.106
Loa Loa (eye worm)	hypothetical protein	0.0111	0.1304	0.2503
Mycobacterium ulcerans	DNA gyrase subunit A	0.0059	0.0499	0.1241
Leishmania major	mitochondrial DNA topoisomerase II	0.0306	0.4306	0.8262
Schistosoma mansoni	family S12 unassigned peptidase (S12 family)	0.0035	0.014	0.014
Brugia malayi	Carboxylesterase family protein	0.0045	0.029	0.0558
Brugia malayi	hypothetical protein	0.0045	0.029	0.0558
Brugia malayi	beta-lactamase family protein	0.0035	0.014	0.0269
Loa Loa (eye worm)	hypothetical protein	0.0035	0.014	0.0269
Trypanosoma brucei	DNA topoisomerase IB, large subunit	0.0364	0.5208	1
Trypanosoma brucei	DNA topoisomerase ii	0.0306	0.4306	0.8262
Trypanosoma brucei	mitogen activated protein kinase 4, putative	0.005	0.0365	0.0665
Echinococcus multilocularis	neuroligin	0.0045	0.029	0.029
Trichomonas vaginalis	DNA topoisomerase II, putative	0.0272	0.3792	0.4438
Loa Loa (eye worm)	hypothetical protein	0.0045	0.029	0.0558
Loa Loa (eye worm)	cytochrome P450 family protein	0.0027	0.002	0.0039
Leishmania major	mitogen activated protein kinase 4, putative;with=GeneDB:LmxM19.1440	0.005	0.0365	0.0665
Brugia malayi	RNA recognition motif domain containing protein	0.0062	0.0552	0.106
Mycobacterium ulcerans	beta-lactamase	0.0035	0.014	0.031
Mycobacterium tuberculosis	DNA gyrase (subunit A) GyrA (DNA topoisomerase (ATP-hydrolysing)) (DNA topoisomerase II) (type II DNA topoisomerase)	0.0059	0.0499	0.0961
Schistosoma mansoni	aryl hydrocarbon receptor	0.0047	0.0324	0.0324
Echinococcus multilocularis	mitogen activated protein kinase	0.005	0.0365	0.0365
Toxoplasma gondii	CMGC kinase, MAPK family (ERK) MAPK-1	0.005	0.0365	0.0445
Schistosoma mansoni	tar DNA-binding protein	0.0062	0.0552	0.0552
Echinococcus granulosus	DNA topoisomerase 2 alpha	0.0272	0.3792	0.3792
Brugia malayi	Bromodomain containing protein	0.0037	0.0174	0.0335
Brugia malayi	Probable DNA topoisomerase II	0.0272	0.3792	0.7282
Plasmodium vivax	topoisomerase I, putative	0.0364	0.5208	1
Echinococcus multilocularis	microtubule associated protein 2	0.0675	1	1
Trypanosoma cruzi	mitogen-activated protein kinase 11, putative	0.005	0.0365	0.0665
Echinococcus granulosus	single minded 2	0.0035	0.0135	0.0135
Echinococcus granulosus	bromodomain adjacent to zinc finger domain	0.0058	0.0497	0.0497
Echinococcus multilocularis	DNA topoisomerase 1	0.0364	0.5208	0.5208
Loa Loa (eye worm)	hypothetical protein	0.0037	0.0174	0.0333
Loa Loa (eye worm)	TAR-binding protein	0.0062	0.0552	0.106
Schistosoma mansoni	family S9 non-peptidase homologue (S09 family)	0.0045	0.029	0.029
Loa Loa (eye worm)	hypothetical protein	0.0184	0.2436	0.4678
Brugia malayi	beta-lactamase family protein	0.0035	0.014	0.0269
Loa Loa (eye worm)	hypoxia-induced factor 1	0.0146	0.1846	0.3545
Mycobacterium ulcerans	fructose-bisphosphate aldolase	0.0278	0.3882	1
Echinococcus granulosus	neuroligin	0.0045	0.029	0.029
Toxoplasma gondii	DNA gyrase/topoisomerase IV, A subunit domain-containing protein	0.0059	0.0499	0.0709
Trichomonas vaginalis	spcc417.12 protein, putative	0.0045	0.029	0.0183
Chlamydia trachomatis	DNA gyrase subunit A	0.0059	0.0499	0.2427
Loa Loa (eye worm)	hypothetical protein	0.0045	0.029	0.0558
Trypanosoma brucei	hypothetical protein, conserved	0.0035	0.014	0.0231
Chlamydia trachomatis	DNA gyrase subunit A	0.0059	0.0499	0.2427
Loa Loa (eye worm)	hypothetical protein	0.0266	0.37	0.7104
Onchocerca volvulus	DNA topoisomerase 2 homolog	0.0184	0.2432	1
Mycobacterium ulcerans	lipase LipD	0.0035	0.014	0.031
Trypanosoma cruzi	DNA topoisomerase II, putative	0.0258	0.3566	0.6835
Trichomonas vaginalis	CMGC family protein kinase	0.005	0.0365	0.0274
Trypanosoma cruzi	mitogen activated protein kinase 2, putative	0.005	0.0365	0.0665
Trichomonas vaginalis	CMGC family protein kinase	0.005	0.0365	0.0274

Activities

No activities found for this compound.

Phenotypes

Whole-cell/tissue/organism interactions

We have no records of whole-cell/tissue assays done with this compound What does this mean?

Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.

Annotated phenotypes:

We have no manually annotated phenotypes for this drug. What does this mean? / Care to help?

In TDR Targets, information about phenotypes that are caused by drugs, or by genetic manipulation of cells (e.g. gene knockouts or knockdowns) is manually curated from the literature. These descriptions help to describe the potential of the target for drug development. If no information is available for this gene or if the information is incomplete, this may mean that i) the papers containing this information either appeared after the curation effort for this organism was carried out or they were inadvertently missed by curators; or that ii) the curation effort for this organism has not yet started.

In any case, if you have information about papers containing relevant validation data for this target, please log in using your TDR Targets username and password and send them to us using the corresponding form in this page (only visible to registered users) or contact us.

External resources for this compound

ChEMBL: CHEMBL3309395

Bibliographic References

No literature references available for this target.

If you have references for this compound, please enter them in a user comment (below) or Contact us.

Detailed information for compound 916057