Species | Target name | Source | Bibliographic reference |
---|---|---|---|
Homo sapiens | cannabinoid receptor 1 (brain) | Starlite/ChEMBL | References |
Homo sapiens | cannabinoid receptor 2 (macrophage) | Starlite/ChEMBL | References |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
Ki (binding) | = 27.1 nM | HEK293DHEK293iHEK293sHEK293pHEK293lHEK293aHEK293cHEK293eHEK293mHEK293eHEK293nHEK293tHEK293 HEK293oHEK293fHEK293 HEK293[HEK2933HEK293HHEK293]HEK293CHEK293PHEK293-HEK2935HEK2935HEK293,HEK2939HEK2934HEK2930HEK293 HEK293fHEK293rHEK293oHEK293mHEK293 HEK293hHEK293uHEK293mHEK293aHEK293nHEK293 HEK293rHEK293eHEK293cHEK293oHEK293mHEK293bHEK293iHEK293nHEK293aHEK293nHEK293tHEK293 HEK293CHEK293BHEK2932HEK293RHEK293 HEK293eHEK293xHEK293pHEK293rHEK293eHEK293sHEK293sHEK293eHEK293dHEK293 HEK293iHEK293nHEK293 HEK293HHEK293EHEK293KHEK293-HEK2932HEK2939HEK2933HEK293 HEK293cHEK293eHEK293lHEK293lHEK293sHEK293 HEK293aHEK293fHEK293tHEK293eHEK293rHEK293 HEK2939HEK2930HEK293 HEK293mHEK293iHEK293nHEK293sHEK293 HEK293bHEK293yHEK293 HEK293lHEK293iHEK293qHEK293uHEK293iHEK293dHEK293 HEK293sHEK293cHEK293iHEK293nHEK293tHEK293iHEK293lHEK293lHEK293aHEK293tHEK293iHEK293oHEK293nHEK293 HEK293cHEK293oHEK293uHEK293nHEK293tHEK293iHEK293nHEK293gHEK293 | ChEMBL. | 25272206 |
Ki (binding) | > 10000 nM | HEK293DHEK293iHEK293sHEK293pHEK293lHEK293aHEK293cHEK293eHEK293mHEK293eHEK293nHEK293tHEK293 HEK293oHEK293fHEK293 HEK293[HEK2933HEK293HHEK293]HEK293CHEK293PHEK293-HEK2935HEK2935HEK293,HEK2939HEK2934HEK2930HEK293 HEK293fHEK293rHEK293oHEK293mHEK293 HEK293hHEK293uHEK293mHEK293aHEK293nHEK293 HEK293rHEK293eHEK293cHEK293oHEK293mHEK293bHEK293iHEK293nHEK293aHEK293nHEK293tHEK293 HEK293CHEK293BHEK2931HEK293RHEK293 HEK293eHEK293xHEK293pHEK293rHEK293eHEK293sHEK293sHEK293eHEK293dHEK293 HEK293iHEK293nHEK293 HEK293HHEK293EHEK293KHEK293-HEK2932HEK2939HEK2933HEK293 HEK293cHEK293eHEK293lHEK293lHEK293sHEK293 HEK293aHEK293fHEK293tHEK293eHEK293rHEK293 HEK2939HEK2930HEK293 HEK293mHEK293iHEK293nHEK293sHEK293 HEK293bHEK293yHEK293 HEK293lHEK293iHEK293qHEK293uHEK293iHEK293dHEK293 HEK293sHEK293cHEK293iHEK293nHEK293tHEK293iHEK293lHEK293lHEK293aHEK293tHEK293iHEK293oHEK293nHEK293 HEK293cHEK293oHEK293uHEK293nHEK293tHEK293iHEK293nHEK293gHEK293 | ChEMBL. | 25272206 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.