Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Echinococcus granulosus | hyperpolarization activated cyclic | 0.0103 | 0.0035 | 0.0053 |
Trichomonas vaginalis | voltage and ligand gated potassium channel, putative | 0.0103 | 0.0035 | 0.0035 |
Schistosoma mansoni | voltage-gated potassium channel | 0.0103 | 0.0035 | 0.0053 |
Echinococcus multilocularis | voltage gated potassium channel | 0.0151 | 0.0185 | 0.0278 |
Trichomonas vaginalis | AGC family protein kinase | 0.3297 | 1 | 1 |
Plasmodium falciparum | cGMP-dependent protein kinase | 0.0092 | 0.0002 | 0.0004 |
Schistosoma mansoni | serine/threonine protein kinase | 0.1098 | 0.3141 | 0.4725 |
Echinococcus multilocularis | ribosomal protein S6 kinase alpha 3 | 0.1098 | 0.3141 | 0.4725 |
Trichomonas vaginalis | AGC family protein kinase | 0.0115 | 0.0074 | 0.0074 |
Leishmania major | rac serine-threonine kinase, putative,protein kinase, putative | 0.0115 | 0.0074 | 1 |
Echinococcus multilocularis | serine:threonine protein kinase N2 | 0.1098 | 0.3141 | 0.4725 |
Loa Loa (eye worm) | AGC/RSK/MSK protein kinase | 0.1098 | 0.3141 | 0.3141 |
Brugia malayi | Cyclic-nucleotide gated cation channel | 0.0103 | 0.0035 | 0.0035 |
Leishmania major | protein kinase, putative | 0.0092 | 0.0002 | 0.0326 |
Trichomonas vaginalis | AGC family protein kinase | 0.0115 | 0.0074 | 0.0074 |
Schistosoma mansoni | voltage-gated potassium channel | 0.0151 | 0.0185 | 0.0278 |
Schistosoma mansoni | serine/threonine protein kinase | 0.1098 | 0.3141 | 0.4725 |
Brugia malayi | Voltage-gated potassium channel, EAG (KCNH1)-related. C. elegans egl-2 ortholog | 0.0151 | 0.0185 | 0.0185 |
Schistosoma mansoni | serine/threonine protein kinase | 0.1098 | 0.3141 | 0.4725 |
Schistosoma mansoni | serine/threonine protein kinase | 0.1098 | 0.3141 | 0.4725 |
Echinococcus granulosus | potassium:sodium hyperpolarization activated | 0.0103 | 0.0035 | 0.0053 |
Trypanosoma cruzi | rac serine-threonine kinase, putative | 0.213 | 0.6361 | 0.957 |
Trypanosoma cruzi | Serine/threonine-protein kinase NEK21, putative | 0.0115 | 0.0074 | 0.0111 |
Schistosoma mansoni | serine/threonine kinase | 0.1098 | 0.3141 | 0.4725 |
Onchocerca volvulus | 0.0092 | 0 | 0.5 | |
Entamoeba histolytica | protein kinase, putative | 0.3205 | 0.9714 | 0.9714 |
Echinococcus multilocularis | expressed conserved protein | 0.0092 | 0.0002 | 0.0004 |
Trypanosoma brucei | serine/threonine-protein kinase NRKB, putative | 0.0115 | 0.0074 | 0.0074 |
Plasmodium vivax | calcium-dependent protein kinase 7, putative | 0.0115 | 0.0074 | 0.0116 |
Trichomonas vaginalis | AGC family protein kinase | 0.0115 | 0.0074 | 0.0074 |
Onchocerca volvulus | Abnormal cell migration protein 10 homolog | 0.0092 | 0 | 0.5 |
Trypanosoma cruzi | serine/threonine protein kinase, putative | 0.0115 | 0.0074 | 0.0111 |
Brugia malayi | Voltage-gated potassium channel, HERG (KCNH2)-related. C. elegans unc-103 ortholog | 0.0521 | 0.1339 | 0.1339 |
Trypanosoma cruzi | NIMA-related kinase, putative | 0.0115 | 0.0074 | 0.0111 |
Brugia malayi | Protein kinase domain containing protein | 0.1098 | 0.3141 | 0.3141 |
Brugia malayi | Hr1 repeat family protein | 0.1098 | 0.3141 | 0.3141 |
Echinococcus granulosus | nervana 2 | 0.2107 | 0.6287 | 0.9458 |
Echinococcus granulosus | protein kinase C gamma type | 0.1098 | 0.3141 | 0.4725 |
Trichomonas vaginalis | AGC family protein kinase | 0.0115 | 0.0074 | 0.0074 |
Echinococcus granulosus | calcium:calmodulin dependent protein kinase | 0.213 | 0.6361 | 0.957 |
Toxoplasma gondii | protein kinase G AGC kinase family member PKG | 0.0092 | 0.0002 | 0.0002 |
Schistosoma mansoni | voltage-gated potassium channel | 0.0151 | 0.0185 | 0.0278 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.0115 | 0.0074 | 0.0074 |
Trypanosoma brucei | protein kinase, putative | 0.0115 | 0.0074 | 0.0074 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.0115 | 0.0074 | 0.0074 |
Trypanosoma cruzi | Protein kinase B | 0.2222 | 0.6647 | 1 |
Schistosoma mansoni | cyclic-nucleotide-gated cation channel | 0.0103 | 0.0035 | 0.0053 |
Echinococcus granulosus | NDR protein kinase | 0.1098 | 0.3141 | 0.4725 |
Leishmania major | protein kinase, putative | 0.0115 | 0.0074 | 1 |
Echinococcus multilocularis | serine threonine protein kinase nrc serine threonine protein kinase gad | 0.213 | 0.6361 | 0.957 |
Onchocerca volvulus | 0.0092 | 0 | 0.5 | |
Echinococcus multilocularis | nervana 2 | 0.2107 | 0.6287 | 0.9458 |
Trypanosoma cruzi | rac serine-threonine kinase, putative | 0.0115 | 0.0074 | 0.0111 |
Leishmania major | protein kinase, putative,serine/threonine protein kinase, putative | 0.0115 | 0.0074 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.0115 | 0.0074 | 0.0074 |
Echinococcus multilocularis | hyperpolarization activated cyclic | 0.0103 | 0.0035 | 0.0053 |
Trichomonas vaginalis | AGC family protein kinase | 0.3297 | 1 | 1 |
Schistosoma mansoni | cyclic-nucleotide-gated cation channel | 0.0103 | 0.0035 | 0.0053 |
Echinococcus multilocularis | serine:threonine protein kinase N2 | 0.1098 | 0.3141 | 0.4725 |
Echinococcus multilocularis | cGMP dependent protein kinase 1 | 0.0092 | 0.0002 | 0.0004 |
Onchocerca volvulus | 0.0092 | 0 | 0.5 | |
Echinococcus multilocularis | cGMP dependent protein kinase 1 | 0.0092 | 0.0002 | 0.0004 |
Echinococcus granulosus | sodium:potassium dependent atpase beta subunit | 0.2107 | 0.6287 | 0.9458 |
Onchocerca volvulus | outspread protein homolog | 0.0092 | 0 | 0.5 |
Entamoeba histolytica | protein kinase, putative | 0.0115 | 0.0074 | 0.0074 |
Echinococcus granulosus | cyclic nucleotide gated cation channel alpha 3 | 0.0103 | 0.0035 | 0.0053 |
Onchocerca volvulus | 0.0092 | 0 | 0.5 | |
Schistosoma mansoni | serine/threonine protein kinase | 0.0092 | 0.0002 | 0.0004 |
Echinococcus granulosus | potassium voltage gated channel subfamily H | 0.0521 | 0.1339 | 0.2014 |
Echinococcus granulosus | voltage gated potassium channel | 0.0151 | 0.0185 | 0.0278 |
Echinococcus granulosus | protein kinase c iota type | 0.1098 | 0.3141 | 0.4725 |
Echinococcus granulosus | serine:threonine protein kinase N2 | 0.1098 | 0.3141 | 0.4725 |
Leishmania major | protein kinase, putative | 0.0115 | 0.0074 | 1 |
Toxoplasma gondii | calcium dependent protein kinase CDPK7 | 0.0115 | 0.0074 | 0.0076 |
Echinococcus granulosus | cyclic nucleotide gated cation channel | 0.0103 | 0.0035 | 0.0053 |
Trichomonas vaginalis | AGC family protein kinase | 0.0115 | 0.0074 | 0.0074 |
Echinococcus multilocularis | nervana 2 | 0.2107 | 0.6287 | 0.9458 |
Trypanosoma cruzi | serine/threonine-protein kinase NRKB, putative | 0.0115 | 0.0074 | 0.0111 |
Trichomonas vaginalis | AGC family protein kinase | 0.0115 | 0.0074 | 0.0074 |
Echinococcus multilocularis | potassium voltage gated channel subfamily H | 0.0521 | 0.1339 | 0.2014 |
Schistosoma mansoni | serine/threonine protein kinase | 0.1098 | 0.3141 | 0.4725 |
Trypanosoma cruzi | Serine/threonine-protein kinase NEK21, putative | 0.0115 | 0.0074 | 0.0111 |
Brugia malayi | protein kinase C II. | 0.1098 | 0.3141 | 0.3141 |
Onchocerca volvulus | Protein melted homolog | 0.0092 | 0 | 0.5 |
Entamoeba histolytica | protein kinase, putative | 0.3297 | 1 | 1 |
Plasmodium falciparum | calcium-dependent protein kinase 7 | 0.0115 | 0.0074 | 0.0116 |
Schistosoma mansoni | serine/threonine protein kinase | 0.1098 | 0.3141 | 0.4725 |
Echinococcus multilocularis | Glutaredoxin protein 5 | 0.2107 | 0.6287 | 0.9458 |
Trypanosoma brucei | NEK family Serine/threonine-protein kinase, putative | 0.0115 | 0.0074 | 0.0074 |
Echinococcus multilocularis | Ribosomal protein S6 kinase beta 2 | 0.1098 | 0.3141 | 0.4725 |
Trypanosoma cruzi | rac serine-threonine kinase, putative | 0.2222 | 0.6647 | 1 |
Echinococcus multilocularis | Protein kinase C, brain isozyme | 0.1098 | 0.3141 | 0.4725 |
Echinococcus multilocularis | hyperpolarization activated cyclic | 0.0103 | 0.0035 | 0.0053 |
Schistosoma mansoni | hyperpolarization activated cyclic nucleotide-gated potassium channel | 0.0103 | 0.0035 | 0.0053 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.2222 | 0.6647 | 0.6647 |
Trichomonas vaginalis | voltage and ligand gated potassium channel, putative | 0.0103 | 0.0035 | 0.0035 |
Echinococcus granulosus | potassium voltage gated channel subfamily H | 0.0151 | 0.0185 | 0.0278 |
Trichomonas vaginalis | 3-phosphoinositide dependent protein kinase-1, putative | 0.0115 | 0.0074 | 0.0074 |
Trichomonas vaginalis | AGC family protein kinase | 0.0115 | 0.0074 | 0.0074 |
Echinococcus multilocularis | potassium voltage gated channel subfamily H | 0.0151 | 0.0185 | 0.0278 |
Loa Loa (eye worm) | voltage and ligand gated potassium channel | 0.0521 | 0.1339 | 0.1339 |
Trichomonas vaginalis | voltage and ligand gated potassium channel, putative | 0.0487 | 0.1232 | 0.1232 |
Trichomonas vaginalis | AGC family protein kinase | 0.0115 | 0.0074 | 0.0074 |
Trypanosoma brucei | Serine/threonine-protein kinase NEK21, putative | 0.0115 | 0.0074 | 0.0074 |
Trichomonas vaginalis | AGC family protein kinase | 0.0115 | 0.0074 | 0.0074 |
Trichomonas vaginalis | AGC family protein kinase | 0.0115 | 0.0074 | 0.0074 |
Echinococcus granulosus | nervana 2 | 0.2107 | 0.6287 | 0.9458 |
Trichomonas vaginalis | AGC family protein kinase | 0.1098 | 0.3141 | 0.3141 |
Echinococcus granulosus | ribosomal protein S6 kinase alpha 3 | 0.1098 | 0.3141 | 0.4725 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.0115 | 0.0074 | 0.0074 |
Loa Loa (eye worm) | AGC/AKT protein kinase | 0.3297 | 1 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.0115 | 0.0074 | 0.0074 |
Echinococcus granulosus | ribosomal protein s6 kinase beta 1 | 0.1098 | 0.3141 | 0.4725 |
Entamoeba histolytica | protein kinase, putative | 0.1098 | 0.3141 | 0.3141 |
Trichomonas vaginalis | AGC family protein kinase | 0.3297 | 1 | 1 |
Entamoeba histolytica | protein kinase, putative | 0.0115 | 0.0074 | 0.0074 |
Trichomonas vaginalis | AGC family protein kinase | 0.3297 | 1 | 1 |
Schistosoma mansoni | voltage-gated potassium channel | 0.0569 | 0.1488 | 0.2239 |
Plasmodium falciparum | RAC-beta serine/threonine protein kinase | 0.213 | 0.6361 | 1 |
Schistosoma mansoni | voltage-gated potassium channel | 0.0569 | 0.1488 | 0.2239 |
Echinococcus granulosus | Glutaredoxin protein 5 | 0.2107 | 0.6287 | 0.9458 |
Brugia malayi | Protein kinase domain containing protein | 0.1098 | 0.3141 | 0.3141 |
Echinococcus multilocularis | protein kinase c epsilon type | 0.1098 | 0.3141 | 0.4725 |
Leishmania major | serine/threonine-protein kinase a, putative | 0.0115 | 0.0074 | 1 |
Entamoeba histolytica | hypothetical protein | 0.0115 | 0.0074 | 0.0074 |
Echinococcus granulosus | serine/threonine protein kinase | 0.2222 | 0.6647 | 1 |
Toxoplasma gondii | AGC kinase | 0.3205 | 0.9714 | 1 |
Brugia malayi | p70 ribosomal S6 kinase beta | 0.3205 | 0.9714 | 0.9714 |
Trypanosoma cruzi | Serine/threonine-protein kinase NEK17, putative | 0.0115 | 0.0074 | 0.0111 |
Trichomonas vaginalis | AGC family protein kinase | 0.0115 | 0.0074 | 0.0074 |
Onchocerca volvulus | 0.0092 | 0 | 0.5 | |
Loa Loa (eye worm) | hypothetical protein | 0.1098 | 0.3141 | 0.3141 |
Trypanosoma brucei | serine/threonine-protein kinase NrkA | 0.0115 | 0.0074 | 0.0074 |
Echinococcus granulosus | hyperpolarization activated cyclic | 0.0103 | 0.0035 | 0.0053 |
Trichomonas vaginalis | AGC family protein kinase | 0.119 | 0.3427 | 0.3427 |
Echinococcus granulosus | serine threonine protein kinase nrc | 0.213 | 0.6361 | 0.957 |
Giardia lamblia | Kinase, AGC PKA | 0.213 | 0.6361 | 0.5 |
Loa Loa (eye worm) | AGC/NDR protein kinase | 0.1098 | 0.3141 | 0.3141 |
Loa Loa (eye worm) | AGC/PKN protein kinase | 0.1098 | 0.3141 | 0.3141 |
Trichomonas vaginalis | AGC family protein kinase | 0.0115 | 0.0074 | 0.0074 |
Schistosoma mansoni | serine/threonine-protein kinase | 0.2222 | 0.6647 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0103 | 0.0035 | 0.0035 |
Echinococcus multilocularis | serine:threonine protein kinase 38 | 0.1098 | 0.3141 | 0.4725 |
Echinococcus granulosus | Ribosomal protein S6 kinase beta 2 | 0.1098 | 0.3141 | 0.4725 |
Schistosoma mansoni | hyperpolarization activated cyclic nucleotide-gated potassium channel | 0.0103 | 0.0035 | 0.0053 |
Trichomonas vaginalis | serine/threonine-protein kinase sgk, putative | 0.1075 | 0.3067 | 0.3067 |
Echinococcus multilocularis | serine threonine protein kinase | 0.1098 | 0.3141 | 0.4725 |
Onchocerca volvulus | 0.0092 | 0 | 0.5 | |
Echinococcus multilocularis | cyclic nucleotide gated cation channel alpha 3 | 0.0103 | 0.0035 | 0.0053 |
Loa Loa (eye worm) | AGC/PKG protein kinase | 0.0092 | 0.0002 | 0.0002 |
Echinococcus granulosus | protein kinase c epsilon type | 0.1098 | 0.3141 | 0.4725 |
Echinococcus granulosus | Protein kinase C brain isozyme | 0.1098 | 0.3141 | 0.4725 |
Trypanosoma cruzi | NEK family Serine/threonine-protein kinase, putative | 0.0115 | 0.0074 | 0.0111 |
Entamoeba histolytica | hypothetical protein | 0.0115 | 0.0074 | 0.0074 |
Trichomonas vaginalis | AGC family protein kinase | 0.1098 | 0.3141 | 0.3141 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.0115 | 0.0074 | 0.0074 |
Echinococcus multilocularis | potassium:sodium hyperpolarization activated | 0.0103 | 0.0035 | 0.0053 |
Trichomonas vaginalis | voltage and ligand gated potassium channel, putative | 0.0487 | 0.1232 | 0.1232 |
Echinococcus granulosus | cGMP dependent protein kinase 1 | 0.0092 | 0.0002 | 0.0004 |
Trichomonas vaginalis | AGC family protein kinase | 0.0115 | 0.0074 | 0.0074 |
Loa Loa (eye worm) | AGC/RSK/P70 protein kinase | 0.3205 | 0.9714 | 0.9714 |
Entamoeba histolytica | protein kinase, putative | 0.3297 | 1 | 1 |
Trypanosoma brucei | rac serine-threonine kinase, putative | 0.3297 | 1 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.3297 | 1 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.3297 | 1 | 1 |
Onchocerca volvulus | 0.0092 | 0 | 0.5 | |
Echinococcus granulosus | cGMP dependent protein kinase | 0.0092 | 0.0002 | 0.0004 |
Loa Loa (eye worm) | hypothetical protein | 0.0452 | 0.1124 | 0.1124 |
Trichomonas vaginalis | AGC family protein kinase | 0.0115 | 0.0074 | 0.0074 |
Echinococcus multilocularis | protein kinase c iota type | 0.1098 | 0.3141 | 0.4725 |
Trypanosoma cruzi | NIMA-related kinase, putative | 0.0115 | 0.0074 | 0.0111 |
Leishmania major | folate/biopterin transporter, putative | 0.0115 | 0.0074 | 1 |
Loa Loa (eye worm) | cyclic-nucleotide gated cation channel | 0.0103 | 0.0035 | 0.0035 |
Schistosoma mansoni | serine/threonine-protein kinase | 0.2222 | 0.6647 | 1 |
Trichomonas vaginalis | ribosomal protein S6 kinase, 90kD, polypeptide, putative | 0.0115 | 0.0074 | 0.0074 |
Onchocerca volvulus | Putative neuronal RhoA GEF protein | 0.0092 | 0 | 0.5 |
Loa Loa (eye worm) | hypothetical protein | 0.0151 | 0.0185 | 0.0185 |
Trichomonas vaginalis | AGC family protein kinase | 0.1098 | 0.3141 | 0.3141 |
Echinococcus multilocularis | ribosomal protein s6 kinase beta 1 | 0.1098 | 0.3141 | 0.4725 |
Trichomonas vaginalis | AGC family protein kinase | 0.3297 | 1 | 1 |
Schistosoma mansoni | cyclic-nucleotide-gated cation channel | 0.0103 | 0.0035 | 0.0053 |
Loa Loa (eye worm) | AGC/DMPK/GEK protein kinase | 0.1098 | 0.3141 | 0.3141 |
Entamoeba histolytica | p21-activated kinase | 0.0115 | 0.0074 | 0.0074 |
Schistosoma mansoni | memapsin-2 (A01 family) | 0.0501 | 0.1276 | 0.192 |
Entamoeba histolytica | protein kinase, putative | 0.0115 | 0.0074 | 0.0074 |
Loa Loa (eye worm) | AGC/PKC/ETA protein kinase | 0.1098 | 0.3141 | 0.3141 |
Echinococcus granulosus | cyclic nucleotide gated cation channel | 0.0103 | 0.0035 | 0.0053 |
Trichomonas vaginalis | AGC family protein kinase | 0.0115 | 0.0074 | 0.0074 |
Echinococcus multilocularis | sodium:potassium dependent atpase beta subunit | 0.2107 | 0.6287 | 0.9458 |
Trichomonas vaginalis | AGC family protein kinase | 0.0115 | 0.0074 | 0.0074 |
Echinococcus multilocularis | rac serine:threonine kinase | 0.2222 | 0.6647 | 1 |
Brugia malayi | Egg laying defective protein 4 | 0.0092 | 0.0002 | 0.0002 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.2222 | 0.6647 | 0.6647 |
Trypanosoma cruzi | Serine/threonine-protein kinase NEK17, putative | 0.0115 | 0.0074 | 0.0111 |
Entamoeba histolytica | protein kinase, putative | 0.0115 | 0.0074 | 0.0074 |
Loa Loa (eye worm) | AGC/RSK/RSK protein kinase | 0.1098 | 0.3141 | 0.3141 |
Trichomonas vaginalis | AGC family protein kinase | 0.0115 | 0.0074 | 0.0074 |
Onchocerca volvulus | Putative zinc finger protein | 0.0092 | 0 | 0.5 |
Schistosoma mansoni | serine/threonine protein kinase | 0.1098 | 0.3141 | 0.4725 |
Schistosoma mansoni | serine/threonine protein kinase | 0.0092 | 0.0002 | 0.0004 |
Trichomonas vaginalis | AGC family protein kinase | 0.0115 | 0.0074 | 0.0074 |
Entamoeba histolytica | protein kinase, putative | 0.0115 | 0.0074 | 0.0074 |
Leishmania major | protein kinase, putative | 0.0092 | 0.0002 | 0.0326 |
Echinococcus multilocularis | cyclic nucleotide gated cation channel | 0.0103 | 0.0035 | 0.0053 |
Schistosoma mansoni | atypical protein kinase C | 0.1098 | 0.3141 | 0.4725 |
Schistosoma mansoni | serine/threonine protein kinase | 0.0092 | 0.0002 | 0.0004 |
Plasmodium vivax | rac-beta serine/threonine protein kinase, putative | 0.213 | 0.6361 | 1 |
Entamoeba histolytica | protein kinase 2, putative | 0.213 | 0.6361 | 0.6361 |
Toxoplasma gondii | protein kinase domain-containing protein | 0.0115 | 0.0074 | 0.0076 |
Loa Loa (eye worm) | cyclic-nucleotide gated cation channel | 0.0103 | 0.0035 | 0.0035 |
Echinococcus granulosus | cGMP dependent protein kinase 1 | 0.0092 | 0.0002 | 0.0004 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
Km (binding) | = 32 uM | Induction of human histidine10-tagged MDR1 ATPase activity expressed in BHK cells by apparent Michaelis-Menten constant | ChEMBL. | 19402665 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.