Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Echinococcus granulosus | serine/threonine protein kinase | 0.1001 | 0.6568 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.0547 | 0.3273 | 0.0743 |
Echinococcus granulosus | calcium:calmodulin dependent protein kinase | 0.0937 | 0.6104 | 0.8766 |
Trichomonas vaginalis | AGC family protein kinase | 0.0483 | 0.2809 | 0.0104 |
Trypanosoma cruzi | rac serine-threonine kinase, putative | 0.0937 | 0.6104 | 0.9293 |
Trypanosoma brucei | rac serine-threonine kinase, putative | 0.1473 | 1 | 1 |
Loa Loa (eye worm) | AGC/DMPK/GEK protein kinase | 0.0483 | 0.2809 | 0.2809 |
Trypanosoma cruzi | Protein kinase B | 0.1001 | 0.6568 | 1 |
Brugia malayi | Cytochrome P450 family protein | 0.0252 | 0.1129 | 0.1129 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.1001 | 0.6568 | 0.5228 |
Echinococcus granulosus | sodium:potassium dependent atpase beta subunit | 0.0926 | 0.6029 | 0.8564 |
Brugia malayi | Protein kinase domain containing protein | 0.0483 | 0.2809 | 0.2809 |
Entamoeba histolytica | protein kinase 2, putative | 0.0937 | 0.6104 | 0.4583 |
Trichomonas vaginalis | AGC family protein kinase | 0.1473 | 1 | 1 |
Brugia malayi | p70 ribosomal S6 kinase beta | 0.1409 | 0.9536 | 0.9536 |
Giardia lamblia | Kinase, AGC PKA | 0.0937 | 0.6104 | 0.5 |
Trichomonas vaginalis | AGC family protein kinase | 0.0483 | 0.2809 | 0.0104 |
Echinococcus multilocularis | Glutaredoxin protein 5 | 0.0926 | 0.6029 | 0.8564 |
Entamoeba histolytica | protein kinase, putative | 0.1409 | 0.9536 | 0.9355 |
Trichomonas vaginalis | AGC family protein kinase | 0.0483 | 0.2809 | 0.0104 |
Echinococcus multilocularis | sodium:potassium dependent atpase beta subunit | 0.0926 | 0.6029 | 0.8564 |
Loa Loa (eye worm) | AGC/RSK/MSK protein kinase | 0.0483 | 0.2809 | 0.2809 |
Loa Loa (eye worm) | cytochrome P450 family protein | 0.0252 | 0.1129 | 0.1129 |
Entamoeba histolytica | protein kinase, putative | 0.1473 | 1 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.1473 | 1 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.1473 | 1 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.1473 | 1 | 1 |
Brugia malayi | Hr1 repeat family protein | 0.0483 | 0.2809 | 0.2809 |
Toxoplasma gondii | AGC kinase | 0.1409 | 0.9536 | 0.5 |
Loa Loa (eye worm) | AGC/RSK/P70 protein kinase | 0.1409 | 0.9536 | 0.9536 |
Entamoeba histolytica | protein kinase, putative | 0.1473 | 1 | 1 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.1001 | 0.6568 | 0.5228 |
Leishmania major | cytochrome p450-like protein | 0.0096 | 0 | 0.5 |
Loa Loa (eye worm) | hypothetical protein | 0.0483 | 0.2809 | 0.2809 |
Plasmodium vivax | rac-beta serine/threonine protein kinase, putative | 0.0937 | 0.6104 | 0.5 |
Brugia malayi | Protein kinase domain containing protein | 0.0483 | 0.2809 | 0.2809 |
Loa Loa (eye worm) | AGC/AKT protein kinase | 0.1473 | 1 | 1 |
Echinococcus multilocularis | nervana 2 | 0.0926 | 0.6029 | 0.8564 |
Echinococcus multilocularis | rac serine:threonine kinase | 0.1001 | 0.6568 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.1473 | 1 | 1 |
Loa Loa (eye worm) | AGC/PKC/ETA protein kinase | 0.0483 | 0.2809 | 0.2809 |
Loa Loa (eye worm) | AGC/NDR protein kinase | 0.0483 | 0.2809 | 0.2809 |
Schistosoma mansoni | serine/threonine-protein kinase | 0.1001 | 0.6568 | 1 |
Echinococcus multilocularis | nervana 2 | 0.0926 | 0.6029 | 0.8564 |
Mycobacterium ulcerans | cytochrome P450 185A4 Cyp185A4 | 0.0096 | 0 | 0.5 |
Plasmodium falciparum | RAC-beta serine/threonine protein kinase | 0.0937 | 0.6104 | 0.5 |
Echinococcus granulosus | nervana 2 | 0.0926 | 0.6029 | 0.8564 |
Trichomonas vaginalis | AGC family protein kinase | 0.1473 | 1 | 1 |
Echinococcus granulosus | Glutaredoxin protein 5 | 0.0926 | 0.6029 | 0.8564 |
Trichomonas vaginalis | AGC family protein kinase | 0.1473 | 1 | 1 |
Brugia malayi | protein kinase C II. | 0.0483 | 0.2809 | 0.2809 |
Echinococcus multilocularis | serine threonine protein kinase nrc serine threonine protein kinase gad | 0.0937 | 0.6104 | 0.8766 |
Echinococcus granulosus | nervana 2 | 0.0926 | 0.6029 | 0.8564 |
Echinococcus granulosus | serine threonine protein kinase nrc | 0.0937 | 0.6104 | 0.8766 |
Loa Loa (eye worm) | AGC/RSK/RSK protein kinase | 0.0483 | 0.2809 | 0.2809 |
Loa Loa (eye worm) | AGC/PKN protein kinase | 0.0483 | 0.2809 | 0.2809 |
Trypanosoma cruzi | rac serine-threonine kinase, putative | 0.1001 | 0.6568 | 1 |
Schistosoma mansoni | serine/threonine-protein kinase | 0.1001 | 0.6568 | 1 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
Potency (functional) | = 25.1189 um | PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Thyroid Stimulating Hormone Receptor. (Class of assay: confirmatory) | ChEMBL. | No reference |
Potency (functional) | = 39.8107 um | PUBCHEM_BIOASSAY: qHTS Assay for Inhibitors Targeting the Menin-MLL Interaction in MLL Related Leukemias: Competition With Texas Red Labeled MLL-derived Mutant Peptide. (Class of assay: confirmatory) | ChEMBL. | No reference |
Potency (functional) | 50.1187 uM | PubChem BioAssay. qHTS for Agonist of gsp, the Etiologic Mutation Responsible for Fibrous Dysplasia/McCune-Albright Syndrome: qHTS. (Class of assay: confirmatory) | ChEMBL. | No reference |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.