Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Entamoeba histolytica | serine/threonine- protein kinase 6 , putative | 0.0906 | 1 | 1 |
Schistosoma mansoni | serine/threonine protein kinase | 0.0906 | 1 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.0591 | 0.5562 | 0.5562 |
Echinococcus granulosus | sodium calcium exchanger | 0.0572 | 0.5291 | 0.5212 |
Loa Loa (eye worm) | AUR protein kinase | 0.0906 | 1 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0229 | 0.0464 | 0.0305 |
Echinococcus multilocularis | sodium:potassium dependent atpase beta subunit | 0.0384 | 0.2644 | 0.2521 |
Entamoeba histolytica | protein kinase, putative | 0.0591 | 0.5562 | 0.5488 |
Entamoeba histolytica | protein kinase, putative | 0.0906 | 1 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.0591 | 0.5562 | 0.5562 |
Brugia malayi | Protein kinase domain containing protein | 0.0591 | 0.5562 | 0.5488 |
Echinococcus granulosus | nervana 2 | 0.0384 | 0.2644 | 0.2521 |
Trichomonas vaginalis | AGC family protein kinase | 0.0906 | 1 | 1 |
Brugia malayi | serine/threonine-protein kinase 6 | 0.0906 | 1 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.0591 | 0.5562 | 0.5562 |
Echinococcus multilocularis | serine threonine protein kinase nrc serine threonine protein kinase gad | 0.0395 | 0.2809 | 0.2689 |
Leishmania major | protein kinase, putative | 0.0906 | 1 | 0.5 |
Loa Loa (eye worm) | AUR protein kinase | 0.0906 | 1 | 1 |
Echinococcus granulosus | Glutaredoxin protein 5 | 0.0384 | 0.2644 | 0.2521 |
Brugia malayi | serine/threonine kinase 12 | 0.0906 | 1 | 1 |
Echinococcus multilocularis | serine:threonine protein kinase 12 B | 0.0906 | 1 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.0207 | 0.0164 | 0.0164 |
Echinococcus multilocularis | nervana 2 | 0.0384 | 0.2644 | 0.2521 |
Echinococcus multilocularis | sodium calcium exchanger | 0.0572 | 0.5291 | 0.5212 |
Trichomonas vaginalis | AGC family protein kinase | 0.0591 | 0.5562 | 0.5562 |
Loa Loa (eye worm) | AUR protein kinase | 0.0906 | 1 | 1 |
Echinococcus granulosus | serine threonine protein kinase nrc | 0.0395 | 0.2809 | 0.2689 |
Echinococcus granulosus | aurora kinase A | 0.0906 | 1 | 1 |
Entamoeba histolytica | protein kinase, putative | 0.0906 | 1 | 1 |
Entamoeba histolytica | serine/threonine- protein kinase 6, putative | 0.0906 | 1 | 1 |
Echinococcus multilocularis | aurora kinase A | 0.0906 | 1 | 1 |
Echinococcus granulosus | serine:threonine protein kinase 12 B | 0.0906 | 1 | 1 |
Loa Loa (eye worm) | AGC/RSK/P70 protein kinase | 0.0591 | 0.5562 | 0.5488 |
Entamoeba histolytica | protein kinase , putative | 0.0906 | 1 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.0207 | 0.0164 | 0.0164 |
Echinococcus granulosus | serine/threonine protein kinase | 0.0395 | 0.2809 | 0.2689 |
Trichomonas vaginalis | AGC family protein kinase | 0.0591 | 0.5562 | 0.5562 |
Toxoplasma gondii | aurora kinase | 0.0906 | 1 | 1 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.0395 | 0.2809 | 0.2689 |
Entamoeba histolytica | serine/threonine protein kinase 6, putative | 0.0906 | 1 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.0591 | 0.5562 | 0.5562 |
Trichomonas vaginalis | AGC family protein kinase | 0.0906 | 1 | 1 |
Schistosoma mansoni | serine/threonine-protein kinase | 0.0395 | 0.2809 | 0.2689 |
Giardia lamblia | Aurora kinase | 0.0906 | 1 | 1 |
Echinococcus granulosus | calcium:calmodulin dependent protein kinase | 0.0395 | 0.2809 | 0.2689 |
Loa Loa (eye worm) | AGC/AKT protein kinase | 0.0591 | 0.5562 | 0.5488 |
Echinococcus granulosus | nervana 2 | 0.0384 | 0.2644 | 0.2521 |
Echinococcus multilocularis | Glutaredoxin protein 5 | 0.0384 | 0.2644 | 0.2521 |
Trichomonas vaginalis | AGC family protein kinase | 0.0207 | 0.0164 | 0.0164 |
Brugia malayi | p70 ribosomal S6 kinase beta | 0.0591 | 0.5562 | 0.5488 |
Entamoeba histolytica | protein kinase, putative | 0.0591 | 0.5562 | 0.5488 |
Trypanosoma brucei | aurora B kinase | 0.0906 | 1 | 1 |
Echinococcus multilocularis | rac serine:threonine kinase | 0.0395 | 0.2809 | 0.2689 |
Schistosoma mansoni | serine/threonine-protein kinase | 0.0395 | 0.2809 | 0.2689 |
Plasmodium falciparum | serine/threonine protein kinase, putative | 0.0906 | 1 | 1 |
Echinococcus granulosus | sodium:potassium dependent atpase beta subunit | 0.0384 | 0.2644 | 0.2521 |
Entamoeba histolytica | protein kinase 2, putative | 0.0395 | 0.2809 | 0.2689 |
Echinococcus multilocularis | nervana 2 | 0.0384 | 0.2644 | 0.2521 |
Trichomonas vaginalis | AGC family protein kinase | 0.0207 | 0.0164 | 0.0164 |
Entamoeba histolytica | protein kinase, putative | 0.0591 | 0.5562 | 0.5488 |
Schistosoma mansoni | protein kinase | 0.0906 | 1 | 1 |
Plasmodium vivax | serine/threonine protein kinase 6, putative | 0.0906 | 1 | 1 |
Entamoeba histolytica | protein kinase domain containing protein | 0.0906 | 1 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.0906 | 1 | 1 |
Brugia malayi | Sodium/calcium exchanger protein | 0.0229 | 0.0464 | 0.0305 |
Schistosoma mansoni | sodium/calcium exchanger | 0.0572 | 0.5291 | 0.5212 |
Trypanosoma cruzi | aurora B kinase, putative | 0.0906 | 1 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.0906 | 1 | 1 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.0395 | 0.2809 | 0.2689 |
Loa Loa (eye worm) | solute carrier family 8 | 0.0572 | 0.5291 | 0.5212 |
Trichomonas vaginalis | AGC family protein kinase | 0.0591 | 0.5562 | 0.5562 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
GI50 (functional) | -4.707 | PUBCHEM_BIOASSAY: NCI human tumor cell line growth inhibition assay. Data for the DU-145 Prostate cell line. (Class of assay: confirmatory) | ChEMBL. | No reference |
GI50 (functional) | -4.619 | PUBCHEM_BIOASSAY: NCI human tumor cell line growth inhibition assay. Data for the HOP-92 Non-Small Cell Lung cell line. (Class of assay: confirmatory) | ChEMBL. | No reference |
GI50 (functional) | -4.507 | PUBCHEM_BIOASSAY: NCI human tumor cell line growth inhibition assay. Data for the SF-539 Central Nervous System cell line. (Class of assay: confirmatory) | ChEMBL. | No reference |
GI50 (functional) | -4.47 | PUBCHEM_BIOASSAY: NCI human tumor cell line growth inhibition assay. Data for the MDA-N Breast cell line. (Class of assay: confirmatory) | ChEMBL. | No reference |
GI50 (functional) | -4.409 | PUBCHEM_BIOASSAY: NCI human tumor cell line growth inhibition assay. Data for the SN12C Renal cell line. (Class of assay: confirmatory) | ChEMBL. | No reference |
GI50 (functional) | -4.296 | PUBCHEM_BIOASSAY: NCI human tumor cell line growth inhibition assay. Data for the NCI-H23 Non-Small Cell Lung cell line. (Class of assay: confirmatory) | ChEMBL. | No reference |
GI50 (functional) | -4 | PUBCHEM_BIOASSAY: NCI human tumor cell line growth inhibition assay. Data for the UO-31 Renal cell line. (Class of assay: confirmatory) | ChEMBL. | No reference |
GI50 (functional) | -4 | PUBCHEM_BIOASSAY: NCI human tumor cell line growth inhibition assay. Data for the ACHN Renal cell line. (Class of assay: confirmatory) | ChEMBL. | No reference |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.