Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Trichomonas vaginalis | phosphatidylinositol 3-kinase catalytic subunit gamma, putative | 0.118017 | 0.769847 | 1 |
Loa Loa (eye worm) | phosphatidylinositol 3 | 0.12615 | 0.836844 | 1 |
Brugia malayi | Phosphatidylinositol 3- and 4-kinase family protein | 0.0890817 | 0.531505 | 0.678773 |
Entamoeba histolytica | phosphatidylinositol 3-kinase, putative | 0.0581228 | 0.276491 | 0.225291 |
Trichomonas vaginalis | phosphatidylinositol 3-kinase catalytic subunit alpha, beta, delta, putative | 0.0876456 | 0.519675 | 0.607159 |
Brugia malayi | Phosphatidylinositol 3- and 4-kinase family protein | 0.0407053 | 0.133019 | 0.14171 |
Entamoeba histolytica | hypothetical protein | 0.0982094 | 0.606692 | 0.7438 |
Trichomonas vaginalis | phopsphatidylinositol 3-kinase, drosophila, putative | 0.118017 | 0.769847 | 1 |
Entamoeba histolytica | phosphatidylinositol 3-kinase, putative | 0.0512691 | 0.220035 | 0.13664 |
Trichomonas vaginalis | phosphatidylinositol 3-kinase class, putative | 0.0876456 | 0.519675 | 0.607159 |
Brugia malayi | Phosphatidylinositol 3- and 4-kinase family protein | 0.118017 | 0.769847 | 1 |
Entamoeba histolytica | phosphatidylinositol 3-kinase, putative | 0.0982094 | 0.606692 | 0.7438 |
Loa Loa (eye worm) | hypothetical protein | 0.0884938 | 0.526663 | 0.5825 |
Trypanosoma cruzi | phosphatidylinositol 3-kinase 2, putative | 0.118017 | 0.769847 | 1 |
Trypanosoma cruzi | phosphatidylinositol 3-kinase 2, putative | 0.118017 | 0.769847 | 1 |
Giardia lamblia | Phosphoinositide-3-kinase, catalytic, alpha polypeptide | 0.0678384 | 0.356519 | 1 |
Trichomonas vaginalis | phosphatidylinositol kinase, putative | 0.118017 | 0.769847 | 1 |
Entamoeba histolytica | phosphatidylinositol 3-kinase 1, putative | 0.113267 | 0.730724 | 0.938566 |
Echinococcus granulosus | phosphatidylinositol 45 bisphosphate 3 kinase | 0.145957 | 1 | 1 |
Trypanosoma cruzi | phosphatidylinositol 3-kinase vps34-like | 0.0407053 | 0.133019 | 0.0578787 |
Schistosoma mansoni | phosphatidylinositol-45-bisphosphate 3-kinase catalytic subunit alpha PI3K | 0.145957 | 1 | 1 |
Trypanosoma brucei | phosphatidylinositol 3-kinase, putative | 0.0407053 | 0.133019 | 0.5 |
Echinococcus multilocularis | phosphatidylinositol 4,5 bisphosphate 3 kinase | 0.145957 | 1 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0469402 | 0.184377 | 0.121787 |
Entamoeba histolytica | phosphatidylinositol 3-kinase, putative | 0.118017 | 0.769847 | 1 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
EC50 (functional) | = 0.18 uM | Antimalarial activity against Plasmodium falciparum 3D7 assessed as inhibition of parasite growth | ChEMBL. | 23313245 |
Species name | Source | Reference | Is orphan |
---|---|---|---|
Plasmodium falciparum | ChEMBL23 | 23313245 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.