Species | Target name | Source | Bibliographic reference |
---|---|---|---|
Homo sapiens | parathyroid hormone 1 receptor | Starlite/ChEMBL | No references |
Species | Potential target | Known druggable target/s | Ortholog Group |
---|---|---|---|
Schistosoma japonicum | ko:K04588 secretin receptor, putative | Get druggable targets OG5_139196 | All targets in OG5_139196 |
Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Echinococcus multilocularis | casein kinase ii subunit alpha | 0.6373 | 1 | 1 |
Entamoeba histolytica | casein kinase II regulatory subunit family protein | 0.3472 | 0.5404 | 0.4586 |
Trichomonas vaginalis | casein kinase II beta chain, putative | 0.3472 | 0.5404 | 0.4586 |
Brugia malayi | Csnk2b protein | 0.3472 | 0.5404 | 0.5404 |
Trypanosoma cruzi | casein kinase II, putative | 0.6373 | 1 | 1 |
Trypanosoma brucei | Casein kinase II | 0.6373 | 1 | 1 |
Plasmodium vivax | casein kinase 2, alpha subunit, putative | 0.6373 | 1 | 1 |
Trichomonas vaginalis | casein kinase II beta chain, putative | 0.3472 | 0.5404 | 0.4586 |
Trichomonas vaginalis | CMGC family protein kinase | 0.6373 | 1 | 1 |
Trichomonas vaginalis | casein kinase II beta chain, putative | 0.3472 | 0.5404 | 0.4586 |
Loa Loa (eye worm) | Csnk2b protein | 0.3472 | 0.5404 | 0.5404 |
Trichomonas vaginalis | CMGC family protein kinase | 0.6373 | 1 | 1 |
Trichomonas vaginalis | casein kinase II beta chain, putative | 0.3472 | 0.5404 | 0.4586 |
Trichomonas vaginalis | CMGC family protein kinase | 0.6373 | 1 | 1 |
Entamoeba histolytica | casein kinase II regulatory subunit family protein | 0.3472 | 0.5404 | 0.4586 |
Onchocerca volvulus | Casein kinase II subunit beta homolog | 0.3472 | 0.5404 | 0.5 |
Onchocerca volvulus | Casein kinase II subunit beta homolog | 0.3472 | 0.5404 | 0.5 |
Trichomonas vaginalis | casein kinase II beta chain, putative | 0.3472 | 0.5404 | 0.4586 |
Giardia lamblia | Kinase, CMGC CK2 | 0.6373 | 1 | 1 |
Entamoeba histolytica | protein kinase domain containing protein | 0.6373 | 1 | 1 |
Entamoeba histolytica | casein kinase, putative | 0.6373 | 1 | 1 |
Leishmania major | casein kinase II, putative | 0.6373 | 1 | 1 |
Trichomonas vaginalis | CMGC family protein kinase | 0.6373 | 1 | 1 |
Loa Loa (eye worm) | casein kinase II | 0.1014 | 0.1511 | 0.1511 |
Giardia lamblia | Casein kinase II beta chain | 0.3472 | 0.5404 | 0.4586 |
Brugia malayi | casein kinase II, putaitve | 0.1014 | 0.1511 | 0.1511 |
Schistosoma mansoni | protein kinase | 0.6373 | 1 | 1 |
Loa Loa (eye worm) | CMGC/CK2 protein kinase | 0.6373 | 1 | 1 |
Trichomonas vaginalis | casein kinase II beta chain, putative | 0.3472 | 0.5404 | 0.4586 |
Trichomonas vaginalis | casein kinase II beta chain, putative | 0.3472 | 0.5404 | 0.4586 |
Trichomonas vaginalis | casein kinase II beta chain, putative | 0.3472 | 0.5404 | 0.4586 |
Trichomonas vaginalis | CMGC family protein kinase | 0.6373 | 1 | 1 |
Echinococcus granulosus | casein kinase ii subunit alpha | 0.6373 | 1 | 1 |
Trichomonas vaginalis | casein kinase II beta chain, putative | 0.3472 | 0.5404 | 0.4586 |
Trichomonas vaginalis | casein kinase II beta chain, putative | 0.3472 | 0.5404 | 0.4586 |
Entamoeba histolytica | casein kinase II regulatory subunit family protein | 0.3472 | 0.5404 | 0.4586 |
Trichomonas vaginalis | casein kinase II beta chain, putative | 0.3472 | 0.5404 | 0.4586 |
Trichomonas vaginalis | casein kinase II beta chain, putative | 0.3472 | 0.5404 | 0.4586 |
Trichomonas vaginalis | casein kinase II beta chain, putative | 0.3472 | 0.5404 | 0.4586 |
Trichomonas vaginalis | casein kinase II beta chain, putative | 0.3472 | 0.5404 | 0.4586 |
Plasmodium falciparum | casein kinase 2, alpha subunit | 0.6373 | 1 | 1 |
Trichomonas vaginalis | CMGC family protein kinase | 0.6373 | 1 | 1 |
Trichomonas vaginalis | casein kinase II beta chain, putative | 0.3472 | 0.5404 | 0.4586 |
Trichomonas vaginalis | CMGC family protein kinase | 0.6373 | 1 | 1 |
Plasmodium vivax | unspecified product | 0.6373 | 1 | 1 |
Toxoplasma gondii | CMGC kinase, CK2 family | 0.6373 | 1 | 1 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
Potency (functional) | 14.1254 uM | PubChem BioAssay. qHTS of PTHR Inhibitors: Primary Screen. (Class of assay: confirmatory) | ChEMBL. | No reference |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.