Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Trichomonas vaginalis | casein kinase II beta chain, putative | 0.7484 | 0.5447 | 0.4716 |
Trichomonas vaginalis | CMGC family protein kinase | 1.3421 | 1 | 1 |
Loa Loa (eye worm) | CMGC/CK2 protein kinase | 1.3421 | 1 | 1 |
Schistosoma mansoni | casein kinase II beta subunit | 0.7484 | 0.5447 | 0.3057 |
Schistosoma mansoni | protein kinase | 1.3421 | 1 | 1 |
Trichomonas vaginalis | casein kinase II beta chain, putative | 0.7484 | 0.5447 | 0.4716 |
Loa Loa (eye worm) | CAMK/PIM protein kinase | 0.487 | 0.3442 | 0.3015 |
Giardia lamblia | Casein kinase II beta chain | 0.7484 | 0.5447 | 0.4716 |
Entamoeba histolytica | casein kinase, putative | 1.3421 | 1 | 1 |
Trichomonas vaginalis | casein kinase II beta chain, putative | 0.7484 | 0.5447 | 0.4716 |
Echinococcus granulosus | casein kinase ii subunit beta | 0.7484 | 0.5447 | 0.3057 |
Echinococcus multilocularis | casein kinase ii subunit alpha | 1.3421 | 1 | 1 |
Trichomonas vaginalis | casein kinase II beta chain, putative | 0.7484 | 0.5447 | 0.4716 |
Loa Loa (eye worm) | casein kinase II | 0.2186 | 0.1383 | 0.0822 |
Trichomonas vaginalis | casein kinase II beta chain, putative | 0.7484 | 0.5447 | 0.4716 |
Trichomonas vaginalis | CMGC family protein kinase | 1.3421 | 1 | 1 |
Trichomonas vaginalis | CMGC family protein kinase | 1.3421 | 1 | 1 |
Plasmodium vivax | casein kinase 2, alpha subunit, putative | 1.3421 | 1 | 1 |
Brugia malayi | Serine/threonine-protein kinase Pim-3 | 0.487 | 0.3442 | 0.3333 |
Trichomonas vaginalis | CMGC family protein kinase | 1.3421 | 1 | 1 |
Echinococcus multilocularis | casein kinase ii subunit beta | 0.7484 | 0.5447 | 0.3057 |
Onchocerca volvulus | Casein kinase II subunit beta homolog | 0.7484 | 0.5447 | 1 |
Trichomonas vaginalis | casein kinase II beta chain, putative | 0.7484 | 0.5447 | 0.4716 |
Giardia lamblia | Kinase, CMGC CK2 | 1.3421 | 1 | 1 |
Trichomonas vaginalis | casein kinase II beta chain, putative | 0.7484 | 0.5447 | 0.4716 |
Loa Loa (eye worm) | CAMK/PIM protein kinase | 0.487 | 0.3442 | 0.3015 |
Plasmodium vivax | unspecified product | 1.3421 | 1 | 1 |
Plasmodium falciparum | casein kinase 2, alpha subunit | 1.3421 | 1 | 1 |
Entamoeba histolytica | protein kinase domain containing protein | 1.3421 | 1 | 1 |
Trichomonas vaginalis | CMGC family protein kinase | 1.3421 | 1 | 1 |
Entamoeba histolytica | casein kinase II regulatory subunit family protein | 0.7484 | 0.5447 | 0.4716 |
Trypanosoma brucei | Casein kinase II | 1.3421 | 1 | 1 |
Mycobacterium tuberculosis | Probable epoxide hydrolase EphA (epoxide hydratase) (arene-oxide hydratase) | 0.0383 | 0 | 0.5 |
Trichomonas vaginalis | casein kinase II beta chain, putative | 0.7484 | 0.5447 | 0.4716 |
Trichomonas vaginalis | CMGC family protein kinase | 1.3421 | 1 | 1 |
Trichomonas vaginalis | casein kinase II beta chain, putative | 0.7484 | 0.5447 | 0.4716 |
Trichomonas vaginalis | casein kinase II beta chain, putative | 0.7484 | 0.5447 | 0.4716 |
Onchocerca volvulus | Casein kinase II subunit beta homolog | 0.7484 | 0.5447 | 1 |
Trichomonas vaginalis | casein kinase II beta chain, putative | 0.7484 | 0.5447 | 0.4716 |
Trichomonas vaginalis | casein kinase II beta chain, putative | 0.7484 | 0.5447 | 0.4716 |
Entamoeba histolytica | casein kinase II regulatory subunit family protein | 0.7484 | 0.5447 | 0.4716 |
Trichomonas vaginalis | CMGC family protein kinase | 1.3421 | 1 | 1 |
Echinococcus granulosus | casein kinase ii subunit alpha | 1.3421 | 1 | 1 |
Trypanosoma cruzi | casein kinase II, putative | 1.3421 | 1 | 1 |
Mycobacterium ulcerans | epoxide hydrolase EphA | 0.0383 | 0 | 0.5 |
Leishmania major | casein kinase II, putative | 1.3421 | 1 | 1 |
Brugia malayi | Csnk2b protein | 0.7484 | 0.5447 | 0.5371 |
Brugia malayi | casein kinase II, putaitve | 0.2186 | 0.1383 | 0.124 |
Toxoplasma gondii | CMGC kinase, CK2 family | 1.3421 | 1 | 1 |
Trichomonas vaginalis | casein kinase II beta chain, putative | 0.7484 | 0.5447 | 0.4716 |
Entamoeba histolytica | casein kinase II regulatory subunit family protein | 0.7484 | 0.5447 | 0.4716 |
Trichomonas vaginalis | casein kinase II beta chain, putative | 0.7484 | 0.5447 | 0.4716 |
Brugia malayi | Protein kinase domain containing protein | 0.487 | 0.3442 | 0.3333 |
Loa Loa (eye worm) | Csnk2b protein | 0.7484 | 0.5447 | 0.515 |
Onchocerca volvulus | Serine\/threonine protein kinase homolog | 0.487 | 0.3442 | 0.5847 |
Trichomonas vaginalis | casein kinase II beta chain, putative | 0.7484 | 0.5447 | 0.4716 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
IC50 (functional) | > 10 uM | Cytotoxicity against human SNU387 cells after 48 hrs by MTT assay | ChEMBL. | 23701597 |
Species name | Source | Reference | Is orphan |
---|---|---|---|
Homo sapiens | ChEMBL23 | 23701597 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.