Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Entamoeba histolytica | hypothetical protein | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | hypothetical protein | 0.0151 | 0 | 0.5 |
Mycobacterium tuberculosis | Probable transmembrane carbonic anhydrase (carbonate dehydratase) (carbonic dehydratase) | 0.0326 | 0.0188 | 0.0669 |
Entamoeba histolytica | protein kinase domain containing protein | 0.0151 | 0 | 0.5 |
Toxoplasma gondii | calcium dependent protein kinase CDPK8 | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | protein kinase domain containing protein | 0.0151 | 0 | 0.5 |
Plasmodium vivax | protein kinase, putative | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | protein kinase, putative | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | tyrosine kinase, putative | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | tyrosin kinase, putative | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | receptor protein kinase, putative | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | SH2-protein kinase domain containing protein | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | protein kinase domain containing protein | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | tyrosine kinase, putative | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | protein tyrosine kinase domain-containing protein | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | protein tyrosine kinase domain-containing protein | 0.0151 | 0 | 0.5 |
Onchocerca volvulus | Putative sulfate transporter | 0.0233 | 0.0089 | 1 |
Entamoeba histolytica | tyrosine kinase, putative | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | protein kinase domain containing protein | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | serine/threonine kinase, putative | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | protein kinase with ankyrin repeats, putative | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | hypothetical protein | 0.0151 | 0 | 0.5 |
Plasmodium falciparum | tyrosine kinase-like protein | 0.0151 | 0 | 0.5 |
Onchocerca volvulus | 0.0233 | 0.0089 | 1 | |
Entamoeba histolytica | protein tyrosine kinase domain-containing protein | 0.0151 | 0 | 0.5 |
Loa Loa (eye worm) | eukaryotic-type carbonic anhydrase | 0.0203 | 0.0056 | 0.0057 |
Entamoeba histolytica | hypothetical protein | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | ankyrin repeat protein | 0.0151 | 0 | 0.5 |
Mycobacterium leprae | Probable transmembrane transport protein | 0.0269 | 0.0128 | 0.5 |
Entamoeba histolytica | protein kinase domain containing protein | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | hypothetical protein | 0.0151 | 0 | 0.5 |
Plasmodium vivax | tyrosine kinase-like protein, putative | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | tyrosin kinase, putative | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | protein kinase, putative | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | protein tyrosine kinase domain-containing protein | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | protein kinase, putative | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | tyrosin kinase, putative | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | protein tyrosine kinase domain-containing protein | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | tyrosine kinase, putative | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | protein kinase domain containing protein | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | tyrosine kinase, putative | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | tyrosine kinase, putative | 0.0151 | 0 | 0.5 |
Toxoplasma gondii | Tyrosine kinase-like (TKL) protein | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | protein kinase, putative | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | leucine-rich repeat domain-containing protein | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | protein kinase, putative | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | protein kinase domain containing protein | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | tyrosine kinase, putative | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | protein kinase domain containing protein | 0.0151 | 0 | 0.5 |
Schistosoma mansoni | carbonic anhydrase II (carbonate dehydratase II) | 0.0203 | 0.0056 | 0.0056 |
Entamoeba histolytica | protein kinase, putative | 0.0151 | 0 | 0.5 |
Plasmodium vivax | tyrosine kinase-like protein, putative | 0.0151 | 0 | 0.5 |
Plasmodium falciparum | tyrosine kinase-like protein | 0.0151 | 0 | 0.5 |
Mycobacterium ulcerans | carbonic anhydrase | 0.1168 | 0.1093 | 0.5 |
Schistosoma mansoni | carbonic anhydrase II (carbonate dehydratase II) | 0.0203 | 0.0056 | 0.0056 |
Plasmodium falciparum | protein kinase, putative | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | protein kinase domain containing protein | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | hypothetical protein | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | serine/threonine kinase, putative | 0.0151 | 0 | 0.5 |
Toxoplasma gondii | protein kinase domain-containing protein | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | protein kinase, putative | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | protein kinase domain containing protein | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | protein tyrosine kinase domain-containing protein | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | protein kinase domain containing protein | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | protein kinase domain containing protein | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | tyrosine kinase, putative | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | receptor protein kinase, putative | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | tyrosine kinase, putative | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | hypothetical protein | 0.0151 | 0 | 0.5 |
Plasmodium falciparum | protein kinase, putative | 0.0151 | 0 | 0.5 |
Toxoplasma gondii | protein kinase | 0.0151 | 0 | 0.5 |
Giardia lamblia | Kinase | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | protein kinase, putative | 0.0151 | 0 | 0.5 |
Trypanosoma cruzi | carbonic anhydrase-like protein, putative | 0.0203 | 0.0056 | 1 |
Entamoeba histolytica | hypothetical protein, conserved | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | serine/threonine kinase, putative | 0.0151 | 0 | 0.5 |
Brugia malayi | Putative carbonic anhydrase 5 precursor | 0.0203 | 0.0056 | 0.0057 |
Loa Loa (eye worm) | hypothetical protein | 0.9304 | 0.9838 | 1 |
Entamoeba histolytica | tyrosine kinase, putative | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | protein kinase, putative | 0.0151 | 0 | 0.5 |
Trypanosoma brucei | carbonic anhydrase-like protein | 0.0203 | 0.0056 | 1 |
Brugia malayi | Eukaryotic-type carbonic anhydrase family protein | 0.0203 | 0.0056 | 0.0057 |
Entamoeba histolytica | protein kinase, putative | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | tyrosine kinase, putative | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | serine/threonine kinase, putative | 0.0151 | 0 | 0.5 |
Brugia malayi | Protein kinase domain containing protein | 0.9304 | 0.9838 | 1 |
Entamoeba histolytica | protein kinase, putative | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | hypothetical protein | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | tyrosine kinase, putative | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | protein kinase domain containing protein | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | protein kinase, putative | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | serine/threonine kinase, putative | 0.0151 | 0 | 0.5 |
Giardia lamblia | Protein 21.1 | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | hypothetical protein | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | protein kinase domain containing protein | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | protein kinase domain containing protein | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | protein tyrosine kinase domain-containing protein | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | serine/threonine kinase, putative | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | hypothetical protein | 0.0151 | 0 | 0.5 |
Toxoplasma gondii | Tyrosine kinase-like (TKL) protein | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | protein kinase, putative | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | protein tyrosine kinase domain-containing protein | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | protein kinase domain containing protein | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | protein kinase, putative | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | hypothetical protein | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | protein kinase domain containing protein | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | protein kinase domain containing protein | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | protein tyrosine kinase domain-containing protein | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | protein kinase, putative | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | protein kinase, putative | 0.0151 | 0 | 0.5 |
Echinococcus multilocularis | mitogen activated protein kinase kinase kinase | 0.9304 | 0.9838 | 1 |
Entamoeba histolytica | tyrosine kinase, putative | 0.0151 | 0 | 0.5 |
Plasmodium falciparum | protein kinase, putative | 0.0151 | 0 | 0.5 |
Giardia lamblia | Kinase, NEK | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | protein kinase, putative | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | protein tyrosine kinase domain-containing protein | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | tyrosine kinase, putative | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | protein kinase, putative | 0.0151 | 0 | 0.5 |
Loa Loa (eye worm) | TKL/MLK/LZK protein kinase | 0.9304 | 0.9838 | 1 |
Entamoeba histolytica | tyrosine kinase, putative | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | protein kinase domain containing protein | 0.0151 | 0 | 0.5 |
Leishmania major | carbonic anhydrase-like protein | 0.0203 | 0.0056 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.9304 | 0.9838 | 1 |
Giardia lamblia | Kinase, NEK | 0.0151 | 0 | 0.5 |
Trichomonas vaginalis | conserved hypothetical protein | 0.1168 | 0.1093 | 1 |
Echinococcus granulosus | mitogen activated protein kinase kinase kinase | 0.9304 | 0.9838 | 1 |
Entamoeba histolytica | cysteine surface protein, putative | 0.0151 | 0 | 0.5 |
Trichomonas vaginalis | conserved hypothetical protein | 0.1168 | 0.1093 | 1 |
Toxoplasma gondii | STE kinase | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | tyrosine kinase, putative | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | protein tyrosine kinase domain-containing protein | 0.0151 | 0 | 0.5 |
Echinococcus granulosus | carbonic anhydrase II | 0.0203 | 0.0056 | 0.0057 |
Echinococcus multilocularis | carbonic anhydrase II | 0.0203 | 0.0056 | 0.0057 |
Entamoeba histolytica | protein kinase domain containing protein | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | tyrosine- protein kinase 2, putative | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | tyrosin kinase, putative | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | protein tyrosine kinase domain-containing protein | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | protein kinase, putative | 0.0151 | 0 | 0.5 |
Trypanosoma cruzi | carbonic anhydrase-like protein, putative | 0.0203 | 0.0056 | 1 |
Entamoeba histolytica | protein kinase domain containing protein | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | tyrosine kinase, putative | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | protein tyrosine kinase domain-containing protein | 0.0151 | 0 | 0.5 |
Mycobacterium tuberculosis | Beta-carbonic anhydrase | 0.1111 | 0.1032 | 1 |
Entamoeba histolytica | protein kinase domain containing protein | 0.0151 | 0 | 0.5 |
Entamoeba histolytica | ankyrin repeat protein | 0.0151 | 0 | 0.5 |
Loa Loa (eye worm) | carbonic anhydrase 3 | 0.0203 | 0.0056 | 0.0057 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
IZ (functional) | = 11 mm | Antibacterial activity against Escherichia coli ATCC 25922 assessed as growth inhibition at 1.56 to 25 ug/mL | ChEMBL. | No reference |
MIC (functional) | = 12.5 ug ml-1 | Antibacterial activity against Escherichia coli ATCC 25922 assessed as growth inhibition by serial plate dilution method | ChEMBL. | No reference |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.