Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Trichomonas vaginalis | casein kinase II beta chain, putative | 0.1202 | 0.4586 | 0.4586 |
Leishmania major | casein kinase II, putative | 0.2207 | 1 | 1 |
Echinococcus granulosus | casein kinase ii subunit alpha | 0.2207 | 1 | 1 |
Schistosoma mansoni | protein kinase | 0.2207 | 1 | 1 |
Trichomonas vaginalis | casein kinase II beta chain, putative | 0.1202 | 0.4586 | 0.4586 |
Onchocerca volvulus | Casein kinase II subunit beta homolog | 0.1202 | 0.4586 | 0.5 |
Giardia lamblia | Casein kinase II beta chain | 0.1202 | 0.4586 | 0.4586 |
Trichomonas vaginalis | casein kinase II beta chain, putative | 0.1202 | 0.4586 | 0.4586 |
Trichomonas vaginalis | casein kinase II beta chain, putative | 0.1202 | 0.4586 | 0.4586 |
Trichomonas vaginalis | casein kinase II beta chain, putative | 0.1202 | 0.4586 | 0.4586 |
Trichomonas vaginalis | CMGC family protein kinase | 0.2207 | 1 | 1 |
Trichomonas vaginalis | CMGC family protein kinase | 0.2207 | 1 | 1 |
Plasmodium vivax | casein kinase 2, alpha subunit, putative | 0.2207 | 1 | 1 |
Giardia lamblia | Kinase, CMGC CK2 | 0.2207 | 1 | 1 |
Trypanosoma cruzi | casein kinase II, putative | 0.2207 | 1 | 1 |
Trichomonas vaginalis | CMGC family protein kinase | 0.2207 | 1 | 1 |
Trichomonas vaginalis | casein kinase II beta chain, putative | 0.1202 | 0.4586 | 0.4586 |
Plasmodium vivax | unspecified product | 0.2207 | 1 | 1 |
Trichomonas vaginalis | CMGC family protein kinase | 0.2207 | 1 | 1 |
Onchocerca volvulus | Casein kinase II subunit beta homolog | 0.1202 | 0.4586 | 0.5 |
Trichomonas vaginalis | casein kinase II beta chain, putative | 0.1202 | 0.4586 | 0.4586 |
Trichomonas vaginalis | casein kinase II beta chain, putative | 0.1202 | 0.4586 | 0.4586 |
Trichomonas vaginalis | casein kinase II beta chain, putative | 0.1202 | 0.4586 | 0.4586 |
Plasmodium falciparum | casein kinase 2, alpha subunit | 0.2207 | 1 | 1 |
Trichomonas vaginalis | CMGC family protein kinase | 0.2207 | 1 | 1 |
Entamoeba histolytica | casein kinase II regulatory subunit family protein | 0.1202 | 0.4586 | 0.4586 |
Trichomonas vaginalis | casein kinase II beta chain, putative | 0.1202 | 0.4586 | 0.4586 |
Brugia malayi | Csnk2b protein | 0.1202 | 0.4586 | 0.4586 |
Entamoeba histolytica | protein kinase domain containing protein | 0.2207 | 1 | 1 |
Trichomonas vaginalis | casein kinase II beta chain, putative | 0.1202 | 0.4586 | 0.4586 |
Entamoeba histolytica | casein kinase II regulatory subunit family protein | 0.1202 | 0.4586 | 0.4586 |
Trichomonas vaginalis | CMGC family protein kinase | 0.2207 | 1 | 1 |
Trichomonas vaginalis | casein kinase II beta chain, putative | 0.1202 | 0.4586 | 0.4586 |
Loa Loa (eye worm) | CMGC/CK2 protein kinase | 0.2207 | 1 | 1 |
Loa Loa (eye worm) | Csnk2b protein | 0.1202 | 0.4586 | 0.4586 |
Entamoeba histolytica | casein kinase, putative | 0.2207 | 1 | 1 |
Toxoplasma gondii | CMGC kinase, CK2 family | 0.2207 | 1 | 1 |
Trichomonas vaginalis | CMGC family protein kinase | 0.2207 | 1 | 1 |
Trichomonas vaginalis | casein kinase II beta chain, putative | 0.1202 | 0.4586 | 0.4586 |
Trichomonas vaginalis | casein kinase II beta chain, putative | 0.1202 | 0.4586 | 0.4586 |
Trichomonas vaginalis | casein kinase II beta chain, putative | 0.1202 | 0.4586 | 0.4586 |
Entamoeba histolytica | casein kinase II regulatory subunit family protein | 0.1202 | 0.4586 | 0.4586 |
Trypanosoma brucei | Casein kinase II | 0.2207 | 1 | 1 |
Echinococcus multilocularis | casein kinase ii subunit alpha | 0.2207 | 1 | 1 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
log(1/MIC) (functional) | = -0.716 | Antibacterial activity against Mycobacterium tuberculosis H37Rv assessed as growth inhibition by two-fold serial dilution method | ChEMBL. | 817022 |
log(1/MIC) (functional) | = 0.10453 | Antitubercular activity against Mycobacterium tuberculosis H37Rv | ChEMBL. | 24246731 |
MIC (functional) | = 0.79 ug ml-1 | Antitubercular activity against Mycobacterium tuberculosis H37Rv | ChEMBL. | 24246731 |
MIC (functional) | = 5.2 uM | Antitubercular activity against Mycobacterium tuberculosis H37Rv ATCC 27294 by BACTEC 960 assay | ChEMBL. | 24836065 |
MIC (functional) | = 5.2 umol/L | Antibacterial activity against Mycobacterium tuberculosis H37Rv assessed as growth inhibition by two-fold serial dilution method | ChEMBL. | 817022 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.