Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Brugia malayi | hypothetical protein | 0.0021 | 0.1049 | 0.1049 |
Brugia malayi | follicle stimulating hormone receptor | 0.0021 | 0.1049 | 0.1049 |
Giardia lamblia | Cytidine deaminase | 0.0118 | 1 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Entamoeba histolytica | cytidine deaminase, putative | 0.0118 | 1 | 0.5 |
Brugia malayi | G protein-coupled receptor | 0.0021 | 0.1049 | 0.1049 |
Loa Loa (eye worm) | G-protein coupled receptor | 0.0021 | 0.1049 | 1 |
Brugia malayi | hypothetical protein | 0.0021 | 0.1049 | 0.1049 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Loa Loa (eye worm) | follicle stimulating hormone receptor | 0.0021 | 0.1049 | 1 |
Trichomonas vaginalis | cytidine deaminase, putative | 0.0118 | 1 | 1 |
Trypanosoma cruzi | cytidine deaminase-like protein, putative | 0.0118 | 1 | 1 |
Brugia malayi | hypothetical protein | 0.0021 | 0.1049 | 0.1049 |
Brugia malayi | hypothetical protein | 0.0021 | 0.1049 | 0.1049 |
Echinococcus granulosus | cytidine deaminase | 0.0118 | 1 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Brugia malayi | hypothetical protein | 0.0021 | 0.1049 | 0.1049 |
Brugia malayi | putative neuropeptide receptor NPR1 | 0.0021 | 0.1049 | 0.1049 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Trypanosoma brucei | hypothetical protein, conserved | 0.0024 | 0.133 | 0.133 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Brugia malayi | Dopamine receptor protein 1, putative (partial) | 0.0021 | 0.1049 | 0.1049 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Loa Loa (eye worm) | unidentified vitellogenin-linked transcript protein 6 | 0.0021 | 0.1049 | 1 |
Mycobacterium ulcerans | cytidine deaminase | 0.0118 | 1 | 1 |
Schistosoma mansoni | phosphoglucomutase | 0.0022 | 0.1161 | 0.0199 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Wolbachia endosymbiont of Brugia malayi | ribonuclease HI | 0.0022 | 0.1161 | 0.5 |
Schistosoma mansoni | hypothetical protein | 0.0081 | 0.6644 | 1 |
Brugia malayi | neuropeptide F receptor | 0.0021 | 0.1049 | 0.1049 |
Brugia malayi | AKH receptor | 0.0021 | 0.1049 | 0.1049 |
Brugia malayi | Serotonin receptor | 0.0021 | 0.1049 | 0.1049 |
Brugia malayi | hypothetical protein | 0.0021 | 0.1049 | 0.1049 |
Mycobacterium tuberculosis | Probable cytidine deaminase Cdd (cytidine aminohydrolase) (cytidine nucleoside deaminase) | 0.0118 | 1 | 0.5 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Leishmania major | cytidine deaminase-like protein | 0.0118 | 1 | 1 |
Schistosoma mansoni | phosphoglucomutase | 0.0022 | 0.1161 | 0.0199 |
Brugia malayi | neuropeptide F receptor | 0.0021 | 0.1049 | 0.1049 |
Leishmania major | ribonuclease H1, putative | 0.0022 | 0.1161 | 0.1161 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Onchocerca volvulus | 0.0118 | 1 | 1 | |
Trypanosoma brucei | ingi protein (ORF1) | 0.0024 | 0.133 | 0.133 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Brugia malayi | gonadotropin-releasing hormone receptor 2 | 0.0021 | 0.1049 | 0.1049 |
Trypanosoma brucei | retrotransposon hot spot protein 4 (RHS4), interrupted | 0.0024 | 0.133 | 0.133 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Brugia malayi | hypothetical protein | 0.0021 | 0.1049 | 0.1049 |
Brugia malayi | Serotonin/octopamine receptor family protein 7 | 0.0021 | 0.1049 | 0.1049 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Brugia malayi | Unidentified vitellogenin-linked transcript protein 6, putative | 0.0021 | 0.1049 | 0.1049 |
Brugia malayi | G-protein coupled receptor | 0.0021 | 0.1049 | 0.1049 |
Loa Loa (eye worm) | G-protein coupled receptor | 0.0021 | 0.1049 | 1 |
Loa Loa (eye worm) | TYRA-2 protein | 0.0021 | 0.1049 | 1 |
Trypanosoma brucei | unspecified product | 0.0024 | 0.133 | 0.133 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Loa Loa (eye worm) | neuropeptide F receptor | 0.0021 | 0.1049 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Brugia malayi | putative neuropeptide receptor | 0.0021 | 0.1049 | 0.1049 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Brugia malayi | hypothetical protein | 0.0021 | 0.1049 | 0.1049 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Brugia malayi | hypothetical protein | 0.0021 | 0.1049 | 0.1049 |
Brugia malayi | Dopamine receptor protein 2 | 0.0021 | 0.1049 | 0.1049 |
Mycobacterium leprae | PROBABLE CYTIDINE DEAMINASE CDD (CYTIDINE AMINOHYDROLASE) (CYTIDINE NUCLEOSIDE DEAMINASE) | 0.0118 | 1 | 0.5 |
Trypanosoma brucei | cytidine deaminase | 0.0118 | 1 | 1 |
Brugia malayi | RE15519p | 0.0021 | 0.1049 | 0.1049 |
Loa Loa (eye worm) | neuropeptide F receptor | 0.0021 | 0.1049 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Onchocerca volvulus | Ribonuclease H1 homolog | 0.0022 | 0.1161 | 0.0125 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Echinococcus multilocularis | ribonuclease H1 | 0.0022 | 0.1161 | 0.0125 |
Brugia malayi | Dopamine receptor protein 1 | 0.0021 | 0.1049 | 0.1049 |
Brugia malayi | GnHR receptor homolog | 0.0021 | 0.1049 | 0.1049 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Brugia malayi | G protein-coupled receptor F59B2.13 | 0.0021 | 0.1049 | 0.1049 |
Loa Loa (eye worm) | G-protein-linked acetylcholine receptor protein 2 | 0.0021 | 0.1049 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Brugia malayi | Tachykinin-like peptides receptor 99D | 0.0021 | 0.1049 | 0.1049 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Brugia malayi | RNase H family protein | 0.0022 | 0.1161 | 0.1161 |
Loa Loa (eye worm) | 5-hydroxytryptamine 2C receptor | 0.0021 | 0.1049 | 1 |
Brugia malayi | hypothetical protein | 0.0021 | 0.1049 | 0.1049 |
Loa Loa (eye worm) | melatonin receptor type 1A | 0.0021 | 0.1049 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Brugia malayi | ORL1-like opioid receptor | 0.0021 | 0.1049 | 0.1049 |
Treponema pallidum | ribonuclease H (rnhA) | 0.0022 | 0.1161 | 0.5 |
Brugia malayi | G-protein-linked acetylcholine receptor protein 2, putative | 0.0021 | 0.1049 | 0.1049 |
Brugia malayi | RNase H family protein | 0.0022 | 0.1161 | 0.1161 |
Onchocerca volvulus | 0.0118 | 1 | 1 | |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Trypanosoma brucei | ribonuclease H1 | 0.0022 | 0.1161 | 0.1161 |
Brugia malayi | sulfakinin receptor protein | 0.0021 | 0.1049 | 0.1049 |
Trypanosoma cruzi | ribonuclease H1, putative | 0.0022 | 0.1161 | 0.1161 |
Echinococcus granulosus | ribonuclease H1 | 0.0022 | 0.1161 | 0.0125 |
Schistosoma mansoni | phosphoglucomutase | 0.0022 | 0.1161 | 0.0199 |
Trypanosoma brucei | ingi protein (ORF1) | 0.0024 | 0.133 | 0.133 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Trypanosoma brucei | RNA helicase, putative | 0.0081 | 0.6644 | 0.6644 |
Brugia malayi | Melatonin receptor type 1A | 0.0021 | 0.1049 | 0.1049 |
Brugia malayi | Serotonin receptor | 0.0021 | 0.1049 | 0.1049 |
Loa Loa (eye worm) | gonadotropin-releasing hormone receptor 2 | 0.0021 | 0.1049 | 1 |
Toxoplasma gondii | cytidine and deoxycytidylate deaminase zinc-binding region domain-containing protein | 0.0118 | 1 | 1 |
Trichomonas vaginalis | cytidine deaminase, putative | 0.0118 | 1 | 1 |
Brugia malayi | G-protein coupled receptor | 0.0021 | 0.1049 | 0.1049 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Brugia malayi | RNase H family protein | 0.0022 | 0.1161 | 0.1161 |
Brugia malayi | larval opioid receptor | 0.0021 | 0.1049 | 0.1049 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Echinococcus multilocularis | cytidine deaminase | 0.0118 | 1 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Trypanosoma cruzi | cytidine deaminase-like protein | 0.0118 | 1 | 1 |
Trypanosoma cruzi | ribonuclease H1, putative | 0.0022 | 0.1161 | 0.1161 |
Brugia malayi | Dopamine receptor | 0.0021 | 0.1049 | 0.1049 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
EC50 (functional) | = 0.991 | Cytotoxicity against Homo sapiens (human) MCF7 cells | ChEMBL. | No reference |
IC50 (functional) | = -4.48 | Antiproliferative activity evaluated against MCF-7 cell line | ChEMBL. | 14741278 |
Log IC50 (functional) | = 4.48 | Antiproliferative activity evaluated against MCF-7 cell line | ChEMBL. | 14741278 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.