Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Trichomonas vaginalis | cytidine deaminase, putative | 0.0118 | 1 | 1 |
Schistosoma mansoni | phosphoglucomutase | 0.0022 | 0.1161 | 0.0199 |
Brugia malayi | Melatonin receptor type 1A | 0.0021 | 0.1049 | 0.1049 |
Schistosoma mansoni | phosphoglucomutase | 0.0022 | 0.1161 | 0.0199 |
Brugia malayi | Serotonin receptor | 0.0021 | 0.1049 | 0.1049 |
Onchocerca volvulus | 0.0118 | 1 | 1 | |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Trypanosoma brucei | ingi protein (ORF1) | 0.0024 | 0.133 | 0.133 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Loa Loa (eye worm) | TYRA-2 protein | 0.0021 | 0.1049 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Brugia malayi | hypothetical protein | 0.0021 | 0.1049 | 0.1049 |
Trypanosoma cruzi | ribonuclease H1, putative | 0.0022 | 0.1161 | 0.1161 |
Schistosoma mansoni | phosphoglucomutase | 0.0022 | 0.1161 | 0.0199 |
Brugia malayi | hypothetical protein | 0.0021 | 0.1049 | 0.1049 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Brugia malayi | neuropeptide F receptor | 0.0021 | 0.1049 | 0.1049 |
Brugia malayi | Dopamine receptor protein 2 | 0.0021 | 0.1049 | 0.1049 |
Trichomonas vaginalis | cytidine deaminase, putative | 0.0118 | 1 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Brugia malayi | hypothetical protein | 0.0021 | 0.1049 | 0.1049 |
Loa Loa (eye worm) | G-protein-linked acetylcholine receptor protein 2 | 0.0021 | 0.1049 | 1 |
Brugia malayi | ORL1-like opioid receptor | 0.0021 | 0.1049 | 0.1049 |
Brugia malayi | RNase H family protein | 0.0022 | 0.1161 | 0.1161 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Brugia malayi | larval opioid receptor | 0.0021 | 0.1049 | 0.1049 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Loa Loa (eye worm) | follicle stimulating hormone receptor | 0.0021 | 0.1049 | 1 |
Loa Loa (eye worm) | 5-hydroxytryptamine 2C receptor | 0.0021 | 0.1049 | 1 |
Trypanosoma brucei | ingi protein (ORF1) | 0.0024 | 0.133 | 0.133 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Brugia malayi | putative neuropeptide receptor NPR1 | 0.0021 | 0.1049 | 0.1049 |
Brugia malayi | neuropeptide F receptor | 0.0021 | 0.1049 | 0.1049 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Echinococcus granulosus | cytidine deaminase | 0.0118 | 1 | 1 |
Toxoplasma gondii | cytidine and deoxycytidylate deaminase zinc-binding region domain-containing protein | 0.0118 | 1 | 1 |
Trypanosoma brucei | retrotransposon hot spot protein 4 (RHS4), interrupted | 0.0024 | 0.133 | 0.133 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Brugia malayi | Serotonin receptor | 0.0021 | 0.1049 | 0.1049 |
Brugia malayi | RNase H family protein | 0.0022 | 0.1161 | 0.1161 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Trypanosoma cruzi | cytidine deaminase-like protein | 0.0118 | 1 | 1 |
Trypanosoma cruzi | cytidine deaminase-like protein, putative | 0.0118 | 1 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Trypanosoma brucei | cytidine deaminase | 0.0118 | 1 | 1 |
Brugia malayi | Tachykinin-like peptides receptor 99D | 0.0021 | 0.1049 | 0.1049 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Wolbachia endosymbiont of Brugia malayi | ribonuclease HI | 0.0022 | 0.1161 | 0.5 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Brugia malayi | Dopamine receptor | 0.0021 | 0.1049 | 0.1049 |
Brugia malayi | G-protein-linked acetylcholine receptor protein 2, putative | 0.0021 | 0.1049 | 0.1049 |
Loa Loa (eye worm) | gonadotropin-releasing hormone receptor 2 | 0.0021 | 0.1049 | 1 |
Brugia malayi | hypothetical protein | 0.0021 | 0.1049 | 0.1049 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Giardia lamblia | Cytidine deaminase | 0.0118 | 1 | 1 |
Brugia malayi | AKH receptor | 0.0021 | 0.1049 | 0.1049 |
Leishmania major | ribonuclease H1, putative | 0.0022 | 0.1161 | 0.1161 |
Brugia malayi | hypothetical protein | 0.0021 | 0.1049 | 0.1049 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Loa Loa (eye worm) | melatonin receptor type 1A | 0.0021 | 0.1049 | 1 |
Mycobacterium ulcerans | cytidine deaminase | 0.0118 | 1 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Brugia malayi | RE15519p | 0.0021 | 0.1049 | 0.1049 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Echinococcus multilocularis | ribonuclease H1 | 0.0022 | 0.1161 | 0.0125 |
Loa Loa (eye worm) | neuropeptide F receptor | 0.0021 | 0.1049 | 1 |
Loa Loa (eye worm) | neuropeptide F receptor | 0.0021 | 0.1049 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Onchocerca volvulus | 0.0118 | 1 | 1 | |
Brugia malayi | G protein-coupled receptor F59B2.13 | 0.0021 | 0.1049 | 0.1049 |
Schistosoma mansoni | hypothetical protein | 0.0081 | 0.6644 | 1 |
Trypanosoma cruzi | ribonuclease H1, putative | 0.0022 | 0.1161 | 0.1161 |
Brugia malayi | RNase H family protein | 0.0022 | 0.1161 | 0.1161 |
Brugia malayi | follicle stimulating hormone receptor | 0.0021 | 0.1049 | 0.1049 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Entamoeba histolytica | cytidine deaminase, putative | 0.0118 | 1 | 0.5 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Brugia malayi | hypothetical protein | 0.0021 | 0.1049 | 0.1049 |
Onchocerca volvulus | Ribonuclease H1 homolog | 0.0022 | 0.1161 | 0.0125 |
Brugia malayi | Unidentified vitellogenin-linked transcript protein 6, putative | 0.0021 | 0.1049 | 0.1049 |
Mycobacterium leprae | PROBABLE CYTIDINE DEAMINASE CDD (CYTIDINE AMINOHYDROLASE) (CYTIDINE NUCLEOSIDE DEAMINASE) | 0.0118 | 1 | 0.5 |
Brugia malayi | sulfakinin receptor protein | 0.0021 | 0.1049 | 0.1049 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Brugia malayi | hypothetical protein | 0.0021 | 0.1049 | 0.1049 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Echinococcus multilocularis | cytidine deaminase | 0.0118 | 1 | 1 |
Trypanosoma brucei | unspecified product | 0.0024 | 0.133 | 0.133 |
Trypanosoma brucei | RNA helicase, putative | 0.0081 | 0.6644 | 0.6644 |
Treponema pallidum | ribonuclease H (rnhA) | 0.0022 | 0.1161 | 0.5 |
Brugia malayi | hypothetical protein | 0.0021 | 0.1049 | 0.1049 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Brugia malayi | Serotonin/octopamine receptor family protein 7 | 0.0021 | 0.1049 | 0.1049 |
Brugia malayi | gonadotropin-releasing hormone receptor 2 | 0.0021 | 0.1049 | 0.1049 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Loa Loa (eye worm) | G-protein coupled receptor | 0.0021 | 0.1049 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Brugia malayi | G-protein coupled receptor | 0.0021 | 0.1049 | 0.1049 |
Mycobacterium tuberculosis | Probable cytidine deaminase Cdd (cytidine aminohydrolase) (cytidine nucleoside deaminase) | 0.0118 | 1 | 0.5 |
Brugia malayi | G-protein coupled receptor | 0.0021 | 0.1049 | 0.1049 |
Leishmania major | cytidine deaminase-like protein | 0.0118 | 1 | 1 |
Trypanosoma brucei | ribonuclease H1 | 0.0022 | 0.1161 | 0.1161 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Brugia malayi | GnHR receptor homolog | 0.0021 | 0.1049 | 0.1049 |
Trypanosoma brucei | hypothetical protein, conserved | 0.0024 | 0.133 | 0.133 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Brugia malayi | Dopamine receptor protein 1 | 0.0021 | 0.1049 | 0.1049 |
Loa Loa (eye worm) | unidentified vitellogenin-linked transcript protein 6 | 0.0021 | 0.1049 | 1 |
Brugia malayi | hypothetical protein | 0.0021 | 0.1049 | 0.1049 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Brugia malayi | hypothetical protein | 0.0021 | 0.1049 | 0.1049 |
Echinococcus granulosus | ribonuclease H1 | 0.0022 | 0.1161 | 0.0125 |
Loa Loa (eye worm) | G-protein coupled receptor | 0.0021 | 0.1049 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Brugia malayi | putative neuropeptide receptor | 0.0021 | 0.1049 | 0.1049 |
Brugia malayi | G protein-coupled receptor | 0.0021 | 0.1049 | 0.1049 |
Brugia malayi | Dopamine receptor protein 1, putative (partial) | 0.0021 | 0.1049 | 0.1049 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.1049 | 1 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
EC50 (functional) | = 0.991 | Cytotoxicity against Homo sapiens (human) MCF7 cells | ChEMBL. | No reference |
IC50 (functional) | = -4.48 | Antiproliferative activity evaluated against MCF-7 cell line | ChEMBL. | 14741278 |
Log IC50 (functional) | = 4.48 | Antiproliferative activity evaluated against MCF-7 cell line | ChEMBL. | 14741278 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.