Species | Target name | Source | Bibliographic reference |
---|---|---|---|
Homo sapiens | amine oxidase, copper containing 2 (retina-specific) | Starlite/ChEMBL | References |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
I50 (binding) | = 10 uM | Effect on plasma amine oxidase (0.1 uM) after 30 min of incubation at pH 7.2 | ChEMBL. | 3127589 |
I50 (binding) | = 10 uM | Effect on plasma amine oxidase (0.1 uM) after 60 min of incubation at pH 7.2 | ChEMBL. | 3127589 |
I50 (binding) | = 50 uM | Effect on plasma amine oxidase (0.1 uM) after 15 min of incubation at pH 7.2 | ChEMBL. | 3127589 |
I50 (binding) | = 100 uM | Effect on plasma amine oxidase (0.1 uM) after 0 min of incubation at pH 7.2 | ChEMBL. | 3127589 |
I50 (binding) | = 100 uM | Effect on placental diamine oxidase (0.1 uM) after 0 min of incubation at pH 7.2 | ChEMBL. | 3127589 |
I50 (binding) | = 100 uM | Effect on placental diamine oxidase (0.1 uM) after 30 min of incubation at pH 7.2 | ChEMBL. | 3127589 |
IC50 (binding) | = 10 uM | Effect on plasma amine oxidase (0.1 uM) after 30 min of incubation at pH 7.2 | ChEMBL. | 3127589 |
IC50 (binding) | = 10 uM | Effect on plasma amine oxidase (0.1 uM) after 60 min of incubation at pH 7.2 | ChEMBL. | 3127589 |
IC50 (binding) | = 50 uM | Effect on plasma amine oxidase (0.1 uM) after 15 min of incubation at pH 7.2 | ChEMBL. | 3127589 |
IC50 (binding) | = 100 uM | Effect on plasma amine oxidase (0.1 uM) after 0 min of incubation at pH 7.2 | ChEMBL. | 3127589 |
Inhibition (functional) | = 0 % | Brain mitochondrial activity measured at 0 min of incubation at 100 microM concentration | ChEMBL. | 3127589 |
Inhibition (functional) | = 0 % | Brain mitochondrial activity measured at 0 min of incubation at 10 microM concentration | ChEMBL. | 3127589 |
Inhibition (functional) | = 0 % | Brain mitochondrial activity measured at 0 min of incubation at 1 microM concentration | ChEMBL. | 3127589 |
Inhibition (functional) | = 0 % | Brain mitochondrial activity measured at 120 min of incubation at 1 microM concentration | ChEMBL. | 3127589 |
Inhibition (binding) | = 0 % | Monoamine oxidase activity measured at 0 min of incubation at 100 microM concentration | ChEMBL. | 3127589 |
Inhibition (binding) | = 0 % | Monoamine oxidase activity measured at 0 min of incubation at 10 microM concentration. | ChEMBL. | 3127589 |
Inhibition (binding) | = 0 % | Monoamine oxidase activity measured at 120 min of incubation at 10 microM concentration | ChEMBL. | 3127589 |
Inhibition (binding) | = 0 % | Monoamine oxidase activity measured at 0 min of incubation at 1 microM concentration | ChEMBL. | 3127589 |
Inhibition (binding) | = 0 % | Monoamine oxidase activity measured at 120 min of incubation at 1 microM concentration | ChEMBL. | 3127589 |
Inhibition (binding) | = 0 % | Monoamine oxidase activity measured at 0 min of incubation at 100 microM concentration | ChEMBL. | 3127589 |
Inhibition (binding) | = 0 % | Monoamine oxidase activity measured at 0 min of incubation at 10 microM concentration. | ChEMBL. | 3127589 |
Inhibition (binding) | = 0 % | Monoamine oxidase activity measured at 120 min of incubation at 10 microM concentration | ChEMBL. | 3127589 |
Inhibition (binding) | = 0 % | Monoamine oxidase activity measured at 0 min of incubation at 1 microM concentration | ChEMBL. | 3127589 |
Inhibition (binding) | = 0 % | Monoamine oxidase activity measured at 120 min of incubation at 1 microM concentration | ChEMBL. | 3127589 |
Inhibition (binding) | = 2 % | Monoamine oxidase activity measured at 120 min of incubation at 100 microM concentration. | ChEMBL. | 3127589 |
Inhibition (binding) | = 2 % | Monoamine oxidase activity measured at 120 min of incubation at 100 microM concentration. | ChEMBL. | 3127589 |
Inhibition (functional) | = 5 % | Brain mitochondrial activity measured at 120 min of incubation at 10 microM concentration | ChEMBL. | 3127589 |
Inhibition (functional) | = 8 % | Brain mitochondrial activity measured at 120 min of incubation at 100 microM concentration | ChEMBL. | 3127589 |
Ki (binding) | = 85 uM | Ki value measured for the inhibition of copper dependent amine oxidase in bovine plasma | ChEMBL. | 3127589 |
Ki (binding) | = 110 uM | Ki value measured for the inhibition of human placenta diamine oxidase | ChEMBL. | 3127589 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.