Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0039 | 0.4166 | 0.6498 |
Schistosoma mansoni | ataxia telangiectasia mutated (atm)-related | 0.0052 | 0.6411 | 0.6187 |
Entamoeba histolytica | phosphatidylinositol3-kinaseTor2, putative | 0.0052 | 0.6411 | 0.5 |
Trypanosoma brucei | target of rapamycin kinase 3, putative | 0.0042 | 0.4626 | 0.6934 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0042 | 0.4618 | 0.7204 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0018 | 0.0587 | 0.0916 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0031 | 0.2885 | 0.4499 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0028 | 0.238 | 0.3713 |
Trypanosoma cruzi | target of rapamycin kinase 3 | 0.0042 | 0.4626 | 0.6934 |
Trypanosoma cruzi | Phosphatidylinositol 3-kinase tor2 | 0.0052 | 0.6411 | 1 |
Schistosoma mansoni | tar DNA-binding protein | 0.0074 | 1 | 1 |
Trypanosoma brucei | FAT domain/Rapamycin binding domain/Phosphatidylinositol 3- and 4-kinase, putative | 0.0022 | 0.1288 | 0.1204 |
Schistosoma mansoni | tar DNA-binding protein | 0.0074 | 1 | 1 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0028 | 0.2373 | 0.3702 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0018 | 0.0587 | 0.0916 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0028 | 0.238 | 0.3713 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0031 | 0.2885 | 0.4499 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0052 | 0.6411 | 1 |
Echinococcus granulosus | FKBP12 rapamycin complex associated protein | 0.0052 | 0.6411 | 0.6187 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0042 | 0.4618 | 0.7204 |
Trypanosoma brucei | phosphatidylinositol 4-kinase, putative | 0.0052 | 0.6411 | 1 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0028 | 0.2373 | 0.3702 |
Echinococcus multilocularis | FKBP12 rapamycin complex associated protein | 0.0052 | 0.6411 | 0.6187 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0028 | 0.238 | 0.3713 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0052 | 0.6411 | 1 |
Echinococcus granulosus | tar DNA binding protein | 0.0074 | 1 | 1 |
Toxoplasma gondii | target of rapamycin (TOR), putative | 0.0039 | 0.4166 | 0.5 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0031 | 0.2833 | 0.4418 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0018 | 0.0587 | 0.0916 |
Trypanosoma brucei | Phosphatidylinositol 3-kinase tor1 | 0.0052 | 0.6411 | 1 |
Schistosoma mansoni | tar DNA-binding protein | 0.0074 | 1 | 1 |
Leishmania major | target of rapamycin (TOR) kinase 2, putative | 0.0052 | 0.6411 | 1 |
Echinococcus multilocularis | tar DNA binding protein | 0.0074 | 1 | 1 |
Loa Loa (eye worm) | phosphatidylinositol 3 | 0.0052 | 0.6411 | 0.6187 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0039 | 0.4166 | 0.6498 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0035 | 0.3527 | 0.5501 |
Entamoeba histolytica | FKBP-rapamycin associated protein (FRAP), putative | 0.0052 | 0.6411 | 0.5 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0031 | 0.2885 | 0.4499 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0039 | 0.4166 | 0.6498 |
Brugia malayi | RNA recognition motif domain containing protein | 0.0074 | 1 | 1 |
Brugia malayi | Phosphatidylinositol 3- and 4-kinase family protein | 0.0052 | 0.6411 | 0.6187 |
Brugia malayi | TAR-binding protein | 0.0074 | 1 | 1 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0039 | 0.4166 | 0.6498 |
Trypanosoma brucei | phosphatidylinositol 3-kinase tor, putative | 0.0025 | 0.1793 | 0.207 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0018 | 0.0587 | 0.0916 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0018 | 0.0587 | 0.0916 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0045 | 0.513 | 0.8002 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0028 | 0.238 | 0.3713 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0042 | 0.4618 | 0.7204 |
Loa Loa (eye worm) | RNA recognition domain-containing protein domain-containing protein | 0.0074 | 1 | 1 |
Giardia lamblia | GTOR | 0.0052 | 0.6411 | 0.5 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0034 | 0.3337 | 0.5205 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0031 | 0.2833 | 0.4418 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0039 | 0.4166 | 0.6498 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0052 | 0.6411 | 1 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0042 | 0.4618 | 0.7204 |
Loa Loa (eye worm) | RNA binding protein | 0.0074 | 1 | 1 |
Trypanosoma cruzi | Phosphatidylinositol 3-kinase tor1 | 0.0052 | 0.6411 | 1 |
Schistosoma mansoni | tar DNA-binding protein | 0.0074 | 1 | 1 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0028 | 0.2373 | 0.3702 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0039 | 0.4166 | 0.6498 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0042 | 0.4618 | 0.7204 |
Leishmania major | target of rapamycin (TOR) kinase 1, putative | 0.0052 | 0.6411 | 1 |
Schistosoma mansoni | tar DNA-binding protein | 0.0074 | 1 | 1 |
Loa Loa (eye worm) | TAR-binding protein | 0.0074 | 1 | 1 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0039 | 0.4166 | 0.6498 |
Leishmania major | target of rapamycin kinase (TOR) kinase 3 | 0.0042 | 0.4626 | 0.6934 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
Clearance (functional) | = 0 % | Mouse oral clearance was measured against H. nana. | ChEMBL. | 7120286 |
Clearance (functional) | = 5 % | Mouse oral clearance was measured against N. dubius | ChEMBL. | 7120286 |
Reduction (functional) | = 40 % | Percent reduction in nematode fecal egg count was measured in sheep following 50 mg/kg p.o. | ChEMBL. | 7120286 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.