Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Schistosoma mansoni | potassium channel beta | 0.005 | 0.2563 | 0.2409 |
Onchocerca volvulus | 0.005 | 0.2563 | 0.2409 | |
Toxoplasma gondii | aldo-keto reductase | 0.005 | 0.2563 | 0.2409 |
Echinococcus multilocularis | aldehyde reductase | 0.0124 | 0.6968 | 0.6968 |
Plasmodium vivax | oxidoreductase, aldo/keto reductase domain containing protein | 0.005 | 0.2563 | 1 |
Echinococcus granulosus | ATP binding cassette subfamily B MDR:TAP | 0.0011 | 0.0203 | 0.0203 |
Trichomonas vaginalis | lipid A export ATP-binding/permease protein msba, putative | 0.0011 | 0.0203 | 0.0203 |
Trichomonas vaginalis | aldo-keto reductase, putative | 0.005 | 0.2563 | 0.2563 |
Echinococcus multilocularis | multidrug resistance protein 1 | 0.0011 | 0.0203 | 0.0203 |
Trichomonas vaginalis | ABC transporter, putative | 0.0011 | 0.0203 | 0.0203 |
Brugia malayi | glutamate-cysteine ligase modifier subunit | 0.005 | 0.2563 | 0.2409 |
Loa Loa (eye worm) | hypothetical protein | 0.0011 | 0.0203 | 0.0007 |
Echinococcus multilocularis | ATP binding cassette subfamily B (MDR:TAP) | 0.0011 | 0.0203 | 0.0203 |
Trichomonas vaginalis | lipid A export ATP-binding/permease protein msba, putative | 0.0011 | 0.0203 | 0.0203 |
Toxoplasma gondii | oxidoreductase, aldo/keto reductase family protein | 0.005 | 0.2563 | 0.2409 |
Echinococcus granulosus | multidrug resistance protein 1 | 0.0011 | 0.0203 | 0.0203 |
Brugia malayi | NADH-dependent xylose reductase | 0.005 | 0.2563 | 0.2409 |
Trichomonas vaginalis | ATP-binding cassette transporter, putative | 0.0011 | 0.0203 | 0.0203 |
Plasmodium falciparum | aldo-keto reductase, putative | 0.005 | 0.2563 | 1 |
Trichomonas vaginalis | lipid A export ATP-binding/permease protein msba, putative | 0.0011 | 0.0203 | 0.0203 |
Trichomonas vaginalis | ABC transporter, putative | 0.0011 | 0.0203 | 0.0203 |
Trichomonas vaginalis | ABC transporter, putative | 0.0011 | 0.0203 | 0.0203 |
Echinococcus multilocularis | ATP binding cassette subfamily B (MDR:TAP) | 0.0011 | 0.0203 | 0.0203 |
Trichomonas vaginalis | aldo-keto reductase, putative | 0.005 | 0.2563 | 0.2563 |
Echinococcus granulosus | ATP binding cassette subfamily B MDR:TAP | 0.0011 | 0.0203 | 0.0203 |
Mycobacterium tuberculosis | Conserved protein | 0.005 | 0.2563 | 0.2409 |
Entamoeba histolytica | alcohol dehydrogenase, putative | 0.005 | 0.2563 | 0.2409 |
Trichomonas vaginalis | lipid A export ATP-binding/permease protein msba, putative | 0.0011 | 0.0203 | 0.0203 |
Echinococcus granulosus | ATP binding cassette subfamily B MDR:TAP | 0.0011 | 0.0203 | 0.0203 |
Mycobacterium leprae | Conserved hypothetical protein | 0.0124 | 0.6968 | 0.5922 |
Toxoplasma gondii | aldo/keto reductase family oxidoreductase | 0.005 | 0.2563 | 0.2409 |
Echinococcus multilocularis | multidrug resistance protein 1 | 0.0011 | 0.0203 | 0.0203 |
Trichomonas vaginalis | ABC transporter, putative | 0.0011 | 0.0203 | 0.0203 |
Trichomonas vaginalis | abcb9, putative | 0.0011 | 0.0203 | 0.0203 |
Trichomonas vaginalis | aldo-keto reductase, putative | 0.005 | 0.2563 | 0.2563 |
Trichomonas vaginalis | abcb9, putative | 0.0011 | 0.0203 | 0.0203 |
Trichomonas vaginalis | ATP-binding cassette transporter, putative | 0.0011 | 0.0203 | 0.0203 |
Trichomonas vaginalis | taga, putative | 0.0011 | 0.0203 | 0.0203 |
Echinococcus granulosus | 5'partial|ATP binding cassette sub family B | 0.0011 | 0.0196 | 0.0196 |
Trichomonas vaginalis | multidrug resistance protein 1, 2, putative | 0.0011 | 0.0203 | 0.0203 |
Trichomonas vaginalis | conserved hypothetical protein | 0.005 | 0.2563 | 0.2563 |
Chlamydia trachomatis | ABC transporter ATP binding protein/permease | 0.0011 | 0.0203 | 0.5 |
Echinococcus multilocularis | ATP binding cassette subfamily B (MDR:TAP) | 0.0011 | 0.0203 | 0.0203 |
Trichomonas vaginalis | ABC transporter, half transporter, putative | 0.0011 | 0.0203 | 0.0203 |
Trichomonas vaginalis | ATP-binding cassette transporter, putative | 0.0011 | 0.0203 | 0.0203 |
Trichomonas vaginalis | lipid A export ATP-binding/permease protein msba, putative | 0.0011 | 0.0203 | 0.0203 |
Trichomonas vaginalis | abcb9, putative | 0.0011 | 0.0203 | 0.0203 |
Trichomonas vaginalis | lipid A export ATP-binding/permease protein msba, putative | 0.0011 | 0.0203 | 0.0203 |
Echinococcus granulosus | aldehyde reductase | 0.0124 | 0.6968 | 0.6968 |
Trichomonas vaginalis | alcohol dehydrogenase, putative | 0.005 | 0.2563 | 0.2563 |
Loa Loa (eye worm) | multidrug resistance protein 3 | 0.0011 | 0.0203 | 0.0007 |
Trichomonas vaginalis | multidrug resistance protein 1, 2, putative | 0.0011 | 0.0203 | 0.0203 |
Trichomonas vaginalis | multidrug resistance protein 1, 2, putative | 0.0011 | 0.0203 | 0.0203 |
Echinococcus granulosus | multidrug resistance protein 1 | 0.0011 | 0.0203 | 0.0203 |
Echinococcus multilocularis | ATP binding cassette sub family B | 0.0011 | 0.0196 | 0.0196 |
Echinococcus granulosus | voltage gated potassium channel subunit | 0.005 | 0.2563 | 0.2563 |
Trichomonas vaginalis | multidrug resistance protein 1, 2, putative | 0.0011 | 0.0203 | 0.0203 |
Echinococcus multilocularis | ATP binding cassette subfamily B (MDR:TAP) | 0.0011 | 0.0203 | 0.0203 |
Plasmodium vivax | aldehyde reductase, putative | 0.005 | 0.2563 | 1 |
Trichomonas vaginalis | ATP-binding cassette transporter, putative | 0.0011 | 0.0203 | 0.0203 |
Loa Loa (eye worm) | ATP-binding cassette sub-family B member 2 | 0.0011 | 0.0203 | 0.0007 |
Trichomonas vaginalis | multidrug resistance protein 1, 2, putative | 0.0011 | 0.0203 | 0.0203 |
Plasmodium falciparum | aldehyde reductase, putative | 0.005 | 0.2563 | 1 |
Trichomonas vaginalis | multidrug resistance protein 1, 2, putative | 0.0011 | 0.0203 | 0.0203 |
Loa Loa (eye worm) | glutamate-cysteine ligase modifier subunit | 0.005 | 0.2563 | 0.2415 |
Loa Loa (eye worm) | hypothetical protein | 0.0011 | 0.0203 | 0.0007 |
Trichomonas vaginalis | ABC transporter, half transporter, putative | 0.0011 | 0.0203 | 0.0203 |
Leishmania major | aldo/keto reductase, putative,aldo/keto reductase family-like protein | 0.005 | 0.2563 | 0.2409 |
Echinococcus multilocularis | voltage gated potassium channel subunit | 0.005 | 0.2563 | 0.2563 |
Echinococcus granulosus | ATP binding cassette subfamily B MDR:TAP | 0.0011 | 0.0203 | 0.0203 |
Trichomonas vaginalis | lipid A export ATP-binding/permease protein msba, putative | 0.0011 | 0.0203 | 0.0203 |
Echinococcus granulosus | multidrug resistance protein 1 | 0.0011 | 0.0203 | 0.0203 |
Echinococcus multilocularis | ATP binding cassette subfamily B (MDR:TAP) | 0.0011 | 0.0203 | 0.0203 |
Trichomonas vaginalis | multidrug resistance protein 1, 2, putative | 0.0011 | 0.0203 | 0.0203 |
Entamoeba histolytica | alcohol dehydrogenase, putative | 0.005 | 0.2563 | 0.2409 |
Echinococcus granulosus | aldo keto reductase family 1, member B4 | 0.005 | 0.2563 | 0.2563 |
Trichomonas vaginalis | lipid A export ATP-binding/permease protein msba, putative | 0.0011 | 0.0203 | 0.0203 |
Trichomonas vaginalis | ATP-binding cassette transporter, putative | 0.0011 | 0.0203 | 0.0203 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
IC50 (functional) | > 50 uM | Cytotoxicity against mouse B16 cells assessed as reduction in cell viability after 48 hrs by MTT assay | ChEMBL. | 21112130 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.