Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Schistosoma mansoni | L-lactate dehydrogenase | 0.0592 | 0.5723 | 0.5723 |
Trypanosoma cruzi | glycosomal malate dehydrogenase, putative | 0.0764 | 0.7621 | 0.7271 |
Echinococcus granulosus | malate dehydrogenase | 0.0764 | 0.7621 | 0.7621 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0829 | 0.8334 | 1 |
Plasmodium vivax | malate dehydrogenase, putative | 0.098 | 1 | 1 |
Echinococcus granulosus | cytosolic malate dehydrogenase | 0.0829 | 0.8334 | 0.8334 |
Loa Loa (eye worm) | malate dehydrogenase | 0.0829 | 0.8334 | 0.8334 |
Trypanosoma cruzi | cytosolic malate dehydrogenase, putative | 0.0829 | 0.8334 | 1 |
Wolbachia endosymbiont of Brugia malayi | malate dehydrogenase | 0.098 | 1 | 0.5 |
Schistosoma mansoni | malate dehydrogenase | 0.098 | 1 | 1 |
Giardia lamblia | Malate dehydrogenase | 0.0829 | 0.8334 | 0.5 |
Trypanosoma brucei | mitochondrial malate dehydrogenase | 0.0764 | 0.7621 | 0.7271 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0592 | 0.5723 | 0.5611 |
Trichomonas vaginalis | malate and lactate dehydrogenase, putative | 0.0829 | 0.8334 | 1 |
Echinococcus granulosus | malate dehydrogenase | 0.0764 | 0.7621 | 0.7621 |
Trichomonas vaginalis | malate and lactate dehydrogenase, putative | 0.0829 | 0.8334 | 1 |
Plasmodium falciparum | L-lactate dehydrogenase | 0.098 | 1 | 1 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0829 | 0.8334 | 1 |
Trypanosoma brucei | glycosomal malate dehydrogenase | 0.0764 | 0.7621 | 0.7271 |
Echinococcus multilocularis | lactate dehydrogenase a | 0.098 | 1 | 1 |
Trypanosoma brucei | cytosolic malate dehydrogenase | 0.0829 | 0.8334 | 1 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0829 | 0.8334 | 1 |
Brugia malayi | Malate dehydrogenase, cytoplasmic | 0.0829 | 0.8334 | 0.8334 |
Chlamydia trachomatis | malate dehydrogenase | 0.0829 | 0.8334 | 0.5 |
Trypanosoma cruzi | malate dehydrogenase, putative | 0.0764 | 0.7621 | 0.7271 |
Echinococcus multilocularis | cytosolic malate dehydrogenase | 0.0829 | 0.8334 | 0.8334 |
Mycobacterium leprae | PROBABLE MALATE DEHYDROGENASE MDH | 0.0829 | 0.8334 | 0.5 |
Echinococcus granulosus | L lactate dehydrogenase B chain | 0.098 | 1 | 1 |
Toxoplasma gondii | lactate dehydrogenase LDH2 | 0.098 | 1 | 0.5 |
Echinococcus multilocularis | cytosolic malate dehydrogenase | 0.0829 | 0.8334 | 0.8334 |
Schistosoma mansoni | malate dehydrogenase | 0.0764 | 0.7621 | 0.7621 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0829 | 0.8334 | 1 |
Entamoeba histolytica | malate dehydrogenase, putative | 0.098 | 1 | 1 |
Echinococcus granulosus | lactate dehydrogenase a | 0.098 | 1 | 1 |
Echinococcus multilocularis | malate dehydrogenase | 0.0764 | 0.7621 | 0.7621 |
Plasmodium falciparum | malate dehydrogenase | 0.098 | 1 | 1 |
Echinococcus granulosus | cytosolic malate dehydrogenase | 0.0829 | 0.8334 | 0.8334 |
Schistosoma mansoni | malate dehydrogenase | 0.0829 | 0.8334 | 0.8334 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0525 | 0.4996 | 0.4389 |
Schistosoma mansoni | malate dehydrogenase | 0.0829 | 0.8334 | 0.8334 |
Toxoplasma gondii | malate dehydrogenase MDH | 0.098 | 1 | 0.5 |
Leishmania major | glycosomal malate dehydrogenase | 0.0764 | 0.7621 | 0.4439 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0829 | 0.8334 | 1 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0829 | 0.8334 | 1 |
Schistosoma mansoni | L-lactate dehydrogenase | 0.098 | 1 | 1 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0829 | 0.8334 | 1 |
Echinococcus granulosus | L lactate dehydrogenase | 0.0389 | 0.3491 | 0.3491 |
Plasmodium vivax | lactate dehydrogenase | 0.098 | 1 | 1 |
Echinococcus multilocularis | lactate dehydrogenase a | 0.098 | 1 | 1 |
Leishmania major | malate dehydrogenase | 0.0764 | 0.7621 | 0.4439 |
Trypanosoma cruzi | mitochondrial malate dehydrogenase, putative | 0.0764 | 0.7621 | 0.7271 |
Echinococcus multilocularis | malate dehydrogenase | 0.0764 | 0.7621 | 0.7621 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0829 | 0.8334 | 1 |
Echinococcus multilocularis | L lactate dehydrogenase B chain | 0.098 | 1 | 1 |
Echinococcus granulosus | lactate dehydrogenase protein | 0.098 | 1 | 1 |
Echinococcus multilocularis | L lactate dehydrogenase | 0.0389 | 0.3491 | 0.3491 |
Trypanosoma cruzi | glycosomal malate dehydrogenase, putative | 0.0764 | 0.7621 | 0.7271 |
Brugia malayi | Probable malate dehydrogenase, mitochondrial precursor | 0.0764 | 0.7621 | 0.7621 |
Trichomonas vaginalis | malate and lactate dehydrogenase, putative | 0.0829 | 0.8334 | 1 |
Echinococcus multilocularis | lactate dehydrogenase a | 0.098 | 1 | 1 |
Echinococcus multilocularis | lactate dehydrogenase protein | 0.098 | 1 | 1 |
Echinococcus granulosus | lactate dehydrogenase a | 0.098 | 1 | 1 |
Loa Loa (eye worm) | malate dehydrogenase | 0.0764 | 0.7621 | 0.7621 |
Leishmania major | mitochondrial malate dehydrogenase | 0.0764 | 0.7621 | 0.4439 |
Leishmania major | cytosolic malate dehydrogenase | 0.0829 | 0.8334 | 0.6105 |
Trypanosoma cruzi | cytosolic malate dehydrogenase, putative | 0.0829 | 0.8334 | 1 |
Trichomonas vaginalis | malate and lactate dehydrogenase, putative | 0.0829 | 0.8334 | 1 |
Mycobacterium tuberculosis | Probable malate dehydrogenase Mdh | 0.0829 | 0.8334 | 0.5 |
Mycobacterium ulcerans | malate dehydrogenase | 0.0829 | 0.8334 | 0.5 |
Loa Loa (eye worm) | hypothetical protein | 0.098 | 1 | 1 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0829 | 0.8334 | 1 |
Toxoplasma gondii | lactate dehydrogenase LDH1 | 0.098 | 1 | 0.5 |
Leishmania major | malate dehydrogenase, putative | 0.098 | 1 | 1 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0829 | 0.8334 | 1 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0829 | 0.8334 | 1 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
Decrease (functional) | = -0.2 % | The hypoglycemic activity in diabetic KK mice,activity expressed as % decrease in blood glucose (21h) | ChEMBL. | 10956213 |
Decrease (functional) | = 14.6 % | The hypoglycemic activity in diabetic KK mice,activity expressed as % decrease in blood glucose (18 h) | ChEMBL. | 10956213 |
EC (functional) | = 0.075 uM | Stimulation of adipogenesis in 3T3-L1 cells is expressed as concentration equivalent to the [ 1-14C] uptake counts after treatment with 0.2 ug/mL troglitazone | ChEMBL. | 10956213 |
EC (functional) | = 0.075 uM | Stimulation of adipogenesis in 3T3-L1 cells is expressed as concentration equivalent to the [ 1-14C] uptake counts after treatment with 0.2 ug/mL troglitazone | ChEMBL. | 10956213 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.