Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Loa Loa (eye worm) | tubulin beta-2A chain | 0.0142 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0142 | 0.5 | 0.5 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0142 | 0.5 | 0.5 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0142 | 0.5 | 0.5 |
Echinococcus multilocularis | tubulin subunit beta | 0.0142 | 0.5 | 0.5 |
Loa Loa (eye worm) | tubulin beta-4 chain | 0.0142 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0142 | 0.5 | 0.5 |
Schistosoma mansoni | tubulin subunit beta | 0.0142 | 0.5 | 0.5 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0142 | 0.5 | 0.5 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0142 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0142 | 0.5 | 0.5 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0142 | 0.5 | 0.5 |
Echinococcus granulosus | tubulin beta 4A class IVa | 0.0142 | 0.5 | 0.5 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0142 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0142 | 0.5 | 0.5 |
Trypanosoma brucei | beta tubulin | 0.0142 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0142 | 0.5 | 0.5 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0142 | 0.5 | 0.5 |
Entamoeba histolytica | tubulin family protein | 0.0142 | 0.5 | 0.5 |
Schistosoma mansoni | tubulin subunit beta | 0.0142 | 0.5 | 0.5 |
Loa Loa (eye worm) | tubulin beta-1 chain | 0.0142 | 0.5 | 0.5 |
Loa Loa (eye worm) | beta-tubulin | 0.0142 | 0.5 | 0.5 |
Toxoplasma gondii | beta tubulin | 0.0142 | 0.5 | 0.5 |
Brugia malayi | beta-tubulin, identical | 0.0142 | 0.5 | 0.5 |
Schistosoma mansoni | tubulin subunit beta | 0.0142 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0142 | 0.5 | 0.5 |
Giardia lamblia | Beta tubulin | 0.0142 | 0.5 | 0.5 |
Echinococcus multilocularis | beta tubulin | 0.0142 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0142 | 0.5 | 0.5 |
Entamoeba histolytica | tubulin family protein | 0.0142 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0142 | 0.5 | 0.5 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0142 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0142 | 0.5 | 0.5 |
Plasmodium falciparum | tubulin beta chain | 0.0142 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0142 | 0.5 | 0.5 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0142 | 0.5 | 0.5 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0142 | 0.5 | 0.5 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0142 | 0.5 | 0.5 |
Trichomonas vaginalis | tubulin, putative | 0.0142 | 0.5 | 0.5 |
Echinococcus multilocularis | beta tubulin | 0.0142 | 0.5 | 0.5 |
Plasmodium vivax | tubulin beta chain, putative | 0.0142 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0142 | 0.5 | 0.5 |
Trypanosoma cruzi | beta tubulin, putative | 0.0142 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0142 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0142 | 0.5 | 0.5 |
Giardia lamblia | Beta tubulin | 0.0142 | 0.5 | 0.5 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0142 | 0.5 | 0.5 |
Schistosoma mansoni | tubulin subunit beta | 0.0142 | 0.5 | 0.5 |
Echinococcus multilocularis | tubulin, beta 4A class IVa | 0.0142 | 0.5 | 0.5 |
Schistosoma mansoni | tubulin subunit beta | 0.0142 | 0.5 | 0.5 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0142 | 0.5 | 0.5 |
Loa Loa (eye worm) | BEN-1 protein | 0.0142 | 0.5 | 0.5 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0142 | 0.5 | 0.5 |
Echinococcus granulosus | tubulin beta 1 chain | 0.0142 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0142 | 0.5 | 0.5 |
Trypanosoma brucei | beta tubulin | 0.0142 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0142 | 0.5 | 0.5 |
Toxoplasma gondii | beta-1 tubulin, putative | 0.0142 | 0.5 | 0.5 |
Trypanosoma brucei | beta tubulin | 0.0142 | 0.5 | 0.5 |
Giardia lamblia | Beta tubulin | 0.0142 | 0.5 | 0.5 |
Schistosoma mansoni | tubulin subunit beta | 0.0142 | 0.5 | 0.5 |
Echinococcus multilocularis | tubulin beta 1 chain | 0.0142 | 0.5 | 0.5 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0142 | 0.5 | 0.5 |
Echinococcus granulosus | beta tubulin | 0.0142 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0142 | 0.5 | 0.5 |
Trypanosoma brucei | beta tubulin | 0.0142 | 0.5 | 0.5 |
Toxoplasma gondii | beta-tubulin, putative | 0.0142 | 0.5 | 0.5 |
Echinococcus granulosus | tubulin subunit beta | 0.0142 | 0.5 | 0.5 |
Loa Loa (eye worm) | tubulin beta chain | 0.0142 | 0.5 | 0.5 |
Echinococcus granulosus | beta tubulin | 0.0142 | 0.5 | 0.5 |
Loa Loa (eye worm) | BEN-1 protein | 0.0142 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0142 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0142 | 0.5 | 0.5 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
Activity (binding) | = 82 % | Inactivation of tyrosinase (unknown origin) assessed as decay half-life using 4-methylcatechol substrate at 850 uM equimolar concentrations resorcinol by spectrophotometry | ChEMBL. | 23352755 |
Activity (binding) | = 97 % | Inactivation of tyrosinase (unknown origin) assessed as initial rate of oxygen utilization using 4-methylcatechol substrate at 850 uM equimolar concentrations resorcinol by spectrophotometry | ChEMBL. | 23352755 |
Activity (binding) | = 103 % | Inactivation of tyrosinase (unknown origin) assessed as initial rate of oxygen utilization at absorbance 400 nm using 4-methylcatechol substrate at 850 uM equimolar concentrations resorcinol by spectrophotometry | ChEMBL. | 23352755 |
Activity (binding) | = 117 % | Inactivation of tyrosinase (unknown origin) assessed as total oxygen uptake using 4-methylcatechol substrate at 850 uM equimolar concentrations resorcinol by spectrophotometry | ChEMBL. | 23352755 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.