Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Echinococcus granulosus | tubulin beta 4A class IVa | 0.0028 | 0.018 | 1 |
Giardia lamblia | Beta tubulin | 0.0028 | 0.018 | 0.5 |
Leishmania major | beta tubulin | 0.0028 | 0.018 | 0.5 |
Loa Loa (eye worm) | beta-tubulin | 0.0028 | 0.018 | 0.2399 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0028 | 0.018 | 1 |
Leishmania major | beta tubulin | 0.0028 | 0.018 | 0.5 |
Leishmania major | beta tubulin | 0.0028 | 0.018 | 0.5 |
Trypanosoma brucei | beta tubulin | 0.0028 | 0.018 | 0.5 |
Entamoeba histolytica | tubulin family protein | 0.0028 | 0.018 | 0.5 |
Echinococcus multilocularis | tubulin, beta 4A class IVa | 0.0028 | 0.018 | 1 |
Trypanosoma brucei | beta tubulin | 0.0028 | 0.018 | 0.5 |
Schistosoma mansoni | o-methyltransferase | 0.006 | 0.0749 | 1 |
Schistosoma mansoni | o-methyltransferase | 0.006 | 0.0749 | 1 |
Toxoplasma gondii | beta-tubulin, putative | 0.0028 | 0.018 | 0.5 |
Trypanosoma cruzi | beta tubulin, putative | 0.0028 | 0.018 | 0.5 |
Toxoplasma gondii | beta tubulin | 0.0028 | 0.018 | 0.5 |
Entamoeba histolytica | tubulin family protein | 0.0028 | 0.018 | 0.5 |
Leishmania major | beta tubulin | 0.0028 | 0.018 | 0.5 |
Brugia malayi | O-methyltransferase | 0.006 | 0.0749 | 1 |
Echinococcus granulosus | tubulin subunit beta | 0.0028 | 0.018 | 1 |
Onchocerca volvulus | 0.006 | 0.0749 | 0.5 | |
Leishmania major | beta tubulin | 0.0028 | 0.018 | 0.5 |
Schistosoma mansoni | tubulin subunit beta | 0.0028 | 0.018 | 0.2399 |
Loa Loa (eye worm) | tubulin beta chain | 0.0028 | 0.018 | 0.2399 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0028 | 0.018 | 1 |
Leishmania major | beta tubulin | 0.0028 | 0.018 | 0.5 |
Leishmania major | beta tubulin | 0.0028 | 0.018 | 0.5 |
Leishmania major | beta tubulin | 0.0028 | 0.018 | 0.5 |
Brugia malayi | Calcitonin receptor-like protein seb-1 | 0.0057 | 0.0697 | 0.9313 |
Echinococcus multilocularis | beta tubulin | 0.0028 | 0.018 | 1 |
Brugia malayi | O-methyltransferase family protein | 0.006 | 0.0749 | 1 |
Giardia lamblia | Beta tubulin | 0.0028 | 0.018 | 0.5 |
Trypanosoma brucei | beta tubulin | 0.0028 | 0.018 | 0.5 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0028 | 0.018 | 1 |
Mycobacterium tuberculosis | Probable catechol-O-methyltransferase | 0.0518 | 0.8929 | 1 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0028 | 0.018 | 0.5 |
Leishmania major | beta tubulin | 0.0028 | 0.018 | 0.5 |
Brugia malayi | latrophilin 2 splice variant baaae | 0.0039 | 0.0375 | 0.5002 |
Loa Loa (eye worm) | hypothetical protein | 0.0039 | 0.0375 | 0.5002 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0028 | 0.018 | 0.5 |
Loa Loa (eye worm) | tubulin beta-2A chain | 0.0028 | 0.018 | 0.2399 |
Schistosoma mansoni | tubulin subunit beta | 0.0028 | 0.018 | 0.2399 |
Leishmania major | beta tubulin | 0.0028 | 0.018 | 0.5 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0028 | 0.018 | 0.5 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0028 | 0.018 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0028 | 0.018 | 0.5 |
Loa Loa (eye worm) | tubulin beta-1 chain | 0.0028 | 0.018 | 0.2399 |
Schistosoma mansoni | hypothetical protein | 0.0039 | 0.0375 | 0.5002 |
Brugia malayi | Tubulin beta-1 chain | 0.0028 | 0.018 | 0.2399 |
Leishmania major | beta tubulin | 0.0028 | 0.018 | 0.5 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0028 | 0.018 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0028 | 0.018 | 0.2399 |
Trichomonas vaginalis | tubulin, putative | 0.0028 | 0.018 | 0.5 |
Schistosoma mansoni | o-methyltransferase | 0.006 | 0.0749 | 1 |
Toxoplasma gondii | beta-1 tubulin, putative | 0.0028 | 0.018 | 0.5 |
Schistosoma mansoni | tubulin subunit beta | 0.0028 | 0.018 | 0.2399 |
Brugia malayi | Corticotropin releasing factor receptor 2 precursor, putative | 0.0057 | 0.0697 | 0.9313 |
Onchocerca volvulus | 0.006 | 0.0749 | 0.5 | |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0028 | 0.018 | 0.5 |
Loa Loa (eye worm) | hypothetical protein | 0.0057 | 0.0697 | 0.9313 |
Loa Loa (eye worm) | BEN-1 protein | 0.0028 | 0.018 | 0.2399 |
Echinococcus multilocularis | beta tubulin | 0.0028 | 0.018 | 1 |
Plasmodium vivax | tubulin beta chain, putative | 0.0028 | 0.018 | 0.5 |
Echinococcus granulosus | beta tubulin | 0.0028 | 0.018 | 1 |
Echinococcus multilocularis | tubulin subunit beta | 0.0028 | 0.018 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0028 | 0.018 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0028 | 0.018 | 1 |
Leishmania major | beta tubulin | 0.0028 | 0.018 | 0.5 |
Loa Loa (eye worm) | O-methyltransferase | 0.006 | 0.0749 | 1 |
Leishmania major | beta tubulin | 0.0028 | 0.018 | 0.5 |
Wolbachia endosymbiont of Brugia malayi | O-methyltransferase | 0.006 | 0.0749 | 0.5 |
Echinococcus granulosus | tubulin beta 1 chain | 0.0028 | 0.018 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.006 | 0.0749 | 1 |
Leishmania major | beta tubulin | 0.0028 | 0.018 | 0.5 |
Mycobacterium leprae | PROBABLE METHYLTRANSFERASE | 0.006 | 0.0749 | 0.5 |
Schistosoma mansoni | o-methyltransferase | 0.006 | 0.0749 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0028 | 0.018 | 1 |
Loa Loa (eye worm) | tubulin beta-4 chain | 0.0028 | 0.018 | 0.2399 |
Loa Loa (eye worm) | pigment dispersing factor receptor c | 0.0057 | 0.0697 | 0.9313 |
Schistosoma mansoni | tubulin subunit beta | 0.0028 | 0.018 | 0.2399 |
Brugia malayi | O-methyltransferase family protein | 0.006 | 0.0749 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0028 | 0.018 | 1 |
Leishmania major | beta tubulin | 0.0028 | 0.018 | 0.5 |
Brugia malayi | beta-tubulin, identical | 0.0028 | 0.018 | 0.2399 |
Leishmania major | beta tubulin | 0.0028 | 0.018 | 0.5 |
Echinococcus granulosus | beta tubulin | 0.0028 | 0.018 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0028 | 0.018 | 0.2399 |
Echinococcus multilocularis | tubulin beta 1 chain | 0.0028 | 0.018 | 1 |
Trypanosoma brucei | beta tubulin | 0.0028 | 0.018 | 0.5 |
Leishmania major | beta tubulin | 0.0028 | 0.018 | 0.5 |
Leishmania major | beta tubulin | 0.0028 | 0.018 | 0.5 |
Loa Loa (eye worm) | BEN-1 protein | 0.0028 | 0.018 | 0.2399 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0028 | 0.018 | 1 |
Plasmodium falciparum | tubulin beta chain | 0.0028 | 0.018 | 0.5 |
Giardia lamblia | Beta tubulin | 0.0028 | 0.018 | 0.5 |
Brugia malayi | O-methyltransferase family protein | 0.006 | 0.0749 | 1 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
Km (binding) | = 28 uM | Tested for inhibition of Nucleoside Triphosphate Diphosphohydrolase (NTPDase) from bovine spleen. | ChEMBL. | 10841802 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.