Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Trypanosoma brucei | beta tubulin | 0.0147 | 0.5 | 0.5 |
Toxoplasma gondii | beta-tubulin, putative | 0.0147 | 0.5 | 0.5 |
Echinococcus granulosus | tubulin subunit beta | 0.0147 | 0.5 | 0.5 |
Loa Loa (eye worm) | tubulin beta chain | 0.0147 | 0.5 | 0.5 |
Echinococcus granulosus | beta tubulin | 0.0147 | 0.5 | 0.5 |
Loa Loa (eye worm) | BEN-1 protein | 0.0147 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0147 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0147 | 0.5 | 0.5 |
Echinococcus granulosus | tubulin beta 1 chain | 0.0147 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0147 | 0.5 | 0.5 |
Trypanosoma brucei | beta tubulin | 0.0147 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0147 | 0.5 | 0.5 |
Toxoplasma gondii | beta-1 tubulin, putative | 0.0147 | 0.5 | 0.5 |
Trypanosoma brucei | beta tubulin | 0.0147 | 0.5 | 0.5 |
Giardia lamblia | Beta tubulin | 0.0147 | 0.5 | 0.5 |
Schistosoma mansoni | tubulin subunit beta | 0.0147 | 0.5 | 0.5 |
Echinococcus multilocularis | tubulin beta 1 chain | 0.0147 | 0.5 | 0.5 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0147 | 0.5 | 0.5 |
Echinococcus granulosus | beta tubulin | 0.0147 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0147 | 0.5 | 0.5 |
Trypanosoma cruzi | beta tubulin, putative | 0.0147 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0147 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0147 | 0.5 | 0.5 |
Giardia lamblia | Beta tubulin | 0.0147 | 0.5 | 0.5 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0147 | 0.5 | 0.5 |
Schistosoma mansoni | tubulin subunit beta | 0.0147 | 0.5 | 0.5 |
Echinococcus multilocularis | tubulin, beta 4A class IVa | 0.0147 | 0.5 | 0.5 |
Schistosoma mansoni | tubulin subunit beta | 0.0147 | 0.5 | 0.5 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0147 | 0.5 | 0.5 |
Loa Loa (eye worm) | BEN-1 protein | 0.0147 | 0.5 | 0.5 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0147 | 0.5 | 0.5 |
Entamoeba histolytica | tubulin family protein | 0.0147 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0147 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0147 | 0.5 | 0.5 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0147 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0147 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0147 | 0.5 | 0.5 |
Plasmodium falciparum | tubulin beta chain | 0.0147 | 0.5 | 0.5 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0147 | 0.5 | 0.5 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0147 | 0.5 | 0.5 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0147 | 0.5 | 0.5 |
Echinococcus multilocularis | beta tubulin | 0.0147 | 0.5 | 0.5 |
Trichomonas vaginalis | tubulin, putative | 0.0147 | 0.5 | 0.5 |
Plasmodium vivax | tubulin beta chain, putative | 0.0147 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0147 | 0.5 | 0.5 |
Toxoplasma gondii | beta tubulin | 0.0147 | 0.5 | 0.5 |
Brugia malayi | beta-tubulin, identical | 0.0147 | 0.5 | 0.5 |
Schistosoma mansoni | tubulin subunit beta | 0.0147 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0147 | 0.5 | 0.5 |
Echinococcus multilocularis | beta tubulin | 0.0147 | 0.5 | 0.5 |
Giardia lamblia | Beta tubulin | 0.0147 | 0.5 | 0.5 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0147 | 0.5 | 0.5 |
Entamoeba histolytica | tubulin family protein | 0.0147 | 0.5 | 0.5 |
Schistosoma mansoni | tubulin subunit beta | 0.0147 | 0.5 | 0.5 |
Loa Loa (eye worm) | tubulin beta-1 chain | 0.0147 | 0.5 | 0.5 |
Loa Loa (eye worm) | beta-tubulin | 0.0147 | 0.5 | 0.5 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0147 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0147 | 0.5 | 0.5 |
Echinococcus granulosus | tubulin beta 4A class IVa | 0.0147 | 0.5 | 0.5 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0147 | 0.5 | 0.5 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0147 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0147 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0147 | 0.5 | 0.5 |
Trypanosoma brucei | beta tubulin | 0.0147 | 0.5 | 0.5 |
Loa Loa (eye worm) | tubulin beta-2A chain | 0.0147 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0147 | 0.5 | 0.5 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0147 | 0.5 | 0.5 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0147 | 0.5 | 0.5 |
Echinococcus multilocularis | tubulin subunit beta | 0.0147 | 0.5 | 0.5 |
Loa Loa (eye worm) | tubulin beta-4 chain | 0.0147 | 0.5 | 0.5 |
Schistosoma mansoni | tubulin subunit beta | 0.0147 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0147 | 0.5 | 0.5 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0147 | 0.5 | 0.5 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
GI50 (functional) | = 7 uM | Cytotoxicity against human NCI-H23 cells after 48 hrs by sulforhodamine B assay | ChEMBL. | 23964644 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.