Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Trypanosoma brucei | Heat shock protein 83, putative | 0.1671 | 1 | 1 |
Trichomonas vaginalis | heat shock protein, putative | 0.1331 | 0.655 | 0.655 |
Entamoeba histolytica | heat shock protein 90, putative | 0.1671 | 1 | 1 |
Echinococcus multilocularis | heat shock protein | 0.1671 | 1 | 1 |
Echinococcus multilocularis | heat shock protein 90 | 0.1331 | 0.655 | 0.655 |
Schistosoma mansoni | endoplasmin | 0.1671 | 1 | 1 |
Trypanosoma cruzi | heat shock protein 90, putative | 0.1331 | 0.655 | 0.655 |
Trypanosoma cruzi | heat shock protein 85, putative | 0.1331 | 0.655 | 0.655 |
Echinococcus multilocularis | endoplasmin | 0.1331 | 0.655 | 0.655 |
Leishmania major | heat shock protein 83-1 | 0.1671 | 1 | 1 |
Trypanosoma brucei | heat shock protein, putative | 0.1671 | 1 | 1 |
Trichomonas vaginalis | endoplasmin, putative | 0.1025 | 0.345 | 0.345 |
Plasmodium falciparum | endoplasmin, putative | 0.1025 | 0.345 | 0.345 |
Leishmania major | heat shock protein 83-1 | 0.1671 | 1 | 1 |
Brugia malayi | heat shock protein 90 | 0.1671 | 1 | 1 |
Trypanosoma brucei | heat shock protein, putative | 0.1671 | 1 | 1 |
Leishmania major | heat shock protein 83-1 | 0.1671 | 1 | 1 |
Leishmania major | heat shock protein 83-1 | 0.1671 | 1 | 1 |
Mycobacterium leprae | PROBABLE CHAPERONE PROTEIN HTPG (HEAT SHOCK PROTEIN) (HSP90 FAMILY PROTEIN) (HIGH TEMPERATURE PROTEIN G) | 0.1331 | 0.655 | 0.5 |
Leishmania major | heat shock protein 83-1 | 0.1671 | 1 | 1 |
Wolbachia endosymbiont of Brugia malayi | heat shock protein 90 | 0.1331 | 0.655 | 0.5 |
Trypanosoma cruzi | heat shock protein 90, putative | 0.1671 | 1 | 1 |
Trypanosoma brucei | heat shock protein, putative | 0.1671 | 1 | 1 |
Echinococcus granulosus | heat shock protein | 0.1671 | 1 | 1 |
Trypanosoma brucei | heat shock protein 90, putative | 0.1671 | 1 | 1 |
Toxoplasma gondii | heat shock protein 90, putative | 0.1671 | 1 | 1 |
Trichomonas vaginalis | heat shock protein, putative | 0.1671 | 1 | 1 |
Plasmodium falciparum | heat shock protein 90 | 0.1671 | 1 | 1 |
Trypanosoma cruzi | heat shock protein 90, putative | 0.0987 | 0.3058 | 0.3058 |
Echinococcus multilocularis | heat shock protein 90 | 0.1671 | 1 | 1 |
Leishmania major | heat shock protein 83-1 | 0.1671 | 1 | 1 |
Leishmania major | heat shock protein 83-1 | 0.1671 | 1 | 1 |
Plasmodium vivax | heat shock protein 86, putative | 0.1671 | 1 | 1 |
Leishmania major | heat shock protein 83-1 | 0.1671 | 1 | 1 |
Onchocerca volvulus | Heat shock protein 75 kDa, mitochondrial homolog | 0.0685 | 0 | 0.5 |
Entamoeba histolytica | heat shock protein 90, putative | 0.1671 | 1 | 1 |
Trypanosoma brucei | heat shock protein 90, putative | 0.1671 | 1 | 1 |
Mycobacterium tuberculosis | Probable chaperone protein HtpG (heat shock protein) (HSP90 family protein) (high temperature protein G) | 0.1331 | 0.655 | 0.5 |
Echinococcus granulosus | heat shock protein 90 | 0.1671 | 1 | 1 |
Giardia lamblia | Heat shock protein HSP 90-alpha | 0.1671 | 1 | 1 |
Trichomonas vaginalis | heat shock protein, putative | 0.1331 | 0.655 | 0.655 |
Trypanosoma brucei | heat shock protein, putative | 0.1671 | 1 | 1 |
Trichomonas vaginalis | heat shock protein, putative | 0.1025 | 0.345 | 0.345 |
Leishmania major | heat shock protein 83-1 | 0.1671 | 1 | 1 |
Schistosoma mansoni | heat shock protein | 0.1671 | 1 | 1 |
Echinococcus granulosus | heat shock protein heat shock protein 90 alpha | 0.1331 | 0.655 | 0.655 |
Trypanosoma cruzi | heat shock protein 85, putative | 0.1671 | 1 | 1 |
Mycobacterium ulcerans | heat shock protein 90 | 0.1331 | 0.655 | 0.5 |
Leishmania major | heat shock protein 83-1 | 0.1671 | 1 | 1 |
Plasmodium vivax | endoplasmin, putative | 0.1671 | 1 | 1 |
Loa Loa (eye worm) | heat shock protein 90 | 0.1671 | 1 | 1 |
Schistosoma mansoni | heat shock protein | 0.1671 | 1 | 1 |
Trypanosoma brucei | heat shock protein, putative | 0.1671 | 1 | 1 |
Treponema pallidum | heat shock protein 90 | 0.1331 | 0.655 | 0.5 |
Leishmania major | heat shock protein 83-1 | 0.1671 | 1 | 1 |
Echinococcus granulosus | heat shock protein 90 | 0.1331 | 0.655 | 0.655 |
Leishmania major | lipophosphoglycan biosynthetic protein, putative,heat shock protein 90, putative,glucose regulated protein 94, putative | 0.1331 | 0.655 | 0.655 |
Trichomonas vaginalis | heat shock protein, putative | 0.1331 | 0.655 | 0.655 |
Leishmania major | heat shock protein 83-1 | 0.1671 | 1 | 1 |
Schistosoma mansoni | endoplasmin | 0.1671 | 1 | 1 |
Leishmania major | heat shock protein 83-1 | 0.1671 | 1 | 1 |
Trypanosoma cruzi | heat shock protein 85, putative | 0.1671 | 1 | 1 |
Trypanosoma brucei | heat shock protein, putative | 0.1671 | 1 | 1 |
Toxoplasma gondii | heat shock protein HSP90 | 0.1671 | 1 | 1 |
Leishmania major | heat shock protein 83-1 | 0.1671 | 1 | 1 |
Trypanosoma cruzi | heat shock protein 85, putative | 0.1671 | 1 | 1 |
Trypanosoma cruzi | Heat shock protein 83, putative | 0.1671 | 1 | 1 |
Leishmania major | heat shock protein 83-1 | 0.1671 | 1 | 1 |
Leishmania major | heat shock protein 83-1 | 0.1671 | 1 | 1 |
Loa Loa (eye worm) | endoplasmin | 0.1671 | 1 | 1 |
Trypanosoma brucei | heat shock protein, putative | 0.1671 | 1 | 1 |
Leishmania major | heat shock protein 83-1 | 0.1671 | 1 | 1 |
Trypanosoma brucei | heat shock protein, putative | 0.1671 | 1 | 1 |
Echinococcus granulosus | endoplasmin | 0.1331 | 0.655 | 0.655 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
IC50 (functional) | = 177 uM | Antiplasmodial activity against intraerythrocytic Plasmodium falciparum 3D7 infected in human erythrocytes in fresh RPMI-1640 culture medium assessed as parasite growth inhibition after 96 hrs by microscopic analysis in presence of pantetheinase | ChEMBL. | 24900746 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.