Species | Target name | Source | Bibliographic reference |
---|---|---|---|
Rattus norvegicus | Sigma opioid receptor | Starlite/ChEMBL | References |
Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Echinococcus granulosus | calcium:calmodulin dependent protein kinase | 0.0085 | 0.1008 | 0.2273 |
Loa Loa (eye worm) | TTK protein kinase | 0.0222 | 0.4435 | 0.4435 |
Brugia malayi | Protein kinase domain containing protein | 0.0222 | 0.4435 | 0.4435 |
Echinococcus multilocularis | Glutaredoxin protein 5 | 0.0082 | 0.0949 | 0.2141 |
Trichomonas vaginalis | AGC family protein kinase | 0.0135 | 0.2263 | 0.5104 |
Giardia lamblia | Kinase, TTK | 0.0222 | 0.4435 | 1 |
Brugia malayi | Protein kinase domain containing protein | 0.0135 | 0.2263 | 0.2263 |
Loa Loa (eye worm) | AGC/AKT protein kinase | 0.0135 | 0.2263 | 0.2263 |
Echinococcus granulosus | Glutaredoxin protein 5 | 0.0082 | 0.0949 | 0.2141 |
Echinococcus granulosus | sodium:potassium dependent atpase beta subunit | 0.0082 | 0.0949 | 0.2141 |
Trichomonas vaginalis | AGC family protein kinase | 0.0135 | 0.2263 | 0.5104 |
Trichomonas vaginalis | CAMK family protein kinase | 0.0222 | 0.4435 | 1 |
Echinococcus multilocularis | sodium:potassium dependent atpase beta subunit | 0.0082 | 0.0949 | 0.2141 |
Entamoeba histolytica | protein kinase, putative | 0.0127 | 0.2057 | 0.909 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.0093 | 0.1214 | 0.5363 |
Echinococcus multilocularis | nervana 2 | 0.0082 | 0.0949 | 0.2141 |
Trichomonas vaginalis | AGC family protein kinase | 0.0135 | 0.2263 | 0.5104 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.0093 | 0.1214 | 0.5363 |
Trichomonas vaginalis | AGC family protein kinase | 0.0135 | 0.2263 | 0.5104 |
Trichomonas vaginalis | AGC family protein kinase | 0.0135 | 0.2263 | 0.5104 |
Toxoplasma gondii | AGC kinase | 0.0127 | 0.2057 | 0.5 |
Schistosoma mansoni | serine/threonine-protein kinase | 0.0093 | 0.1214 | 0.2737 |
Echinococcus multilocularis | serine threonine protein kinase nrc serine threonine protein kinase gad | 0.0085 | 0.1008 | 0.2273 |
Trichomonas vaginalis | AGC family protein kinase | 0.0053 | 0.0206 | 0.0464 |
Echinococcus granulosus | serine threonine protein kinase nrc | 0.0085 | 0.1008 | 0.2273 |
Trypanosoma cruzi | Protein kinase B | 0.0093 | 0.1214 | 0.0229 |
Brugia malayi | p70 ribosomal S6 kinase beta | 0.0127 | 0.2057 | 0.2057 |
Onchocerca volvulus | Dual specificity protein kinase TTK homolog | 0.0222 | 0.4435 | 0.5 |
Entamoeba histolytica | protein kinase 2, putative | 0.0085 | 0.1008 | 0.4453 |
Echinococcus multilocularis | nervana 2 | 0.0082 | 0.0949 | 0.2141 |
Plasmodium falciparum | RAC-beta serine/threonine protein kinase | 0.0085 | 0.1008 | 0.5 |
Trichomonas vaginalis | AGC family protein kinase | 0.0135 | 0.2263 | 0.5104 |
Entamoeba histolytica | protein kinase, putative | 0.0135 | 0.2263 | 1 |
Plasmodium vivax | rac-beta serine/threonine protein kinase, putative | 0.0085 | 0.1008 | 0.5 |
Loa Loa (eye worm) | hypothetical protein | 0.0227 | 0.4569 | 0.4569 |
Echinococcus granulosus | serine/threonine protein kinase | 0.0093 | 0.1214 | 0.2737 |
Echinococcus granulosus | dual specificity serine:threonine tyrosine | 0.0222 | 0.4435 | 1 |
Loa Loa (eye worm) | AGC/RSK/P70 protein kinase | 0.0127 | 0.2057 | 0.2057 |
Echinococcus granulosus | nervana 2 | 0.0082 | 0.0949 | 0.2141 |
Echinococcus multilocularis | dual specificity serine:threonine tyrosine | 0.0222 | 0.4435 | 1 |
Trypanosoma cruzi | rac serine-threonine kinase, putative | 0.0093 | 0.1214 | 0.0229 |
Echinococcus multilocularis | rac serine:threonine kinase | 0.0093 | 0.1214 | 0.2737 |
Schistosoma mansoni | dual specificity serine/threonine tyrosine kinase | 0.0222 | 0.4435 | 1 |
Echinococcus granulosus | nervana 2 | 0.0082 | 0.0949 | 0.2141 |
Trichomonas vaginalis | CAMK family protein kinase | 0.0222 | 0.4435 | 1 |
Schistosoma mansoni | serine/threonine-protein kinase | 0.0093 | 0.1214 | 0.2737 |
Entamoeba histolytica | protein kinase, putative | 0.0135 | 0.2263 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.0135 | 0.2263 | 0.5104 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
Ki (binding) | = 155 nM | Displacement of [3H](+)-pentazocine from sigma 1 receptor in rat liver homogenate after 120 mins by liquid scintillation counting | ChEMBL. | 24486131 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.