Species | Target name | Source | Bibliographic reference |
---|---|---|---|
Homo sapiens | melanocortin 4 receptor | Starlite/ChEMBL | No references |
Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Echinococcus granulosus | Tubulin beta 2C chain | 0.0027 | 0.5 | 0.5 |
Plasmodium falciparum | tubulin beta chain | 0.0027 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0027 | 0.5 | 0.5 |
Trypanosoma brucei | beta tubulin | 0.0027 | 0.5 | 0.5 |
Schistosoma mansoni | tubulin subunit beta | 0.0027 | 0.5 | 0.5 |
Toxoplasma gondii | beta-tubulin, putative | 0.0027 | 0.5 | 0.5 |
Echinococcus granulosus | tubulin beta 4A class IVa | 0.0027 | 0.5 | 0.5 |
Loa Loa (eye worm) | tubulin beta-2A chain | 0.0027 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0027 | 0.5 | 0.5 |
Loa Loa (eye worm) | BEN-1 protein | 0.0027 | 0.5 | 0.5 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0027 | 0.5 | 0.5 |
Echinococcus granulosus | beta tubulin | 0.0027 | 0.5 | 0.5 |
Echinococcus granulosus | beta tubulin | 0.0027 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0027 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0027 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0027 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0027 | 0.5 | 0.5 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0027 | 0.5 | 0.5 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0027 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0027 | 0.5 | 0.5 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0027 | 0.5 | 0.5 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0027 | 0.5 | 0.5 |
Brugia malayi | beta-tubulin, identical | 0.0027 | 0.5 | 0.5 |
Schistosoma mansoni | tubulin subunit beta | 0.0027 | 0.5 | 0.5 |
Echinococcus multilocularis | tubulin beta 1 chain | 0.0027 | 0.5 | 0.5 |
Echinococcus multilocularis | beta tubulin | 0.0027 | 0.5 | 0.5 |
Loa Loa (eye worm) | BEN-1 protein | 0.0027 | 0.5 | 0.5 |
Trypanosoma brucei | beta tubulin | 0.0027 | 0.5 | 0.5 |
Giardia lamblia | Beta tubulin | 0.0027 | 0.5 | 0.5 |
Echinococcus multilocularis | tubulin, beta 4A class IVa | 0.0027 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0027 | 0.5 | 0.5 |
Giardia lamblia | Beta tubulin | 0.0027 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0027 | 0.5 | 0.5 |
Loa Loa (eye worm) | beta-tubulin | 0.0027 | 0.5 | 0.5 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0027 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0027 | 0.5 | 0.5 |
Schistosoma mansoni | tubulin subunit beta | 0.0027 | 0.5 | 0.5 |
Trypanosoma cruzi | beta tubulin, putative | 0.0027 | 0.5 | 0.5 |
Plasmodium vivax | tubulin beta chain, putative | 0.0027 | 0.5 | 0.5 |
Echinococcus granulosus | tubulin beta 1 chain | 0.0027 | 0.5 | 0.5 |
Trypanosoma brucei | beta tubulin | 0.0027 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0027 | 0.5 | 0.5 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0027 | 0.5 | 0.5 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0027 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0027 | 0.5 | 0.5 |
Toxoplasma gondii | beta tubulin | 0.0027 | 0.5 | 0.5 |
Schistosoma mansoni | tubulin subunit beta | 0.0027 | 0.5 | 0.5 |
Echinococcus multilocularis | beta tubulin | 0.0027 | 0.5 | 0.5 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0027 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0027 | 0.5 | 0.5 |
Loa Loa (eye worm) | tubulin beta-1 chain | 0.0027 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0027 | 0.5 | 0.5 |
Trypanosoma brucei | beta tubulin | 0.0027 | 0.5 | 0.5 |
Trichomonas vaginalis | tubulin, putative | 0.0027 | 0.5 | 0.5 |
Entamoeba histolytica | tubulin family protein | 0.0027 | 0.5 | 0.5 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0027 | 0.5 | 0.5 |
Entamoeba histolytica | tubulin family protein | 0.0027 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0027 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0027 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0027 | 0.5 | 0.5 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0027 | 0.5 | 0.5 |
Echinococcus granulosus | tubulin subunit beta | 0.0027 | 0.5 | 0.5 |
Toxoplasma gondii | beta-1 tubulin, putative | 0.0027 | 0.5 | 0.5 |
Schistosoma mansoni | tubulin subunit beta | 0.0027 | 0.5 | 0.5 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0027 | 0.5 | 0.5 |
Loa Loa (eye worm) | tubulin beta-4 chain | 0.0027 | 0.5 | 0.5 |
Echinococcus multilocularis | tubulin subunit beta | 0.0027 | 0.5 | 0.5 |
Schistosoma mansoni | tubulin subunit beta | 0.0027 | 0.5 | 0.5 |
Giardia lamblia | Beta tubulin | 0.0027 | 0.5 | 0.5 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0027 | 0.5 | 0.5 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0027 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0027 | 0.5 | 0.5 |
Loa Loa (eye worm) | tubulin beta chain | 0.0027 | 0.5 | 0.5 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
Ki (binding) | = 20 nM | Competitive Inhibition Assay Using [I125]-NDP-a-MSH | BINDINGDB. | No reference |
Ki (binding) | = 20 nM | Competitive Inhibition Assay | BINDINGDB. | No reference |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.