Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Brugia malayi | Malate dehydrogenase, cytoplasmic | 0.0134 | 0.3565 | 0.3421 |
Leishmania major | malate dehydrogenase | 0.0134 | 0.3565 | 0.3421 |
Leishmania major | malate dehydrogenase, putative | 0.0346 | 1 | 1 |
Leishmania major | glycosomal malate dehydrogenase | 0.0134 | 0.3565 | 0.3421 |
Echinococcus multilocularis | lactate dehydrogenase a | 0.0346 | 1 | 1 |
Plasmodium falciparum | malate dehydrogenase | 0.0346 | 1 | 1 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0134 | 0.3565 | 1 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0134 | 0.3565 | 1 |
Echinococcus multilocularis | L lactate dehydrogenase B chain | 0.0346 | 1 | 1 |
Mycobacterium leprae | PROBABLE MALATE DEHYDROGENASE MDH | 0.0134 | 0.3565 | 1 |
Mycobacterium ulcerans | aldehyde dehydrogenase | 0.0063 | 0.1385 | 0.3832 |
Plasmodium falciparum | lactate dehydrogenase, putative | 0.0134 | 0.3565 | 0.3545 |
Echinococcus granulosus | L lactate dehydrogenase B chain | 0.0346 | 1 | 1 |
Echinococcus multilocularis | cytosolic malate dehydrogenase | 0.0134 | 0.3565 | 0.253 |
Echinococcus multilocularis | L lactate dehydrogenase | 0.0211 | 0.5908 | 0.525 |
Mycobacterium ulcerans | hypothetical protein | 0.0025 | 0.0219 | 0.0534 |
Trypanosoma brucei | glycosomal malate dehydrogenase | 0.0134 | 0.3565 | 1 |
Mycobacterium tuberculosis | Fatty-acid-AMP ligase FadD30 (fatty-acid-AMP synthetase) (fatty-acid-AMP synthase) | 0.0018 | 0.003 | 0.0085 |
Mycobacterium tuberculosis | Probable chain -fatty-acid-CoA ligase FadD13 (fatty-acyl-CoA synthetase) | 0.0025 | 0.0219 | 0.0615 |
Loa Loa (eye worm) | hypothetical protein | 0.0026 | 0.0266 | 0.0237 |
Plasmodium falciparum | ataxin-2 like protein, putative | 0.0026 | 0.0266 | 0.0237 |
Mycobacterium ulcerans | long-chain fatty-acid CoA ligase | 0.0025 | 0.0219 | 0.0534 |
Mycobacterium ulcerans | acyl-CoA synthetase | 0.0025 | 0.0219 | 0.0534 |
Leishmania major | malate dehydrogenase, putative | 0.0134 | 0.3565 | 0.3421 |
Loa Loa (eye worm) | malate dehydrogenase | 0.0134 | 0.3565 | 0.3545 |
Echinococcus multilocularis | lactate dehydrogenase a | 0.0346 | 1 | 1 |
Mycobacterium tuberculosis | Probable fatty-acid-CoA ligase FadD2 (fatty-acid-CoA synthetase) (fatty-acid-CoA synthase) | 0.0025 | 0.0219 | 0.0615 |
Schistosoma mansoni | malate dehydrogenase | 0.0134 | 0.3565 | 0.253 |
Trypanosoma cruzi | glycosomal malate dehydrogenase, putative | 0.0134 | 0.3565 | 1 |
Toxoplasma gondii | lactate dehydrogenase LDH1 | 0.0346 | 1 | 1 |
Echinococcus multilocularis | lactate dehydrogenase protein | 0.0346 | 1 | 1 |
Plasmodium vivax | lactate dehydrogenase | 0.0346 | 1 | 1 |
Plasmodium vivax | malate dehydrogenase, putative | 0.0346 | 1 | 1 |
Schistosoma mansoni | L-lactate dehydrogenase | 0.0346 | 1 | 1 |
Brugia malayi | Probable malate dehydrogenase, mitochondrial precursor | 0.0134 | 0.3565 | 0.3421 |
Loa Loa (eye worm) | hypothetical protein | 0.0025 | 0.0219 | 0.0189 |
Echinococcus multilocularis | cytosolic malate dehydrogenase | 0.0134 | 0.3565 | 0.253 |
Leishmania major | hypothetical protein, conserved | 0.0026 | 0.0266 | 0.0048 |
Plasmodium vivax | ataxin-2 like protein, putative | 0.0026 | 0.0266 | 0.0237 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0134 | 0.3565 | 1 |
Echinococcus granulosus | lactate dehydrogenase protein | 0.0346 | 1 | 1 |
Trypanosoma brucei | malate dehydrogenase-related | 0.0134 | 0.3565 | 1 |
Loa Loa (eye worm) | malate dehydrogenase | 0.0134 | 0.3565 | 0.3545 |
Mycobacterium ulcerans | fatty-acid-CoA ligase | 0.0025 | 0.0219 | 0.0534 |
Mycobacterium ulcerans | long-chain-fatty-acid--CoA ligase | 0.0025 | 0.0219 | 0.0534 |
Toxoplasma gondii | aldehyde dehydrogenase | 0.0063 | 0.1385 | 0.1149 |
Plasmodium vivax | lactate/malate dehydrogenase, putative | 0.0134 | 0.3565 | 0.3545 |
Echinococcus granulosus | malate dehydrogenase | 0.0134 | 0.3565 | 0.253 |
Echinococcus granulosus | cytosolic malate dehydrogenase | 0.0134 | 0.3565 | 0.253 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0134 | 0.3565 | 1 |
Leishmania major | aldehyde dehydrogenase, mitochondrial precursor | 0.0063 | 0.1385 | 0.1192 |
Loa Loa (eye worm) | hypothetical protein | 0.0025 | 0.0219 | 0.0189 |
Echinococcus granulosus | malate dehydrogenase | 0.0134 | 0.3565 | 0.253 |
Trichomonas vaginalis | malate and lactate dehydrogenase, putative | 0.0134 | 0.3565 | 1 |
Trypanosoma cruzi | mitochondrial malate dehydrogenase, putative | 0.0134 | 0.3565 | 1 |
Giardia lamblia | Malate dehydrogenase | 0.0134 | 0.3565 | 0.5 |
Schistosoma mansoni | malate dehydrogenase | 0.0134 | 0.3565 | 0.253 |
Trypanosoma brucei | mitochondrial malate dehydrogenase | 0.0134 | 0.3565 | 1 |
Echinococcus multilocularis | lactate dehydrogenase a | 0.0346 | 1 | 1 |
Echinococcus multilocularis | malate dehydrogenase | 0.0134 | 0.3565 | 0.253 |
Trypanosoma cruzi | cytosolic malate dehydrogenase, putative | 0.0134 | 0.3565 | 1 |
Brugia malayi | hypothetical protein | 0.0026 | 0.0266 | 0.0048 |
Echinococcus multilocularis | malate dehydrogenase | 0.0134 | 0.3565 | 0.253 |
Trichomonas vaginalis | malate and lactate dehydrogenase, putative | 0.0134 | 0.3565 | 1 |
Trypanosoma cruzi | malate dehydrogenase, putative | 0.0134 | 0.3565 | 1 |
Leishmania major | mitochondrial malate dehydrogenase | 0.0134 | 0.3565 | 0.3421 |
Loa Loa (eye worm) | hypothetical protein | 0.0346 | 1 | 1 |
Entamoeba histolytica | malate dehydrogenase,cytoplasmic, putative | 0.0134 | 0.3565 | 0.3421 |
Entamoeba histolytica | malate dehydrogenase, putative | 0.0134 | 0.3565 | 0.3421 |
Echinococcus granulosus | lactate dehydrogenase a | 0.0346 | 1 | 1 |
Schistosoma mansoni | malate dehydrogenase | 0.0134 | 0.3565 | 0.253 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0134 | 0.3565 | 1 |
Plasmodium falciparum | ataxin-2 like protein, putative | 0.0026 | 0.0266 | 0.0237 |
Mycobacterium ulcerans | malate dehydrogenase | 0.0134 | 0.3565 | 1 |
Echinococcus granulosus | L lactate dehydrogenase | 0.0211 | 0.5908 | 0.525 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0134 | 0.3565 | 1 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0134 | 0.3565 | 1 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0134 | 0.3565 | 1 |
Mycobacterium ulcerans | long-chain-fatty-acid-CoA ligase | 0.0025 | 0.0219 | 0.0534 |
Mycobacterium ulcerans | aldehyde dehydrogenase | 0.0063 | 0.1385 | 0.3832 |
Toxoplasma gondii | lactate dehydrogenase LDH2 | 0.0346 | 1 | 1 |
Leishmania major | cytosolic malate dehydrogenase | 0.0134 | 0.3565 | 0.3421 |
Loa Loa (eye worm) | hypothetical protein | 0.0025 | 0.0219 | 0.0189 |
Toxoplasma gondii | malate dehydrogenase MDH | 0.0346 | 1 | 1 |
Trypanosoma cruzi | cytosolic malate dehydrogenase, putative | 0.0134 | 0.3565 | 1 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0134 | 0.3565 | 1 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0134 | 0.3565 | 1 |
Mycobacterium ulcerans | acyl-CoA synthetase | 0.0025 | 0.0219 | 0.0534 |
Mycobacterium tuberculosis | Probable malate dehydrogenase Mdh | 0.0134 | 0.3565 | 1 |
Echinococcus granulosus | cytosolic malate dehydrogenase | 0.0134 | 0.3565 | 0.253 |
Entamoeba histolytica | malate dehydrogenase, putative | 0.0346 | 1 | 1 |
Trichomonas vaginalis | malate and lactate dehydrogenase, putative | 0.0134 | 0.3565 | 1 |
Echinococcus granulosus | lactate dehydrogenase a | 0.0346 | 1 | 1 |
Schistosoma mansoni | L-lactate dehydrogenase | 0.0134 | 0.3565 | 0.253 |
Trypanosoma brucei | cytosolic malate dehydrogenase | 0.0134 | 0.3565 | 1 |
Trypanosoma cruzi | malate dehydrogenase, putative | 0.0134 | 0.3565 | 1 |
Plasmodium falciparum | L-lactate dehydrogenase | 0.0346 | 1 | 1 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0134 | 0.3565 | 1 |
Mycobacterium ulcerans | aldehyde dehydrogenase | 0.0063 | 0.1385 | 0.3832 |
Onchocerca volvulus | 0.0025 | 0.0219 | 0.5 | |
Chlamydia trachomatis | malate dehydrogenase | 0.0134 | 0.3565 | 1 |
Trypanosoma cruzi | glycosomal malate dehydrogenase, putative | 0.0134 | 0.3565 | 1 |
Trichomonas vaginalis | malate and lactate dehydrogenase, putative | 0.0134 | 0.3565 | 1 |
Mycobacterium ulcerans | acyl-CoA synthetase | 0.0025 | 0.0219 | 0.0534 |
Schistosoma mansoni | malate dehydrogenase | 0.0346 | 1 | 1 |
Wolbachia endosymbiont of Brugia malayi | malate dehydrogenase | 0.0346 | 1 | 0.5 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0134 | 0.3565 | 1 |
Mycobacterium tuberculosis | Probable aldehyde dehydrogenase | 0.0063 | 0.1385 | 0.3885 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
pKB (binding) | = 10 | In vitro inhibition of ATII induced contractions of the isolated rabbit aorta. | ChEMBL. | No reference |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.