Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Leishmania major | glycosomal malate dehydrogenase | 0.0084 | 0.6708 | 0.6372 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0091 | 0.8878 | 1 |
Toxoplasma gondii | lactate dehydrogenase LDH1 | 0.0095 | 1 | 0.5 |
Trypanosoma brucei | glycosomal malate dehydrogenase | 0.0084 | 0.6708 | 0.7271 |
Chlamydia trachomatis | malate dehydrogenase | 0.0091 | 0.8878 | 0.5 |
Plasmodium falciparum | malate dehydrogenase | 0.0095 | 1 | 1 |
Plasmodium falciparum | L-lactate dehydrogenase | 0.0095 | 1 | 1 |
Trypanosoma cruzi | glycosomal malate dehydrogenase, putative | 0.0084 | 0.6708 | 0.7271 |
Giardia lamblia | Malate dehydrogenase | 0.0091 | 0.8878 | 0.5 |
Echinococcus granulosus | lactate dehydrogenase a | 0.0095 | 1 | 1 |
Loa Loa (eye worm) | malate dehydrogenase | 0.0091 | 0.8878 | 0.6591 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0091 | 0.8878 | 1 |
Trypanosoma brucei | mitochondrial malate dehydrogenase | 0.0084 | 0.6708 | 0.7271 |
Trypanosoma brucei | cytosolic malate dehydrogenase | 0.0091 | 0.8878 | 1 |
Trypanosoma cruzi | cytosolic malate dehydrogenase, putative | 0.0091 | 0.8878 | 1 |
Echinococcus multilocularis | cytosolic malate dehydrogenase | 0.0091 | 0.8878 | 0.6591 |
Entamoeba histolytica | malate dehydrogenase, putative | 0.0095 | 1 | 1 |
Schistosoma mansoni | malate dehydrogenase | 0.0091 | 0.8878 | 0.8763 |
Echinococcus granulosus | cytosolic malate dehydrogenase | 0.0091 | 0.8878 | 0.6591 |
Leishmania major | malate dehydrogenase, putative | 0.0095 | 1 | 1 |
Trichomonas vaginalis | malate and lactate dehydrogenase, putative | 0.0091 | 0.8878 | 1 |
Echinococcus granulosus | lactate dehydrogenase protein | 0.0095 | 1 | 1 |
Trypanosoma cruzi | cytosolic malate dehydrogenase, putative | 0.0091 | 0.8878 | 1 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0091 | 0.8878 | 1 |
Leishmania major | mitochondrial malate dehydrogenase | 0.0084 | 0.6708 | 0.6372 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0091 | 0.8878 | 1 |
Toxoplasma gondii | lactate dehydrogenase LDH2 | 0.0095 | 1 | 0.5 |
Trichomonas vaginalis | malate and lactate dehydrogenase, putative | 0.0091 | 0.8878 | 1 |
Echinococcus multilocularis | lactate dehydrogenase a | 0.0095 | 1 | 1 |
Echinococcus granulosus | L lactate dehydrogenase B chain | 0.0095 | 1 | 1 |
Schistosoma mansoni | malate dehydrogenase | 0.0084 | 0.6708 | 0.6372 |
Loa Loa (eye worm) | hypothetical protein | 0.0095 | 1 | 1 |
Schistosoma mansoni | malate dehydrogenase | 0.0095 | 1 | 1 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0091 | 0.8878 | 1 |
Echinococcus multilocularis | lactate dehydrogenase a | 0.0095 | 1 | 1 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0091 | 0.8878 | 1 |
Mycobacterium tuberculosis | Probable malate dehydrogenase Mdh | 0.0091 | 0.8878 | 0.5 |
Trypanosoma cruzi | glycosomal malate dehydrogenase, putative | 0.0084 | 0.6708 | 0.7271 |
Echinococcus multilocularis | L lactate dehydrogenase B chain | 0.0095 | 1 | 1 |
Leishmania major | malate dehydrogenase | 0.0084 | 0.6708 | 0.6372 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0091 | 0.8878 | 1 |
Echinococcus granulosus | lactate dehydrogenase a | 0.0095 | 1 | 1 |
Wolbachia endosymbiont of Brugia malayi | malate dehydrogenase | 0.0095 | 1 | 0.5 |
Trichomonas vaginalis | malate and lactate dehydrogenase, putative | 0.0091 | 0.8878 | 1 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0063 | 0.0926 | 0.1043 |
Schistosoma mansoni | L-lactate dehydrogenase | 0.0095 | 1 | 1 |
Mycobacterium leprae | PROBABLE MALATE DEHYDROGENASE MDH | 0.0091 | 0.8878 | 0.5 |
Leishmania major | cytosolic malate dehydrogenase | 0.0091 | 0.8878 | 0.8763 |
Trypanosoma cruzi | mitochondrial malate dehydrogenase, putative | 0.0084 | 0.6708 | 0.7271 |
Schistosoma mansoni | malate dehydrogenase | 0.0091 | 0.8878 | 0.8763 |
Mycobacterium ulcerans | malate dehydrogenase | 0.0091 | 0.8878 | 0.5 |
Plasmodium vivax | malate dehydrogenase, putative | 0.0095 | 1 | 1 |
Echinococcus multilocularis | cytosolic malate dehydrogenase | 0.0091 | 0.8878 | 0.6591 |
Trypanosoma cruzi | malate dehydrogenase, putative | 0.0084 | 0.6708 | 0.7271 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0091 | 0.8878 | 1 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0091 | 0.8878 | 1 |
Toxoplasma gondii | malate dehydrogenase MDH | 0.0095 | 1 | 0.5 |
Echinococcus multilocularis | lactate dehydrogenase protein | 0.0095 | 1 | 1 |
Plasmodium vivax | lactate dehydrogenase | 0.0095 | 1 | 1 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0091 | 0.8878 | 1 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0091 | 0.8878 | 1 |
Echinococcus granulosus | cytosolic malate dehydrogenase | 0.0091 | 0.8878 | 0.6591 |
Trichomonas vaginalis | malate and lactate dehydrogenase, putative | 0.0091 | 0.8878 | 1 |
Echinococcus multilocularis | lactate dehydrogenase a | 0.0095 | 1 | 1 |
Brugia malayi | Malate dehydrogenase, cytoplasmic | 0.0091 | 0.8878 | 0.6591 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
Decrease (functional) | NA 0 % | Percent decrease in serum haptoglobin evaluated in a developing adjuvant arthritis model rats; No significant effect | ChEMBL. | 1995900 |
Inhibition (functional) | NA 0 % | Compound was evaluated in developing adjuvant arthritis model rats for its effect on paw edema; No significant effect | ChEMBL. | 1995900 |
logP (ADMET) | = 0.23 | Partition coefficient (logP) | ChEMBL. | 1995900 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.