Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0081 | 0.2137 | 0.3282 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0109 | 0.5582 | 1 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0109 | 0.5582 | 1 |
Toxoplasma gondii | lactate dehydrogenase LDH1 | 0.0145 | 1 | 0.5 |
Trypanosoma cruzi | cytosolic malate dehydrogenase, putative | 0.0109 | 0.5582 | 1 |
Leishmania major | malate dehydrogenase, putative | 0.0145 | 1 | 1 |
Schistosoma mansoni | malate dehydrogenase | 0.0109 | 0.5582 | 0.4382 |
Echinococcus granulosus | cytosolic malate dehydrogenase | 0.0109 | 0.5582 | 0.5582 |
Schistosoma mansoni | malate dehydrogenase | 0.0109 | 0.5582 | 0.4382 |
Loa Loa (eye worm) | malate dehydrogenase | 0.0109 | 0.5582 | 0.1755 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0109 | 0.5582 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0145 | 1 | 1 |
Schistosoma mansoni | L-lactate dehydrogenase | 0.0145 | 1 | 1 |
Toxoplasma gondii | malate dehydrogenase MDH | 0.0145 | 1 | 0.5 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0109 | 0.5582 | 1 |
Trypanosoma cruzi | glycosomal malate dehydrogenase, putative | 0.0102 | 0.4642 | 0.7271 |
Echinococcus multilocularis | cytosolic malate dehydrogenase | 0.0109 | 0.5582 | 0.5582 |
Echinococcus granulosus | malate dehydrogenase | 0.0102 | 0.4642 | 0.4642 |
Schistosoma mansoni | malate dehydrogenase | 0.0102 | 0.4642 | 0.3186 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0109 | 0.5582 | 1 |
Trypanosoma cruzi | malate dehydrogenase, putative | 0.0102 | 0.4642 | 0.7271 |
Plasmodium vivax | malate dehydrogenase, putative | 0.0145 | 1 | 1 |
Trichomonas vaginalis | malate and lactate dehydrogenase, putative | 0.0109 | 0.5582 | 1 |
Echinococcus multilocularis | lactate dehydrogenase a | 0.0145 | 1 | 1 |
Leishmania major | malate dehydrogenase | 0.0102 | 0.4642 | 0.3186 |
Mycobacterium leprae | PROBABLE MALATE DEHYDROGENASE MDH | 0.0109 | 0.5582 | 0.5 |
Echinococcus granulosus | lactate dehydrogenase a | 0.0145 | 1 | 1 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0109 | 0.5582 | 1 |
Echinococcus multilocularis | L lactate dehydrogenase B chain | 0.0145 | 1 | 1 |
Chlamydia trachomatis | malate dehydrogenase | 0.0109 | 0.5582 | 0.5 |
Trypanosoma brucei | mitochondrial malate dehydrogenase | 0.0102 | 0.4642 | 0.7271 |
Echinococcus multilocularis | malate dehydrogenase | 0.0102 | 0.4642 | 0.4642 |
Plasmodium falciparum | malate dehydrogenase | 0.0145 | 1 | 1 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0109 | 0.5582 | 1 |
Trypanosoma brucei | glycosomal malate dehydrogenase | 0.0102 | 0.4642 | 0.7271 |
Echinococcus multilocularis | lactate dehydrogenase a | 0.0145 | 1 | 1 |
Echinococcus multilocularis | lactate dehydrogenase a | 0.0145 | 1 | 1 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0109 | 0.5582 | 1 |
Leishmania major | cytosolic malate dehydrogenase | 0.0109 | 0.5582 | 0.4382 |
Toxoplasma gondii | lactate dehydrogenase LDH2 | 0.0145 | 1 | 0.5 |
Trichomonas vaginalis | malate and lactate dehydrogenase, putative | 0.0109 | 0.5582 | 1 |
Echinococcus granulosus | L lactate dehydrogenase B chain | 0.0145 | 1 | 1 |
Mycobacterium tuberculosis | Probable malate dehydrogenase Mdh | 0.0109 | 0.5582 | 0.5 |
Brugia malayi | Malate dehydrogenase, cytoplasmic | 0.0109 | 0.5582 | 0.1755 |
Echinococcus granulosus | lactate dehydrogenase a | 0.0145 | 1 | 1 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0109 | 0.5582 | 1 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0109 | 0.5582 | 1 |
Schistosoma mansoni | malate dehydrogenase | 0.0145 | 1 | 1 |
Wolbachia endosymbiont of Brugia malayi | malate dehydrogenase | 0.0145 | 1 | 0.5 |
Trypanosoma cruzi | cytosolic malate dehydrogenase, putative | 0.0109 | 0.5582 | 1 |
Trypanosoma cruzi | glycosomal malate dehydrogenase, putative | 0.0102 | 0.4642 | 0.7271 |
Leishmania major | mitochondrial malate dehydrogenase | 0.0102 | 0.4642 | 0.3186 |
Trypanosoma brucei | cytosolic malate dehydrogenase | 0.0109 | 0.5582 | 1 |
Mycobacterium ulcerans | malate dehydrogenase | 0.0109 | 0.5582 | 0.5 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0109 | 0.5582 | 1 |
Trichomonas vaginalis | malate and lactate dehydrogenase, putative | 0.0109 | 0.5582 | 1 |
Echinococcus multilocularis | lactate dehydrogenase protein | 0.0145 | 1 | 1 |
Trichomonas vaginalis | malate and lactate dehydrogenase, putative | 0.0109 | 0.5582 | 1 |
Giardia lamblia | Malate dehydrogenase | 0.0109 | 0.5582 | 0.5 |
Echinococcus granulosus | lactate dehydrogenase protein | 0.0145 | 1 | 1 |
Echinococcus granulosus | malate dehydrogenase | 0.0102 | 0.4642 | 0.4642 |
Echinococcus multilocularis | malate dehydrogenase | 0.0102 | 0.4642 | 0.4642 |
Plasmodium falciparum | L-lactate dehydrogenase | 0.0145 | 1 | 1 |
Trypanosoma cruzi | mitochondrial malate dehydrogenase, putative | 0.0102 | 0.4642 | 0.7271 |
Plasmodium vivax | lactate dehydrogenase | 0.0145 | 1 | 1 |
Echinococcus granulosus | cytosolic malate dehydrogenase | 0.0109 | 0.5582 | 0.5582 |
Leishmania major | glycosomal malate dehydrogenase | 0.0102 | 0.4642 | 0.3186 |
Echinococcus multilocularis | cytosolic malate dehydrogenase | 0.0109 | 0.5582 | 0.5582 |
Entamoeba histolytica | malate dehydrogenase, putative | 0.0145 | 1 | 1 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
Inhibition (binding) | = 20 % | Displacement of [3H]DPCPX from recombinant human adenosine A2B receptor expressed in HeLa cells at 0.01 uM | ChEMBL. | 16392813 |
Inhibition (binding) | = 20 % | Displacement of [3H]DPCPX from recombinant human adenosine A2B receptor expressed in HeLa cells at 0.01 uM | ChEMBL. | 16392813 |
Inhibition (binding) | = 45 % | Displacement of [3H]ZM241385 from recombinant human adenosine A2A receptor expressed in HEK293 cells at 0.1 uM | ChEMBL. | 16392813 |
Inhibition (binding) | = 45 % | Displacement of [3H]ZM241385 from recombinant human adenosine A2A receptor expressed in HEK293 cells at 0.1 uM | ChEMBL. | 16392813 |
Inhibition (binding) | = 68 % | Displacement of [3H]DPCPX from recombinant human adenosine A2B receptor expressed in HEK293 cells at 0.1 uM | ChEMBL. | 16392813 |
Inhibition (binding) | = 68 % | Displacement of [3H]DPCPX from recombinant human adenosine A2B receptor expressed in HEK293 cells at 0.1 uM | ChEMBL. | 16392813 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.