Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Leishmania major | beta tubulin | 0.0251 | 0.3641 | 0.5 |
Leishmania major | beta tubulin | 0.0251 | 0.3641 | 0.5 |
Schistosoma mansoni | tubulin subunit beta | 0.0251 | 0.3641 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0251 | 0.3641 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0251 | 0.3641 | 1 |
Plasmodium vivax | tubulin beta chain, putative | 0.0251 | 0.3641 | 0.5 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0251 | 0.3641 | 0.5 |
Onchocerca volvulus | 0.0082 | 0 | 0.5 | |
Leishmania major | beta tubulin | 0.0251 | 0.3641 | 0.5 |
Echinococcus multilocularis | tubulin, beta 4A class IVa | 0.0251 | 0.3641 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0251 | 0.3641 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0251 | 0.3641 | 1 |
Onchocerca volvulus | 0.0082 | 0 | 0.5 | |
Toxoplasma gondii | beta-tubulin, putative | 0.0251 | 0.3641 | 0.5 |
Onchocerca volvulus | Dopamine\/Ecdysteroid receptor homolog | 0.0082 | 0 | 0.5 |
Trypanosoma brucei | beta tubulin | 0.0251 | 0.3641 | 0.5 |
Plasmodium falciparum | tubulin beta chain | 0.0251 | 0.3641 | 0.5 |
Loa Loa (eye worm) | follicle stimulating hormone receptor | 0.0545 | 1 | 1 |
Echinococcus granulosus | tubulin beta 4A class IVa | 0.0251 | 0.3641 | 1 |
Leishmania major | beta tubulin | 0.0251 | 0.3641 | 0.5 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0251 | 0.3641 | 0.5 |
Leishmania major | beta tubulin | 0.0251 | 0.3641 | 0.5 |
Entamoeba histolytica | tubulin family protein | 0.0251 | 0.3641 | 0.5 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0251 | 0.3641 | 1 |
Toxoplasma gondii | beta tubulin | 0.0251 | 0.3641 | 0.5 |
Leishmania major | beta tubulin | 0.0251 | 0.3641 | 0.5 |
Schistosoma mansoni | tubulin subunit beta | 0.0251 | 0.3641 | 1 |
Leishmania major | beta tubulin | 0.0251 | 0.3641 | 0.5 |
Toxoplasma gondii | beta-1 tubulin, putative | 0.0251 | 0.3641 | 0.5 |
Leishmania major | beta tubulin | 0.0251 | 0.3641 | 0.5 |
Brugia malayi | beta-tubulin, identical | 0.0251 | 0.3641 | 0.3641 |
Onchocerca volvulus | 0.0082 | 0 | 0.5 | |
Loa Loa (eye worm) | BEN-1 protein | 0.0251 | 0.3641 | 0.3641 |
Loa Loa (eye worm) | BEN-1 protein | 0.0251 | 0.3641 | 0.3641 |
Schistosoma mansoni | tubulin subunit beta | 0.0251 | 0.3641 | 1 |
Onchocerca volvulus | 0.0082 | 0 | 0.5 | |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0251 | 0.3641 | 1 |
Onchocerca volvulus | 0.0082 | 0 | 0.5 | |
Onchocerca volvulus | 0.0082 | 0 | 0.5 | |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0251 | 0.3641 | 1 |
Echinococcus granulosus | beta tubulin | 0.0251 | 0.3641 | 1 |
Leishmania major | beta tubulin | 0.0251 | 0.3641 | 0.5 |
Onchocerca volvulus | 0.0082 | 0 | 0.5 | |
Loa Loa (eye worm) | tubulin beta-1 chain | 0.0251 | 0.3641 | 0.3641 |
Echinococcus multilocularis | tubulin subunit beta | 0.0251 | 0.3641 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0251 | 0.3641 | 1 |
Giardia lamblia | Beta tubulin | 0.0251 | 0.3641 | 0.5 |
Echinococcus granulosus | tubulin beta 1 chain | 0.0251 | 0.3641 | 1 |
Leishmania major | beta tubulin | 0.0251 | 0.3641 | 0.5 |
Trypanosoma cruzi | beta tubulin, putative | 0.0251 | 0.3641 | 0.5 |
Schistosoma mansoni | tubulin subunit beta | 0.0251 | 0.3641 | 1 |
Trichomonas vaginalis | tubulin, putative | 0.0251 | 0.3641 | 0.5 |
Echinococcus multilocularis | tubulin beta 1 chain | 0.0251 | 0.3641 | 1 |
Giardia lamblia | Beta tubulin | 0.0251 | 0.3641 | 0.5 |
Trypanosoma brucei | beta tubulin | 0.0251 | 0.3641 | 0.5 |
Onchocerca volvulus | 0.0082 | 0 | 0.5 | |
Leishmania major | beta tubulin | 0.0251 | 0.3641 | 0.5 |
Loa Loa (eye worm) | tubulin beta chain | 0.0251 | 0.3641 | 0.3641 |
Echinococcus multilocularis | beta tubulin | 0.0251 | 0.3641 | 1 |
Onchocerca volvulus | 0.0082 | 0 | 0.5 | |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0251 | 0.3641 | 0.5 |
Onchocerca volvulus | 0.0082 | 0 | 0.5 | |
Loa Loa (eye worm) | beta-tubulin | 0.0251 | 0.3641 | 0.3641 |
Echinococcus granulosus | beta tubulin | 0.0251 | 0.3641 | 1 |
Leishmania major | beta tubulin | 0.0251 | 0.3641 | 0.5 |
Schistosoma mansoni | tubulin subunit beta | 0.0251 | 0.3641 | 1 |
Echinococcus granulosus | tubulin subunit beta | 0.0251 | 0.3641 | 1 |
Onchocerca volvulus | 0.0082 | 0 | 0.5 | |
Leishmania major | beta tubulin | 0.0251 | 0.3641 | 0.5 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0251 | 0.3641 | 0.5 |
Loa Loa (eye worm) | tubulin beta-2A chain | 0.0251 | 0.3641 | 0.3641 |
Onchocerca volvulus | 0.0082 | 0 | 0.5 | |
Onchocerca volvulus | 0.0082 | 0 | 0.5 | |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0251 | 0.3641 | 1 |
Onchocerca volvulus | 0.0082 | 0 | 0.5 | |
Echinococcus multilocularis | beta tubulin | 0.0251 | 0.3641 | 1 |
Entamoeba histolytica | tubulin family protein | 0.0251 | 0.3641 | 0.5 |
Onchocerca volvulus | 0.0082 | 0 | 0.5 | |
Leishmania major | beta tubulin | 0.0251 | 0.3641 | 0.5 |
Leishmania major | beta tubulin | 0.0251 | 0.3641 | 0.5 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0251 | 0.3641 | 0.5 |
Brugia malayi | Tubulin beta-1 chain | 0.0251 | 0.3641 | 0.3641 |
Onchocerca volvulus | 0.0082 | 0 | 0.5 | |
Leishmania major | beta tubulin | 0.0251 | 0.3641 | 0.5 |
Leishmania major | beta tubulin | 0.0251 | 0.3641 | 0.5 |
Trypanosoma brucei | beta tubulin | 0.0251 | 0.3641 | 0.5 |
Onchocerca volvulus | 0.0082 | 0 | 0.5 | |
Loa Loa (eye worm) | tubulin beta-4 chain | 0.0251 | 0.3641 | 0.3641 |
Trypanosoma brucei | beta tubulin | 0.0251 | 0.3641 | 0.5 |
Onchocerca volvulus | Neuropeptide F receptor homolog | 0.0082 | 0 | 0.5 |
Giardia lamblia | Beta tubulin | 0.0251 | 0.3641 | 0.5 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0251 | 0.3641 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0251 | 0.3641 | 1 |
Leishmania major | beta tubulin | 0.0251 | 0.3641 | 0.5 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
IC50 (ADMET) | > 200 uM | Cytotoxicity against mouse L1210/0 cells after 48 hrs | ChEMBL. | 17341060 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.