Species | Target name | Source | Bibliographic reference |
---|---|---|---|
Homo sapiens | chemokine (C-X-C motif) receptor 2 | Starlite/ChEMBL | References |
Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Loa Loa (eye worm) | AGC/RSK/P70 protein kinase | 0.0423 | 1 | 1 |
Echinococcus granulosus | serine threonine protein kinase nrc | 0.0282 | 0.4899 | 0.8745 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.0282 | 0.4899 | 0.4899 |
Trypanosoma brucei | rac serine-threonine kinase, putative | 0.0423 | 1 | 0.5 |
Schistosoma mansoni | serine/threonine-protein kinase | 0.0282 | 0.4899 | 0.8745 |
Trichomonas vaginalis | AGC family protein kinase | 0.0423 | 1 | 1 |
Echinococcus multilocularis | 3 phosphoinositide dependent protein kinase 1 | 0.0302 | 0.5602 | 1 |
Loa Loa (eye worm) | AGC/AKT protein kinase | 0.0423 | 1 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.0302 | 0.5602 | 0.5602 |
Trypanosoma cruzi | rac serine-threonine kinase, putative | 0.0282 | 0.4899 | 0.5 |
Giardia lamblia | Kinase, AGC PKA | 0.0282 | 0.4899 | 0.5 |
Trichomonas vaginalis | AGC family protein kinase | 0.0423 | 1 | 1 |
Echinococcus granulosus | nervana 2 | 0.0276 | 0.4684 | 0.8361 |
Echinococcus multilocularis | nervana 2 | 0.0276 | 0.4684 | 0.8361 |
Echinococcus multilocularis | serine threonine protein kinase nrc serine threonine protein kinase gad | 0.0282 | 0.4899 | 0.8745 |
Trichomonas vaginalis | AGC family protein kinase | 0.0423 | 1 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.0423 | 1 | 1 |
Echinococcus multilocularis | nervana 2 | 0.0276 | 0.4684 | 0.8361 |
Brugia malayi | Protein kinase domain containing protein | 0.0423 | 1 | 1 |
Echinococcus granulosus | calcium:calmodulin dependent protein kinase | 0.0282 | 0.4899 | 0.8745 |
Entamoeba histolytica | protein kinase, putative | 0.0423 | 1 | 1 |
Plasmodium vivax | rac-beta serine/threonine protein kinase, putative | 0.0282 | 0.4899 | 0.5 |
Brugia malayi | Protein kinase domain containing protein | 0.0302 | 0.5602 | 0.5602 |
Echinococcus granulosus | sodium:potassium dependent atpase beta subunit | 0.0276 | 0.4684 | 0.8361 |
Loa Loa (eye worm) | AGC/PDK1 protein kinase | 0.0302 | 0.5602 | 0.5602 |
Schistosoma mansoni | serine/threonine protein kinase | 0.0302 | 0.5602 | 1 |
Entamoeba histolytica | protein kinase 2, putative | 0.0282 | 0.4899 | 0.4899 |
Echinococcus multilocularis | Glutaredoxin protein 5 | 0.0276 | 0.4684 | 0.8361 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.0282 | 0.4899 | 0.4899 |
Trichomonas vaginalis | AGC family protein kinase | 0.0423 | 1 | 1 |
Entamoeba histolytica | protein kinase, putative | 0.0302 | 0.5602 | 0.5602 |
Trichomonas vaginalis | AGC family protein kinase | 0.0423 | 1 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.0423 | 1 | 1 |
Echinococcus granulosus | 3-phosphoinositide-dependent protein kinase 1 | 0.0302 | 0.5602 | 1 |
Trypanosoma cruzi | Protein kinase B | 0.0282 | 0.4899 | 0.5 |
Entamoeba histolytica | protein kinase, putative | 0.0423 | 1 | 1 |
Echinococcus multilocularis | sodium:potassium dependent atpase beta subunit | 0.0276 | 0.4684 | 0.8361 |
Entamoeba histolytica | protein kinase, putative | 0.0423 | 1 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.0302 | 0.5602 | 0.5602 |
Schistosoma mansoni | serine/threonine-protein kinase | 0.0282 | 0.4899 | 0.8745 |
Echinococcus granulosus | nervana 2 | 0.0276 | 0.4684 | 0.8361 |
Echinococcus granulosus | serine/threonine protein kinase | 0.0282 | 0.4899 | 0.8745 |
Trypanosoma cruzi | rac serine-threonine kinase, putative | 0.0282 | 0.4899 | 0.5 |
Echinococcus granulosus | Glutaredoxin protein 5 | 0.0276 | 0.4684 | 0.8361 |
Echinococcus multilocularis | rac serine:threonine kinase | 0.0282 | 0.4899 | 0.8745 |
Toxoplasma gondii | AGC kinase | 0.0423 | 1 | 0.5 |
Brugia malayi | phosphoinositide-dependent protein kinase I | 0.0302 | 0.5602 | 0.5602 |
Loa Loa (eye worm) | AGC/PDK1 protein kinase | 0.0302 | 0.5602 | 0.5602 |
Plasmodium falciparum | RAC-beta serine/threonine protein kinase | 0.0282 | 0.4899 | 0.5 |
Trichomonas vaginalis | AGC family protein kinase | 0.0302 | 0.5602 | 0.5602 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
IC50 (binding) | = 5.1 uM | Displacement of human recombinant [125I]IL8 from CXCR2 receptor expressed in CHO cells | ChEMBL. | 17524641 |
IC50 (binding) | = 5.1 uM | Displacement of human recombinant [125I]IL8 from CXCR2 receptor expressed in CHO cells | ChEMBL. | 17524641 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.