Species | Target name | Source | Bibliographic reference |
---|---|---|---|
Homo sapiens | nuclear receptor subfamily 1, group H, member 2 | Starlite/ChEMBL | References |
Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Trichomonas vaginalis | phosphoenolpyruvate carboxykinase, putative | 0.0586 | 0.8675 | 0.7357 |
Echinococcus multilocularis | neuropeptide receptor A26 | 0.0409 | 0.5979 | 0.5299 |
Loa Loa (eye worm) | hypothetical protein | 0.0673 | 1 | 1 |
Trichomonas vaginalis | phosphoenolpyruvate carboxykinase, putative | 0.0673 | 1 | 1 |
Trypanosoma cruzi | cytochrome P450, putative | 0.0017 | 0 | 0.5 |
Onchocerca volvulus | 0.0586 | 0.8675 | 0.5 | |
Mycobacterium ulcerans | aldehyde dehydrogenase | 0.0112 | 0.1447 | 0.1447 |
Echinococcus multilocularis | neuropeptide s receptor | 0.0409 | 0.5979 | 0.5299 |
Trichomonas vaginalis | phosphoenolpyruvate carboxykinase, putative | 0.0673 | 1 | 1 |
Trypanosoma cruzi | cytochrome P450, putative | 0.0017 | 0 | 0.5 |
Echinococcus granulosus | neuropeptide receptor A26 | 0.0409 | 0.5979 | 0.5299 |
Mycobacterium ulcerans | aldehyde dehydrogenase | 0.0112 | 0.1447 | 0.1447 |
Mycobacterium tuberculosis | Probable iron-regulated phosphoenolpyruvate carboxykinase [GTP] PckA (phosphoenolpyruvate carboxylase) (PEPCK)(pep carboxykinase | 0.0673 | 1 | 1 |
Trichomonas vaginalis | phosphoenolpyruvate carboxykinase, putative | 0.0673 | 1 | 1 |
Trichomonas vaginalis | phosphoenolpyruvate carboxykinase, putative | 0.0673 | 1 | 1 |
Chlamydia trachomatis | phosphoenolpyruvate carboxykinase | 0.0673 | 1 | 0.5 |
Giardia lamblia | Phosphoenolpyruvate carboxykinase | 0.0673 | 1 | 0.5 |
Leishmania major | aldehyde dehydrogenase, mitochondrial precursor | 0.0112 | 0.1447 | 1 |
Echinococcus granulosus | phosphoenolpyruvate carboxykinase | 0.0673 | 1 | 1 |
Echinococcus multilocularis | phosphoenolpyruvate carboxykinase | 0.0673 | 1 | 1 |
Loa Loa (eye worm) | phosphoenolpyruvate carboxykinase cytosolic family member | 0.0673 | 1 | 1 |
Brugia malayi | phosphoenolpyruvate carboxykinase [GTP] | 0.0673 | 1 | 1 |
Treponema pallidum | phosphoenolpyruvate carboxykinase | 0.0673 | 1 | 0.5 |
Brugia malayi | hypothetical protein | 0.0257 | 0.366 | 0.366 |
Echinococcus granulosus | neuropeptide s receptor | 0.0409 | 0.5979 | 0.5299 |
Trichomonas vaginalis | phosphoenolpyruvate carboxykinase, putative | 0.0673 | 1 | 1 |
Brugia malayi | Cytochrome P450 family protein | 0.0043 | 0.0397 | 0.0397 |
Mycobacterium leprae | PROBABLE IRON-REGULATED PHOSPHOENOLPYRUVATE CARBOXYKINASE [GTP] PCKA (PHOSPHOENOLPYRUVATE CARBOXYLASE) (PEPCK)(PEP CARBOXYKINASE | 0.0673 | 1 | 0.5 |
Trypanosoma brucei | cytochrome P450, putative | 0.0017 | 0 | 0.5 |
Mycobacterium ulcerans | phosphoenolpyruvate carboxykinase | 0.0673 | 1 | 1 |
Loa Loa (eye worm) | cytochrome P450 family protein | 0.0043 | 0.0397 | 0.0397 |
Mycobacterium ulcerans | aldehyde dehydrogenase | 0.0112 | 0.1447 | 0.1447 |
Trichomonas vaginalis | phosphoenolpyruvate carboxykinase, putative | 0.0586 | 0.8675 | 0.7357 |
Schistosoma mansoni | phosphoenolpyruvate carboxykinase | 0.0673 | 1 | 1 |
Loa Loa (eye worm) | phosphoenolpyruvate carboxykinase | 0.0673 | 1 | 1 |
Toxoplasma gondii | aldehyde dehydrogenase | 0.0112 | 0.1447 | 0.5 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
EC50 (functional) | = 5.6 uM | Agonist activity at human LXRbeta receptor after 1 hr by HTRF cofactor recruitment assay | ChEMBL. | 17587573 |
EC50 (functional) | = 5.6 uM | Agonist activity at human LXRbeta receptor after 1 hr by HTRF cofactor recruitment assay | ChEMBL. | 17587573 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.