Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Trichomonas vaginalis | AGC family protein kinase | 0.0222 | 0.7603 | 0.7603 |
Echinococcus granulosus | sodium:potassium dependent atpase beta subunit | 0.0136 | 0.3296 | 0.3158 |
Entamoeba histolytica | protein kinase, putative | 0.0209 | 0.693 | 0.6866 |
Echinococcus multilocularis | nervana 2 | 0.0136 | 0.3296 | 0.3158 |
Trichomonas vaginalis | AGC family protein kinase | 0.0222 | 0.7603 | 0.7603 |
Echinococcus granulosus | Glutaredoxin protein 5 | 0.0136 | 0.3296 | 0.3158 |
Trichomonas vaginalis | AGC family protein kinase | 0.0073 | 0.0202 | 0.0202 |
Trichomonas vaginalis | AGC family protein kinase | 0.0222 | 0.7603 | 0.7603 |
Trichomonas vaginalis | AGC family protein kinase | 0.0073 | 0.0202 | 0.0202 |
Toxoplasma gondii | AGC kinase | 0.0209 | 0.693 | 0.5 |
Trichomonas vaginalis | AGC family protein kinase | 0.0222 | 0.7603 | 0.7603 |
Echinococcus multilocularis | nervana 2 | 0.0136 | 0.3296 | 0.3158 |
Trichomonas vaginalis | AGC family protein kinase | 0.0222 | 0.7603 | 0.7603 |
Trichomonas vaginalis | AGC family protein kinase | 0.0087 | 0.0875 | 0.0875 |
Echinococcus multilocularis | rac serine:threonine kinase | 0.0153 | 0.4171 | 0.4051 |
Echinococcus granulosus | calcium:calmodulin dependent protein kinase | 0.014 | 0.3498 | 0.3364 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.0153 | 0.4171 | 0.4051 |
Echinococcus multilocularis | serine threonine protein kinase nrc serine threonine protein kinase gad | 0.014 | 0.3498 | 0.3364 |
Entamoeba histolytica | protein kinase, putative | 0.0222 | 0.7603 | 0.7554 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.0153 | 0.4171 | 0.4051 |
Echinococcus multilocularis | 3 phosphoinositide dependent protein kinase 1 | 0.0271 | 1 | 1 |
Trypanosoma cruzi | Protein kinase B | 0.0153 | 0.4171 | 1 |
Echinococcus multilocularis | Glutaredoxin protein 5 | 0.0136 | 0.3296 | 0.3158 |
Plasmodium vivax | rac-beta serine/threonine protein kinase, putative | 0.014 | 0.3498 | 0.5 |
Plasmodium falciparum | RAC-beta serine/threonine protein kinase | 0.014 | 0.3498 | 0.5 |
Schistosoma mansoni | serine/threonine protein kinase | 0.0271 | 1 | 1 |
Echinococcus multilocularis | sodium:potassium dependent atpase beta subunit | 0.0136 | 0.3296 | 0.3158 |
Schistosoma mansoni | serine/threonine-protein kinase | 0.0153 | 0.4171 | 0.4051 |
Trichomonas vaginalis | AGC family protein kinase | 0.0222 | 0.7603 | 0.7603 |
Brugia malayi | Protein kinase domain containing protein | 0.0222 | 0.7603 | 0.7554 |
Echinococcus granulosus | serine/threonine protein kinase | 0.0153 | 0.4171 | 0.4051 |
Trypanosoma cruzi | rac serine-threonine kinase, putative | 0.0153 | 0.4171 | 1 |
Schistosoma mansoni | serine/threonine-protein kinase | 0.0153 | 0.4171 | 0.4051 |
Loa Loa (eye worm) | AGC/AKT protein kinase | 0.0222 | 0.7603 | 0.7554 |
Brugia malayi | Protein kinase domain containing protein | 0.0271 | 1 | 1 |
Brugia malayi | p70 ribosomal S6 kinase beta | 0.0209 | 0.693 | 0.6866 |
Trichomonas vaginalis | AGC family protein kinase | 0.0271 | 1 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.0222 | 0.7603 | 0.7603 |
Echinococcus granulosus | 3-phosphoinositide-dependent protein kinase 1 | 0.0271 | 1 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.0271 | 1 | 1 |
Entamoeba histolytica | protein kinase, putative | 0.0271 | 1 | 1 |
Loa Loa (eye worm) | AGC/PDK1 protein kinase | 0.0271 | 1 | 1 |
Echinococcus granulosus | nervana 2 | 0.0136 | 0.3296 | 0.3158 |
Trichomonas vaginalis | AGC family protein kinase | 0.0271 | 1 | 1 |
Echinococcus granulosus | nervana 2 | 0.0136 | 0.3296 | 0.3158 |
Echinococcus granulosus | serine threonine protein kinase nrc | 0.014 | 0.3498 | 0.3364 |
Loa Loa (eye worm) | AGC/RSK/P70 protein kinase | 0.0209 | 0.693 | 0.6866 |
Entamoeba histolytica | protein kinase 2, putative | 0.014 | 0.3498 | 0.3364 |
Trichomonas vaginalis | AGC family protein kinase | 0.0073 | 0.0202 | 0.0202 |
Entamoeba histolytica | protein kinase, putative | 0.0222 | 0.7603 | 0.7554 |
Giardia lamblia | Kinase, AGC PKA | 0.014 | 0.3498 | 0.5 |
Trypanosoma brucei | rac serine-threonine kinase, putative | 0.0222 | 0.7603 | 0.5 |
Loa Loa (eye worm) | AGC/PDK1 protein kinase | 0.0271 | 1 | 1 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
Inhibition (functional) | = 34 % | Irreversible inhibition against Norepinephrine (NE)-induced response in rat vas deferens with benextramine (BHC) as standard at a concentration of 2 x 10e-5 M | ChEMBL. | 2885418 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.