Species | Target name | Source | Bibliographic reference |
---|---|---|---|
Homo sapiens | lactate dehydrogenase C | Starlite/ChEMBL | References |
Species | Potential target | Known druggable target | Length | Alignment span | Identity |
---|---|---|---|---|---|
Plasmodium falciparum | lactate dehydrogenase, putative | lactate dehydrogenase C | 332 aa | 307 aa | 29.6 % |
Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Giardia lamblia | Malate dehydrogenase | 0.0022 | 0 | 0.5 |
Mycobacterium ulcerans | malate dehydrogenase | 0.0022 | 0 | 0.5 |
Trypanosoma brucei | mitochondrial malate dehydrogenase | 0.0022 | 0 | 0.5 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0022 | 0 | 0.5 |
Trichomonas vaginalis | malate and lactate dehydrogenase, putative | 0.0022 | 0 | 0.5 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0022 | 0 | 0.5 |
Echinococcus multilocularis | lactate dehydrogenase a | 0.0056 | 1 | 1 |
Toxoplasma gondii | malate dehydrogenase MDH | 0.0056 | 1 | 0.5 |
Echinococcus granulosus | L lactate dehydrogenase | 0.0034 | 0.3641 | 0.3641 |
Mycobacterium tuberculosis | Probable malate dehydrogenase Mdh | 0.0022 | 0 | 0.5 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0022 | 0 | 0.5 |
Leishmania major | malate dehydrogenase, putative | 0.0056 | 1 | 1 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0022 | 0 | 0.5 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0022 | 0 | 0.5 |
Trypanosoma brucei | malate dehydrogenase-related | 0.0022 | 0 | 0.5 |
Trichomonas vaginalis | malate and lactate dehydrogenase, putative | 0.0022 | 0 | 0.5 |
Trypanosoma cruzi | glycosomal malate dehydrogenase, putative | 0.0022 | 0 | 0.5 |
Trypanosoma cruzi | cytosolic malate dehydrogenase, putative | 0.0022 | 0 | 0.5 |
Trypanosoma cruzi | glycosomal malate dehydrogenase, putative | 0.0022 | 0 | 0.5 |
Toxoplasma gondii | lactate dehydrogenase LDH2 | 0.0056 | 1 | 0.5 |
Schistosoma mansoni | malate dehydrogenase | 0.0056 | 1 | 1 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0022 | 0 | 0.5 |
Plasmodium vivax | malate dehydrogenase, putative | 0.0056 | 1 | 1 |
Echinococcus multilocularis | lactate dehydrogenase a | 0.0056 | 1 | 1 |
Plasmodium falciparum | malate dehydrogenase | 0.0056 | 1 | 1 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0022 | 0 | 0.5 |
Echinococcus multilocularis | lactate dehydrogenase protein | 0.0056 | 1 | 1 |
Echinococcus granulosus | L lactate dehydrogenase B chain | 0.0056 | 1 | 1 |
Trypanosoma cruzi | malate dehydrogenase, putative | 0.0022 | 0 | 0.5 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0022 | 0 | 0.5 |
Toxoplasma gondii | lactate dehydrogenase LDH1 | 0.0056 | 1 | 0.5 |
Entamoeba histolytica | malate dehydrogenase, putative | 0.0056 | 1 | 1 |
Wolbachia endosymbiont of Brugia malayi | malate dehydrogenase | 0.0056 | 1 | 0.5 |
Chlamydia trachomatis | malate dehydrogenase | 0.0022 | 0 | 0.5 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0022 | 0 | 0.5 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0022 | 0 | 0.5 |
Echinococcus granulosus | lactate dehydrogenase protein | 0.0056 | 1 | 1 |
Trypanosoma cruzi | cytosolic malate dehydrogenase, putative | 0.0022 | 0 | 0.5 |
Schistosoma mansoni | L-lactate dehydrogenase | 0.0056 | 1 | 1 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0022 | 0 | 0.5 |
Trypanosoma cruzi | mitochondrial malate dehydrogenase, putative | 0.0022 | 0 | 0.5 |
Plasmodium vivax | lactate dehydrogenase | 0.0056 | 1 | 1 |
Trypanosoma brucei | cytosolic malate dehydrogenase | 0.0022 | 0 | 0.5 |
Echinococcus multilocularis | lactate dehydrogenase a | 0.0056 | 1 | 1 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0022 | 0 | 0.5 |
Echinococcus granulosus | lactate dehydrogenase a | 0.0056 | 1 | 1 |
Trypanosoma brucei | glycosomal malate dehydrogenase | 0.0022 | 0 | 0.5 |
Echinococcus multilocularis | L lactate dehydrogenase | 0.0034 | 0.3641 | 0.3641 |
Loa Loa (eye worm) | hypothetical protein | 0.0056 | 1 | 1 |
Trichomonas vaginalis | malate and lactate dehydrogenase, putative | 0.0022 | 0 | 0.5 |
Trypanosoma cruzi | malate dehydrogenase, putative | 0.0022 | 0 | 0.5 |
Trichomonas vaginalis | malate and lactate dehydrogenase, putative | 0.0022 | 0 | 0.5 |
Mycobacterium leprae | PROBABLE MALATE DEHYDROGENASE MDH | 0.0022 | 0 | 0.5 |
Echinococcus multilocularis | L lactate dehydrogenase B chain | 0.0056 | 1 | 1 |
Plasmodium falciparum | L-lactate dehydrogenase | 0.0056 | 1 | 1 |
Echinococcus granulosus | lactate dehydrogenase a | 0.0056 | 1 | 1 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
IC50 (binding) | = 5 nM | Inhibition of LDHA (unknown origin) | ChEMBL. | 25288186 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.