Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Echinococcus granulosus | serine/threonine protein kinase | 0.0033 | 0.3903 | 0.3903 |
Trichomonas vaginalis | AGC family protein kinase | 0.0057 | 1 | 1 |
Echinococcus multilocularis | serine threonine protein kinase nrc serine threonine protein kinase gad | 0.0033 | 0.3903 | 0.3903 |
Echinococcus granulosus | nervana 2 | 0.0032 | 0.3679 | 0.3679 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.0033 | 0.3903 | 0.3903 |
Trypanosoma cruzi | rac serine-threonine kinase, putative | 0.0033 | 0.3903 | 0.5 |
Echinococcus multilocularis | 3 phosphoinositide dependent protein kinase 1 | 0.0057 | 1 | 1 |
Echinococcus multilocularis | rac serine:threonine kinase | 0.0033 | 0.3903 | 0.3903 |
Schistosoma mansoni | serine/threonine-protein kinase | 0.0033 | 0.3903 | 0.3903 |
Plasmodium vivax | rac-beta serine/threonine protein kinase, putative | 0.0033 | 0.3903 | 0.5 |
Echinococcus granulosus | calcium:calmodulin dependent protein kinase | 0.0033 | 0.3903 | 0.3903 |
Trichomonas vaginalis | AGC family protein kinase | 0.0049 | 0.7966 | 0.7966 |
Trypanosoma brucei | rac serine-threonine kinase, putative | 0.0049 | 0.7966 | 0.5 |
Echinococcus granulosus | nervana 2 | 0.0032 | 0.3679 | 0.3679 |
Loa Loa (eye worm) | AGC/RSK/P70 protein kinase | 0.0049 | 0.7966 | 0.7966 |
Entamoeba histolytica | protein kinase, putative | 0.0049 | 0.7966 | 0.7966 |
Echinococcus granulosus | sodium:potassium dependent atpase beta subunit | 0.0032 | 0.3679 | 0.3679 |
Trichomonas vaginalis | AGC family protein kinase | 0.0049 | 0.7966 | 0.7966 |
Entamoeba histolytica | protein kinase 2, putative | 0.0033 | 0.3903 | 0.3903 |
Echinococcus multilocularis | nervana 2 | 0.0032 | 0.3679 | 0.3679 |
Trichomonas vaginalis | AGC family protein kinase | 0.0049 | 0.7966 | 0.7966 |
Brugia malayi | Protein kinase domain containing protein | 0.0049 | 0.7966 | 0.7966 |
Echinococcus multilocularis | Glutaredoxin protein 5 | 0.0032 | 0.3679 | 0.3679 |
Trichomonas vaginalis | AGC family protein kinase | 0.0049 | 0.7966 | 0.7966 |
Brugia malayi | p70 ribosomal S6 kinase beta | 0.0049 | 0.7966 | 0.7966 |
Loa Loa (eye worm) | AGC/PDK1 protein kinase | 0.0057 | 1 | 1 |
Echinococcus multilocularis | sodium:potassium dependent atpase beta subunit | 0.0032 | 0.3679 | 0.3679 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.0033 | 0.3903 | 0.3903 |
Trichomonas vaginalis | AGC family protein kinase | 0.0049 | 0.7966 | 0.7966 |
Trypanosoma cruzi | Protein kinase B | 0.0033 | 0.3903 | 0.5 |
Entamoeba histolytica | protein kinase, putative | 0.0049 | 0.7966 | 0.7966 |
Echinococcus granulosus | serine threonine protein kinase nrc | 0.0033 | 0.3903 | 0.3903 |
Entamoeba histolytica | protein kinase, putative | 0.0057 | 1 | 1 |
Echinococcus multilocularis | nervana 2 | 0.0032 | 0.3679 | 0.3679 |
Trichomonas vaginalis | AGC family protein kinase | 0.0057 | 1 | 1 |
Brugia malayi | Protein kinase domain containing protein | 0.0057 | 1 | 1 |
Echinococcus granulosus | 3-phosphoinositide-dependent protein kinase 1 | 0.0057 | 1 | 1 |
Loa Loa (eye worm) | AGC/AKT protein kinase | 0.0049 | 0.7966 | 0.7966 |
Loa Loa (eye worm) | AGC/PDK1 protein kinase | 0.0057 | 1 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.0049 | 0.7966 | 0.7966 |
Schistosoma mansoni | serine/threonine protein kinase | 0.0057 | 1 | 1 |
Trypanosoma cruzi | rac serine-threonine kinase, putative | 0.0033 | 0.3903 | 0.5 |
Trichomonas vaginalis | AGC family protein kinase | 0.0057 | 1 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.0049 | 0.7966 | 0.7966 |
Toxoplasma gondii | AGC kinase | 0.0049 | 0.7966 | 0.5 |
Schistosoma mansoni | serine/threonine-protein kinase | 0.0033 | 0.3903 | 0.3903 |
Plasmodium falciparum | RAC-beta serine/threonine protein kinase | 0.0033 | 0.3903 | 0.5 |
Entamoeba histolytica | protein kinase, putative | 0.0049 | 0.7966 | 0.7966 |
Echinococcus granulosus | Glutaredoxin protein 5 | 0.0032 | 0.3679 | 0.3679 |
Giardia lamblia | Kinase, AGC PKA | 0.0033 | 0.3903 | 0.5 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
Activity (functional) | = 31.25 % | Cytotoxicity against human SR cells assessed as cell growth at 10 uM | ChEMBL. | 25440729 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.