Species | Target name | Source | Bibliographic reference |
---|---|---|---|
Homo sapiens | lactate dehydrogenase C | Starlite/ChEMBL | References |
Species | Potential target | Known druggable target | Length | Alignment span | Identity |
---|---|---|---|---|---|
Plasmodium falciparum | lactate dehydrogenase, putative | lactate dehydrogenase C | 332 aa | 307 aa | 29.6 % |
Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Mycobacterium leprae | PROBABLE MALATE DEHYDROGENASE MDH | 0.0022 | 0 | 0.5 |
Giardia lamblia | Malate dehydrogenase | 0.0022 | 0 | 0.5 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0022 | 0 | 0.5 |
Trypanosoma brucei | glycosomal malate dehydrogenase | 0.0022 | 0 | 0.5 |
Loa Loa (eye worm) | hypothetical protein | 0.0056 | 1 | 1 |
Trichomonas vaginalis | malate and lactate dehydrogenase, putative | 0.0022 | 0 | 0.5 |
Echinococcus multilocularis | L lactate dehydrogenase B chain | 0.0056 | 1 | 1 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0022 | 0 | 0.5 |
Chlamydia trachomatis | malate dehydrogenase | 0.0022 | 0 | 0.5 |
Trichomonas vaginalis | malate and lactate dehydrogenase, putative | 0.0022 | 0 | 0.5 |
Toxoplasma gondii | malate dehydrogenase MDH | 0.0056 | 1 | 0.5 |
Echinococcus granulosus | lactate dehydrogenase a | 0.0056 | 1 | 1 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0022 | 0 | 0.5 |
Toxoplasma gondii | lactate dehydrogenase LDH1 | 0.0056 | 1 | 0.5 |
Mycobacterium tuberculosis | Probable malate dehydrogenase Mdh | 0.0022 | 0 | 0.5 |
Trypanosoma cruzi | cytosolic malate dehydrogenase, putative | 0.0022 | 0 | 0.5 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0022 | 0 | 0.5 |
Echinococcus multilocularis | lactate dehydrogenase protein | 0.0056 | 1 | 1 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0022 | 0 | 0.5 |
Trichomonas vaginalis | malate and lactate dehydrogenase, putative | 0.0022 | 0 | 0.5 |
Wolbachia endosymbiont of Brugia malayi | malate dehydrogenase | 0.0056 | 1 | 0.5 |
Trypanosoma cruzi | cytosolic malate dehydrogenase, putative | 0.0022 | 0 | 0.5 |
Echinococcus granulosus | L lactate dehydrogenase | 0.0034 | 0.3641 | 0.3641 |
Mycobacterium ulcerans | malate dehydrogenase | 0.0022 | 0 | 0.5 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0022 | 0 | 0.5 |
Plasmodium vivax | malate dehydrogenase, putative | 0.0056 | 1 | 1 |
Trichomonas vaginalis | malate and lactate dehydrogenase, putative | 0.0022 | 0 | 0.5 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0022 | 0 | 0.5 |
Trypanosoma cruzi | glycosomal malate dehydrogenase, putative | 0.0022 | 0 | 0.5 |
Plasmodium falciparum | malate dehydrogenase | 0.0056 | 1 | 1 |
Plasmodium falciparum | L-lactate dehydrogenase | 0.0056 | 1 | 1 |
Trypanosoma cruzi | mitochondrial malate dehydrogenase, putative | 0.0022 | 0 | 0.5 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0022 | 0 | 0.5 |
Echinococcus multilocularis | lactate dehydrogenase a | 0.0056 | 1 | 1 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0022 | 0 | 0.5 |
Trypanosoma brucei | malate dehydrogenase-related | 0.0022 | 0 | 0.5 |
Entamoeba histolytica | malate dehydrogenase, putative | 0.0056 | 1 | 1 |
Echinococcus multilocularis | L lactate dehydrogenase | 0.0034 | 0.3641 | 0.3641 |
Trypanosoma brucei | mitochondrial malate dehydrogenase | 0.0022 | 0 | 0.5 |
Leishmania major | malate dehydrogenase, putative | 0.0056 | 1 | 1 |
Trypanosoma cruzi | glycosomal malate dehydrogenase, putative | 0.0022 | 0 | 0.5 |
Trypanosoma brucei | cytosolic malate dehydrogenase | 0.0022 | 0 | 0.5 |
Schistosoma mansoni | malate dehydrogenase | 0.0056 | 1 | 1 |
Trypanosoma cruzi | malate dehydrogenase, putative | 0.0022 | 0 | 0.5 |
Toxoplasma gondii | lactate dehydrogenase LDH2 | 0.0056 | 1 | 0.5 |
Trypanosoma cruzi | malate dehydrogenase, putative | 0.0022 | 0 | 0.5 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0022 | 0 | 0.5 |
Echinococcus multilocularis | lactate dehydrogenase a | 0.0056 | 1 | 1 |
Echinococcus granulosus | L lactate dehydrogenase B chain | 0.0056 | 1 | 1 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0022 | 0 | 0.5 |
Echinococcus multilocularis | lactate dehydrogenase a | 0.0056 | 1 | 1 |
Plasmodium vivax | lactate dehydrogenase | 0.0056 | 1 | 1 |
Echinococcus granulosus | lactate dehydrogenase a | 0.0056 | 1 | 1 |
Trichomonas vaginalis | malate dehydrogenase, putative | 0.0022 | 0 | 0.5 |
Echinococcus granulosus | lactate dehydrogenase protein | 0.0056 | 1 | 1 |
Schistosoma mansoni | L-lactate dehydrogenase | 0.0056 | 1 | 1 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
IC50 (binding) | = 5 uM | Inhibition of human LDH-A by biochemical assay | ChEMBL. | 25467161 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.