Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Trypanosoma cruzi | rac serine-threonine kinase, putative | 0.0596 | 0.5205 | 1 |
Loa Loa (eye worm) | AGC/AKT protein kinase | 0.0881 | 1 | 1 |
Echinococcus granulosus | 3-phosphoinositide-dependent protein kinase 1 | 0.0577 | 0.4884 | 0.936 |
Brugia malayi | p70 ribosomal S6 kinase beta | 0.0857 | 0.9597 | 0.9589 |
Plasmodium vivax | rac-beta serine/threonine protein kinase, putative | 0.0572 | 0.4802 | 0.5 |
Trichomonas vaginalis | AGC family protein kinase | 0.0297 | 0.0196 | 0.0196 |
Echinococcus multilocularis | serine threonine protein kinase nrc serine threonine protein kinase gad | 0.0572 | 0.4802 | 0.9195 |
Entamoeba histolytica | protein kinase, putative | 0.0857 | 0.9597 | 0.9589 |
Echinococcus granulosus | serine/threonine protein kinase | 0.0596 | 0.5205 | 1 |
Entamoeba histolytica | protein kinase, putative | 0.0881 | 1 | 1 |
Entamoeba histolytica | protein kinase, putative | 0.0577 | 0.4884 | 0.4782 |
Trichomonas vaginalis | AGC family protein kinase | 0.0297 | 0.0196 | 0.0196 |
Trichomonas vaginalis | AGC family protein kinase | 0.0881 | 1 | 1 |
Echinococcus granulosus | serine threonine protein kinase nrc | 0.0572 | 0.4802 | 0.9195 |
Entamoeba histolytica | protein kinase, putative | 0.0881 | 1 | 1 |
Echinococcus multilocularis | Glutaredoxin protein 5 | 0.056 | 0.4605 | 0.8803 |
Loa Loa (eye worm) | AGC/PDK1 protein kinase | 0.0577 | 0.4884 | 0.4782 |
Trichomonas vaginalis | AGC family protein kinase | 0.0881 | 1 | 1 |
Echinococcus multilocularis | sodium:potassium dependent atpase beta subunit | 0.056 | 0.4605 | 0.8803 |
Trichomonas vaginalis | AGC family protein kinase | 0.0881 | 1 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.0321 | 0.06 | 0.06 |
Loa Loa (eye worm) | AGC/PDK1 protein kinase | 0.0577 | 0.4884 | 0.4782 |
Trichomonas vaginalis | AGC family protein kinase | 0.0577 | 0.4884 | 0.4884 |
Schistosoma mansoni | serine/threonine-protein kinase | 0.0596 | 0.5205 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.0881 | 1 | 1 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.0596 | 0.5205 | 0.5109 |
Echinococcus multilocularis | nervana 2 | 0.056 | 0.4605 | 0.8803 |
Trichomonas vaginalis | AGC family protein kinase | 0.0881 | 1 | 1 |
Trypanosoma brucei | rac serine-threonine kinase, putative | 0.0881 | 1 | 0.5 |
Entamoeba histolytica | protein kinase 2, putative | 0.0572 | 0.4802 | 0.4697 |
Toxoplasma gondii | AGC kinase | 0.0857 | 0.9597 | 0.5 |
Trypanosoma cruzi | Protein kinase B | 0.0596 | 0.5205 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.0881 | 1 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.0297 | 0.0196 | 0.0196 |
Echinococcus multilocularis | rac serine:threonine kinase | 0.0596 | 0.5205 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.0881 | 1 | 1 |
Echinococcus granulosus | nervana 2 | 0.056 | 0.4605 | 0.8803 |
Giardia lamblia | Kinase, AGC PKA | 0.0572 | 0.4802 | 0.5 |
Echinococcus multilocularis | nervana 2 | 0.056 | 0.4605 | 0.8803 |
Echinococcus granulosus | sodium:potassium dependent atpase beta subunit | 0.056 | 0.4605 | 0.8803 |
Schistosoma mansoni | serine/threonine protein kinase | 0.0577 | 0.4884 | 0.936 |
Trichomonas vaginalis | AGC family protein kinase | 0.0577 | 0.4884 | 0.4884 |
Brugia malayi | phosphoinositide-dependent protein kinase I | 0.0577 | 0.4884 | 0.4782 |
Schistosoma mansoni | serine/threonine-protein kinase | 0.0596 | 0.5205 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.0577 | 0.4884 | 0.4884 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.0596 | 0.5205 | 0.5109 |
Loa Loa (eye worm) | AGC/RSK/P70 protein kinase | 0.0857 | 0.9597 | 0.9589 |
Brugia malayi | Protein kinase domain containing protein | 0.0577 | 0.4884 | 0.4782 |
Echinococcus granulosus | Glutaredoxin protein 5 | 0.056 | 0.4605 | 0.8803 |
Echinococcus multilocularis | 3 phosphoinositide dependent protein kinase 1 | 0.0577 | 0.4884 | 0.936 |
Plasmodium falciparum | RAC-beta serine/threonine protein kinase | 0.0572 | 0.4802 | 0.5 |
Echinococcus granulosus | calcium:calmodulin dependent protein kinase | 0.0572 | 0.4802 | 0.9195 |
Echinococcus granulosus | nervana 2 | 0.056 | 0.4605 | 0.8803 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
MIC (functional) | = 0.71 ug ml-1 | Antimycobacterial activity against Mycobacterium tuberculosis H37Rv by agar dilution method | ChEMBL. | 18714980 |
MIC (functional) | = 0.71 ug ml-1 | Antimycobacterial activity against multidrug-resistant Mycobacterium tuberculosis by agar dilution method | ChEMBL. | 18714980 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.