Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Toxoplasma gondii | AGC kinase | 0.084 | 0.9598 | 0.5 |
Plasmodium falciparum | RAC-beta serine/threonine protein kinase | 0.0561 | 0.4814 | 0.5 |
Giardia lamblia | Kinase, AGC PKA | 0.0561 | 0.4814 | 0.5 |
Trichomonas vaginalis | AGC family protein kinase | 0.0292 | 0.022 | 0.022 |
Echinococcus granulosus | serine/threonine protein kinase | 0.0584 | 0.5216 | 0.6948 |
Entamoeba histolytica | protein kinase, putative | 0.084 | 0.9598 | 0.9589 |
Entamoeba histolytica | protein kinase, putative | 0.0712 | 0.7411 | 0.7353 |
Trichomonas vaginalis | AGC family protein kinase | 0.0863 | 1 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.0863 | 1 | 1 |
Loa Loa (eye worm) | AGC/PDK1 protein kinase | 0.0712 | 0.7411 | 0.7353 |
Schistosoma mansoni | serine/threonine-protein kinase | 0.0584 | 0.5216 | 0.6948 |
Trypanosoma cruzi | rac serine-threonine kinase, putative | 0.0584 | 0.5216 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.0863 | 1 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.0316 | 0.0622 | 0.0622 |
Echinococcus multilocularis | sodium:potassium dependent atpase beta subunit | 0.0548 | 0.4594 | 0.6083 |
Trichomonas vaginalis | AGC family protein kinase | 0.0863 | 1 | 1 |
Schistosoma mansoni | serine/threonine-protein kinase | 0.0584 | 0.5216 | 0.6948 |
Trichomonas vaginalis | AGC family protein kinase | 0.0863 | 1 | 1 |
Echinococcus multilocularis | nervana 2 | 0.0548 | 0.4594 | 0.6083 |
Entamoeba histolytica | protein kinase 2, putative | 0.0561 | 0.4814 | 0.4697 |
Trichomonas vaginalis | AGC family protein kinase | 0.0863 | 1 | 1 |
Entamoeba histolytica | protein kinase, putative | 0.0863 | 1 | 1 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.0584 | 0.5216 | 0.5109 |
Trichomonas vaginalis | AGC family protein kinase | 0.0292 | 0.022 | 0.022 |
Brugia malayi | phosphoinositide-dependent protein kinase I | 0.0712 | 0.7411 | 0.7353 |
Echinococcus granulosus | nervana 2 | 0.0548 | 0.4594 | 0.6083 |
Echinococcus granulosus | 3-phosphoinositide-dependent protein kinase 1 | 0.0712 | 0.7411 | 1 |
Schistosoma mansoni | serine/threonine protein kinase | 0.0712 | 0.7411 | 1 |
Echinococcus multilocularis | Glutaredoxin protein 5 | 0.0548 | 0.4594 | 0.6083 |
Echinococcus granulosus | nervana 2 | 0.0548 | 0.4594 | 0.6083 |
Echinococcus granulosus | calcium:calmodulin dependent protein kinase | 0.0561 | 0.4814 | 0.6389 |
Echinococcus multilocularis | 3 phosphoinositide dependent protein kinase 1 | 0.0712 | 0.7411 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.0863 | 1 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.0292 | 0.022 | 0.022 |
Entamoeba histolytica | protein kinase, putative | 0.0863 | 1 | 1 |
Brugia malayi | p70 ribosomal S6 kinase beta | 0.084 | 0.9598 | 0.9589 |
Loa Loa (eye worm) | AGC/PDK1 protein kinase | 0.0712 | 0.7411 | 0.7353 |
Echinococcus granulosus | serine threonine protein kinase nrc | 0.0561 | 0.4814 | 0.6389 |
Trypanosoma brucei | rac serine-threonine kinase, putative | 0.0863 | 1 | 0.5 |
Echinococcus multilocularis | nervana 2 | 0.0548 | 0.4594 | 0.6083 |
Loa Loa (eye worm) | AGC/AKT protein kinase | 0.0863 | 1 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.0712 | 0.7411 | 0.7411 |
Echinococcus granulosus | Glutaredoxin protein 5 | 0.0548 | 0.4594 | 0.6083 |
Echinococcus multilocularis | serine threonine protein kinase nrc serine threonine protein kinase gad | 0.0561 | 0.4814 | 0.6389 |
Plasmodium vivax | rac-beta serine/threonine protein kinase, putative | 0.0561 | 0.4814 | 0.5 |
Trypanosoma cruzi | Protein kinase B | 0.0584 | 0.5216 | 1 |
Echinococcus granulosus | sodium:potassium dependent atpase beta subunit | 0.0548 | 0.4594 | 0.6083 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.0584 | 0.5216 | 0.5109 |
Loa Loa (eye worm) | AGC/RSK/P70 protein kinase | 0.084 | 0.9598 | 0.9589 |
Brugia malayi | Protein kinase domain containing protein | 0.0712 | 0.7411 | 0.7353 |
Trichomonas vaginalis | AGC family protein kinase | 0.0712 | 0.7411 | 0.7411 |
Echinococcus multilocularis | rac serine:threonine kinase | 0.0584 | 0.5216 | 0.6948 |
Trichomonas vaginalis | AGC family protein kinase | 0.0712 | 0.7411 | 0.7411 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
Ki (binding) | = 102 uM | Inhibition of human placental Monoamine oxidase A (competitive inhibition was observed) | ChEMBL. | 2296014 |
Ki (binding) | = 1600 uM | Compounds were tested for inhibition against human liver Monoamine oxidase B (mixed inhibition was observed) | ChEMBL. | 2296014 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.