Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Loa Loa (eye worm) | CAMK/PKD protein kinase | 0.0149 | 0.0048 | 0.0048 |
Loa Loa (eye worm) | AGC/NDR protein kinase | 0.0204 | 0.0285 | 0.0285 |
Loa Loa (eye worm) | raf kinase | 0.0144 | 0.0029 | 0.0029 |
Brugia malayi | Hr1 repeat family protein | 0.0204 | 0.0285 | 0.2872 |
Brugia malayi | Protein kinase domain containing protein | 0.0149 | 0.0048 | 0.0211 |
Trichomonas vaginalis | AGC family protein kinase | 0.0204 | 0.0285 | 1 |
Onchocerca volvulus | 0.0148 | 0.0047 | 0.0019 | |
Schistosoma mansoni | unc-13 (munc13) | 0.0148 | 0.0047 | 0.0122 |
Loa Loa (eye worm) | hypothetical protein | 0.0144 | 0.0029 | 0.0029 |
Brugia malayi | protein kinase C II. | 0.0352 | 0.0919 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0144 | 0.0029 | 0.0029 |
Entamoeba histolytica | protein kinase, putative | 0.0204 | 0.0285 | 1 |
Echinococcus multilocularis | ribosomal protein s6 kinase beta 1 | 0.0204 | 0.0285 | 0.1774 |
Schistosoma mansoni | protein kinase C mu | 0.0149 | 0.0048 | 0.0131 |
Loa Loa (eye worm) | AGC/RSK/MSK protein kinase | 0.0204 | 0.0285 | 0.0285 |
Schistosoma mansoni | serine/threonine protein kinase | 0.0149 | 0.0048 | 0.0131 |
Loa Loa (eye worm) | hypothetical protein | 0.0144 | 0.0029 | 0.0029 |
Echinococcus multilocularis | protein kinase c epsilon type | 0.0352 | 0.0919 | 0.6176 |
Trichomonas vaginalis | AGC family protein kinase | 0.0204 | 0.0285 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0144 | 0.0029 | 0.0029 |
Loa Loa (eye worm) | AGC/PKC/ETA protein kinase | 0.0352 | 0.0919 | 0.0919 |
Trypanosoma brucei | rac serine-threonine kinase, putative | 0.0204 | 0.0285 | 0.5 |
Schistosoma mansoni | serine/threonine kinase | 0.0204 | 0.0285 | 0.1774 |
Brugia malayi | Protein kinase domain containing protein | 0.0204 | 0.0285 | 0.2872 |
Brugia malayi | Protein kinase domain containing protein | 0.0204 | 0.0285 | 0.2872 |
Loa Loa (eye worm) | hypothetical protein | 0.0144 | 0.0029 | 0.0029 |
Echinococcus multilocularis | serine:threonine protein kinase 38 | 0.0204 | 0.0285 | 0.1774 |
Schistosoma mansoni | serine/threonine protein kinase | 0.0481 | 0.1469 | 1 |
Schistosoma mansoni | unc-13 (munc13) | 0.0148 | 0.0047 | 0.0122 |
Entamoeba histolytica | protein kinase, putative | 0.0204 | 0.0285 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.2417 | 0.9745 | 0.9745 |
Loa Loa (eye worm) | AGC/DMPK/GEK protein kinase | 0.0204 | 0.0285 | 0.0285 |
Loa Loa (eye worm) | AGC/PKN protein kinase | 0.0204 | 0.0285 | 0.0285 |
Echinococcus granulosus | Serine/threonine-protein kinase Genghis Khan | 0.0149 | 0.0048 | 0.0131 |
Echinococcus granulosus | unc 13 munc13 | 0.0148 | 0.0047 | 0.0122 |
Schistosoma mansoni | serine/threonine protein kinase | 0.0204 | 0.0285 | 0.1774 |
Trichomonas vaginalis | AGC family protein kinase | 0.0204 | 0.0285 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0273 | 0.058 | 0.058 |
Loa Loa (eye worm) | AGC/AKT protein kinase | 0.0204 | 0.0285 | 0.0285 |
Echinococcus multilocularis | C2 calcium dependent membrane targeting | 0.0148 | 0.0047 | 0.0122 |
Trichomonas vaginalis | AGC family protein kinase | 0.0204 | 0.0285 | 1 |
Echinococcus granulosus | serine:threonine protein kinase N2 | 0.0204 | 0.0285 | 0.1774 |
Echinococcus granulosus | ribosomal protein S6 kinase alpha 3 | 0.0204 | 0.0285 | 0.1774 |
Loa Loa (eye worm) | AGC/PKC/IOTA protein kinase | 0.0149 | 0.0048 | 0.0048 |
Trichomonas vaginalis | AGC family protein kinase | 0.0204 | 0.0285 | 1 |
Echinococcus granulosus | protein kinase c epsilon type | 0.0352 | 0.0919 | 0.6176 |
Trichomonas vaginalis | AGC family protein kinase | 0.0204 | 0.0285 | 1 |
Echinococcus multilocularis | serine threonine protein kinase | 0.0337 | 0.0853 | 0.5719 |
Schistosoma mansoni | serine/threonine protein kinase | 0.0352 | 0.0919 | 0.6176 |
Trichomonas vaginalis | AGC family protein kinase | 0.0204 | 0.0285 | 1 |
Echinococcus multilocularis | unc 13 (munc13) | 0.0148 | 0.0047 | 0.0122 |
Echinococcus granulosus | protein kinase C gamma type | 0.0337 | 0.0853 | 0.5719 |
Loa Loa (eye worm) | hypothetical protein | 0.0144 | 0.0029 | 0.0029 |
Echinococcus multilocularis | serine:threonine protein kinase MRCK beta | 0.0149 | 0.0048 | 0.0131 |
Loa Loa (eye worm) | hypothetical protein | 0.0144 | 0.0029 | 0.0029 |
Brugia malayi | Protein kinase c protein 2 | 0.0281 | 0.0616 | 0.66 |
Loa Loa (eye worm) | AGC/RSK/P70 protein kinase | 0.0204 | 0.0285 | 0.0285 |
Loa Loa (eye worm) | hypothetical protein | 0.0148 | 0.0047 | 0.0047 |
Schistosoma mansoni | serine/threonine protein kinase | 0.0204 | 0.0285 | 0.1774 |
Echinococcus multilocularis | serine:threonine protein kinase N2 | 0.0204 | 0.0285 | 0.1774 |
Schistosoma mansoni | protein kinase C | 0.0148 | 0.0047 | 0.0122 |
Brugia malayi | C1-like domain containing protein | 0.0149 | 0.0048 | 0.0211 |
Toxoplasma gondii | AGC kinase | 0.0204 | 0.0285 | 1 |
Echinococcus granulosus | Ribosomal protein S6 kinase beta 2 | 0.0204 | 0.0285 | 0.1774 |
Echinococcus granulosus | protein kinase c iota type | 0.0348 | 0.0901 | 0.6054 |
Brugia malayi | p70 ribosomal S6 kinase beta | 0.0204 | 0.0285 | 0.2872 |
Loa Loa (eye worm) | hypothetical protein | 0.0144 | 0.0029 | 0.0029 |
Loa Loa (eye worm) | variant SH3 domain-containing protein | 0.0144 | 0.0029 | 0.0029 |
Trichomonas vaginalis | AGC family protein kinase | 0.0204 | 0.0285 | 1 |
Echinococcus multilocularis | Protein kinase C, brain isozyme | 0.0481 | 0.1469 | 1 |
Loa Loa (eye worm) | RasGEF domain-containing protein | 0.0144 | 0.0029 | 0.0029 |
Brugia malayi | Protein kinase domain containing protein | 0.0204 | 0.0285 | 0.2872 |
Schistosoma mansoni | serine/threonine protein kinase | 0.0204 | 0.0285 | 0.1774 |
Schistosoma mansoni | atypical protein kinase C | 0.0348 | 0.0901 | 0.6054 |
Echinococcus granulosus | Protein kinase C brain isozyme | 0.0481 | 0.1469 | 1 |
Echinococcus multilocularis | protein kinase c iota type | 0.0348 | 0.0901 | 0.6054 |
Trichomonas vaginalis | AGC family protein kinase | 0.0204 | 0.0285 | 1 |
Schistosoma mansoni | serine/threonine protein kinase | 0.0204 | 0.0285 | 0.1774 |
Schistosoma mansoni | serine/threonine protein kinase | 0.0481 | 0.1469 | 1 |
Onchocerca volvulus | 0.2273 | 0.9128 | 1 | |
Entamoeba histolytica | protein kinase, putative | 0.0204 | 0.0285 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.2273 | 0.9128 | 0.9128 |
Brugia malayi | protein kinase C3,putative | 0.0149 | 0.0048 | 0.0211 |
Brugia malayi | Phorbol esters/diacylglycerol binding domain | 0.0149 | 0.0048 | 0.0211 |
Entamoeba histolytica | protein kinase, putative | 0.0204 | 0.0285 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.0204 | 0.0285 | 1 |
Echinococcus granulosus | C2 calcium dependent membrane targeting | 0.0148 | 0.0047 | 0.0122 |
Loa Loa (eye worm) | hypothetical protein | 0.2273 | 0.9128 | 0.9128 |
Loa Loa (eye worm) | Ras association domain family 1 isoform A | 0.0144 | 0.0029 | 0.0029 |
Trichomonas vaginalis | AGC family protein kinase | 0.0204 | 0.0285 | 1 |
Echinococcus multilocularis | ribosomal protein S6 kinase alpha 3 | 0.0204 | 0.0285 | 0.1774 |
Schistosoma mansoni | serine/threonine protein kinase | 0.0149 | 0.0048 | 0.0131 |
Echinococcus granulosus | ribosomal protein s6 kinase beta 1 | 0.0204 | 0.0285 | 0.1774 |
Loa Loa (eye worm) | hypothetical protein | 0.0144 | 0.0029 | 0.0029 |
Echinococcus multilocularis | Ribosomal protein S6 kinase beta 2 | 0.0204 | 0.0285 | 0.1774 |
Loa Loa (eye worm) | hypothetical protein | 0.2273 | 0.9128 | 0.9128 |
Echinococcus multilocularis | serine:threonine protein kinase N2 | 0.0204 | 0.0285 | 0.1774 |
Loa Loa (eye worm) | RhoGAP domain-containing protein | 0.0144 | 0.0029 | 0.0029 |
Loa Loa (eye worm) | AGC/RSK/RSK protein kinase | 0.0204 | 0.0285 | 0.0285 |
Echinococcus granulosus | NDR protein kinase | 0.0204 | 0.0285 | 0.1774 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
clogP | = -1.23 | Calculated partition coefficient (clogP) (Pomona) | ChEMBL. | 2549245 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.