Species | Target name | Source | Bibliographic reference |
---|---|---|---|
Homo sapiens | v-akt murine thymoma viral oncogene homolog 1 | Starlite/ChEMBL | References |
Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Plasmodium falciparum | RAC-beta serine/threonine protein kinase | 0.0025 | 0.0738 | 0.5 |
Giardia lamblia | Kinase, AGC PKA | 0.0025 | 0.0738 | 1 |
Entamoeba histolytica | protein kinase, putative | 0.0038 | 0.1507 | 0.909 |
Entamoeba histolytica | protein kinase, putative | 0.004 | 0.1658 | 1 |
Trichomonas vaginalis | ribokinase, putative | 0.002 | 0.0443 | 0.2673 |
Echinococcus granulosus | sodium:potassium dependent atpase beta subunit | 0.0025 | 0.0721 | 0.0721 |
Echinococcus multilocularis | serine threonine protein kinase nrc serine threonine protein kinase gad | 0.0025 | 0.0738 | 0.0738 |
Mycobacterium ulcerans | fructokinase, PfkB | 0.002 | 0.0443 | 0.5 |
Entamoeba histolytica | ribokinase, putative | 0.002 | 0.0443 | 0.2673 |
Loa Loa (eye worm) | hypothetical protein | 0.002 | 0.0443 | 0.0443 |
Brugia malayi | Ribokinase | 0.002 | 0.0443 | 0.0443 |
Loa Loa (eye worm) | AGC/AKT protein kinase | 0.004 | 0.1658 | 0.1658 |
Schistosoma mansoni | serine/threonine-protein kinase | 0.0028 | 0.0889 | 0.0889 |
Trypanosoma cruzi | rac serine-threonine kinase, putative | 0.0028 | 0.0889 | 0.0467 |
Echinococcus multilocularis | pseudouridine metabolizing bifunctional protein | 0.002 | 0.0443 | 0.0443 |
Trichomonas vaginalis | ribokinase, putative | 0.002 | 0.0443 | 0.2673 |
Onchocerca volvulus | 0.0157 | 0.8771 | 1 | |
Echinococcus granulosus | nervana 2 | 0.0025 | 0.0721 | 0.0721 |
Mycobacterium ulcerans | carbohydrate kinase CbhK | 0.002 | 0.0443 | 0.5 |
Echinococcus granulosus | Glutaredoxin protein 5 | 0.0025 | 0.0721 | 0.0721 |
Echinococcus granulosus | serine/threonine protein kinase | 0.0028 | 0.0889 | 0.0889 |
Echinococcus multilocularis | ribokinase | 0.002 | 0.0443 | 0.0443 |
Echinococcus multilocularis | sodium:potassium dependent atpase beta subunit | 0.0025 | 0.0721 | 0.0721 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.0028 | 0.0889 | 0.5363 |
Trichomonas vaginalis | AGC family protein kinase | 0.004 | 0.1658 | 1 |
Trypanosoma brucei | rac serine-threonine kinase, putative | 0.004 | 0.1658 | 0.1271 |
Trichomonas vaginalis | AGC family protein kinase | 0.0015 | 0.0151 | 0.091 |
Loa Loa (eye worm) | hypothetical protein | 0.002 | 0.0443 | 0.0443 |
Trichomonas vaginalis | ribokinase, putative | 0.002 | 0.0443 | 0.2673 |
Plasmodium vivax | rac-beta serine/threonine protein kinase, putative | 0.0025 | 0.0738 | 0.5 |
Entamoeba histolytica | Hypothetical protein T24C12.3, putative | 0.002 | 0.0443 | 0.2673 |
Brugia malayi | p70 ribosomal S6 kinase beta | 0.0038 | 0.1507 | 0.1507 |
Mycobacterium tuberculosis | Adenosine kinase | 0.002 | 0.0443 | 0.5 |
Trichomonas vaginalis | AGC family protein kinase | 0.004 | 0.1658 | 1 |
Echinococcus multilocularis | rac serine:threonine kinase | 0.0028 | 0.0889 | 0.0889 |
Entamoeba histolytica | tagatose-6-phosphate kinase, putative | 0.002 | 0.0443 | 0.2673 |
Echinococcus granulosus | calcium:calmodulin dependent protein kinase | 0.0025 | 0.0738 | 0.0738 |
Mycobacterium tuberculosis | 6-phosphofructokinase PfkB (phosphohexokinase) (phosphofructokinase) | 0.002 | 0.0443 | 0.5 |
Echinococcus granulosus | ribokinase | 0.002 | 0.0443 | 0.0443 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.0028 | 0.0889 | 0.5363 |
Entamoeba histolytica | protein kinase 2, putative | 0.0025 | 0.0738 | 0.4453 |
Mycobacterium leprae | Probable adenosine kinase adk | 0.002 | 0.0443 | 0.5 |
Entamoeba histolytica | protein kinase, putative | 0.004 | 0.1658 | 1 |
Echinococcus multilocularis | nervana 2 | 0.0025 | 0.0721 | 0.0721 |
Trypanosoma cruzi | Protein kinase B | 0.0028 | 0.0889 | 0.0467 |
Brugia malayi | hypothetical protein | 0.002 | 0.0443 | 0.0443 |
Trichomonas vaginalis | AGC family protein kinase | 0.004 | 0.1658 | 1 |
Echinococcus granulosus | nervana 2 | 0.0025 | 0.0721 | 0.0721 |
Trypanosoma cruzi | rac serine-threonine kinase, putative | 0.0025 | 0.0738 | 0.0309 |
Trichomonas vaginalis | conserved hypothetical protein | 0.002 | 0.0443 | 0.2673 |
Entamoeba histolytica | kinase, PfkB family | 0.002 | 0.0443 | 0.2673 |
Echinococcus multilocularis | Glutaredoxin protein 5 | 0.0025 | 0.0721 | 0.0721 |
Echinococcus granulosus | serine threonine protein kinase nrc | 0.0025 | 0.0738 | 0.0738 |
Schistosoma mansoni | serine/threonine-protein kinase | 0.0028 | 0.0889 | 0.0889 |
Trichomonas vaginalis | AGC family protein kinase | 0.004 | 0.1658 | 1 |
Schistosoma mansoni | ribokinase | 0.002 | 0.0443 | 0.0443 |
Brugia malayi | Protein kinase domain containing protein | 0.004 | 0.1658 | 0.1658 |
Trichomonas vaginalis | AGC family protein kinase | 0.004 | 0.1658 | 1 |
Entamoeba histolytica | fructokinase, putative | 0.002 | 0.0443 | 0.2673 |
Trichomonas vaginalis | AGC family protein kinase | 0.004 | 0.1658 | 1 |
Echinococcus granulosus | pseudouridine metabolizing bifunctional protein | 0.002 | 0.0443 | 0.0443 |
Loa Loa (eye worm) | AGC/RSK/P70 protein kinase | 0.0038 | 0.1507 | 0.1507 |
Trichomonas vaginalis | AGC family protein kinase | 0.004 | 0.1658 | 1 |
Mycobacterium tuberculosis | Ribokinase RbsK | 0.002 | 0.0443 | 0.5 |
Toxoplasma gondii | AGC kinase | 0.0038 | 0.1507 | 0.1113 |
Echinococcus multilocularis | nervana 2 | 0.0025 | 0.0721 | 0.0721 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.