Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Trichomonas vaginalis | AGC family protein kinase | 0.0339 | 0.5912 | 1 |
Trichomonas vaginalis | CMGC family protein kinase | 0.0195 | 0.242 | 0.4093 |
Trichomonas vaginalis | AGC family protein kinase | 0.0339 | 0.5912 | 1 |
Brugia malayi | hypothetical protein | 0.0243 | 0.3589 | 0.5353 |
Trichomonas vaginalis | CMGC family protein kinase | 0.0132 | 0.0913 | 0.1545 |
Giardia lamblia | Kinase, CMGC GSK | 0.0195 | 0.242 | 0.3014 |
Echinococcus multilocularis | glycogen synthase kinase 3 beta | 0.0195 | 0.242 | 0.1658 |
Leishmania major | cyclin | 0.0161 | 0.1615 | 0.1403 |
Leishmania major | protein kinase, putative | 0.0339 | 0.5912 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0507 | 1 | 1 |
Loa Loa (eye worm) | AUR protein kinase | 0.0339 | 0.5912 | 0.5572 |
Schistosoma mansoni | serine/threonine protein kinase | 0.0339 | 0.5912 | 0.5501 |
Entamoeba histolytica | protein kinase domain containing protein | 0.0339 | 0.5912 | 1 |
Entamoeba histolytica | protein kinase domain containing protein | 0.0195 | 0.242 | 0.3014 |
Trichomonas vaginalis | CMGC family protein kinase | 0.0195 | 0.242 | 0.4093 |
Loa Loa (eye worm) | hypothetical protein | 0.0243 | 0.3589 | 0.3055 |
Echinococcus multilocularis | cyclin B | 0.0161 | 0.1615 | 0.0772 |
Schistosoma mansoni | protein kinase | 0.0339 | 0.5912 | 0.5501 |
Trypanosoma brucei | mitotic cyclin 6 | 0.0161 | 0.1615 | 0.1403 |
Trichomonas vaginalis | CMGC family protein kinase | 0.0132 | 0.0913 | 0.1545 |
Loa Loa (eye worm) | CMGC/CDK/CDC2 protein kinase | 0.0132 | 0.0913 | 0.0156 |
Echinococcus granulosus | serine:threonine protein kinase 12 B | 0.0339 | 0.5912 | 0.5501 |
Trypanosoma brucei | protein kinase, putative | 0.0195 | 0.242 | 0.3014 |
Loa Loa (eye worm) | CMGC/CDK/CDK5 protein kinase | 0.0132 | 0.0913 | 0.0156 |
Toxoplasma gondii | cell-cycle-associated protein kinase GSK, putative | 0.0195 | 0.242 | 0.3014 |
Loa Loa (eye worm) | AUR protein kinase | 0.0339 | 0.5912 | 0.5572 |
Trichomonas vaginalis | cyclins, putative | 0.0161 | 0.1615 | 0.2731 |
Plasmodium falciparum | serine/threonine protein kinase, putative | 0.0339 | 0.5912 | 1 |
Leishmania major | CYC2-like cyclin, putative,cyclin 6, putative | 0.0161 | 0.1615 | 0.1403 |
Trichomonas vaginalis | AGC family protein kinase | 0.0339 | 0.5912 | 1 |
Trichomonas vaginalis | cyclins, putative | 0.0161 | 0.1615 | 0.2731 |
Brugia malayi | serine/threonine kinase 12 | 0.0339 | 0.5912 | 1 |
Trichomonas vaginalis | cyclin B, putative | 0.0161 | 0.1615 | 0.2731 |
Echinococcus granulosus | glycogen synthase kinase 3 beta | 0.0195 | 0.242 | 0.1658 |
Entamoeba histolytica | serine/threonine- protein kinase 6 , putative | 0.0339 | 0.5912 | 1 |
Trypanosoma cruzi | cyclin, putative | 0.0161 | 0.1615 | 0.1403 |
Trichomonas vaginalis | cyclin B, putative | 0.0161 | 0.1615 | 0.2731 |
Trichomonas vaginalis | cyclins, putative | 0.0161 | 0.1615 | 0.2731 |
Brugia malayi | Cyclin, N-terminal domain containing protein | 0.0161 | 0.1615 | 0.1403 |
Leishmania major | glycogen synthase kinase, putative;with=GeneDB:LinJ18_V3.0270 | 0.0195 | 0.242 | 0.3014 |
Echinococcus multilocularis | cyclin dependent kinase 5 activator 1 | 0.0507 | 1 | 1 |
Trypanosoma cruzi | glycogen synthase kinase 3, putative | 0.0195 | 0.242 | 0.3014 |
Plasmodium vivax | serine/threonine protein kinase 6, putative | 0.0339 | 0.5912 | 1 |
Plasmodium falciparum | glycogen synthase kinase 3 | 0.0195 | 0.242 | 0.3014 |
Entamoeba histolytica | cyclin, putative | 0.0161 | 0.1615 | 0.1403 |
Loa Loa (eye worm) | hypothetical protein | 0.0161 | 0.1615 | 0.0915 |
Loa Loa (eye worm) | cyclin domain-containing protein | 0.0308 | 0.5176 | 0.4774 |
Schistosoma mansoni | glycogen synthase kinase 3-related (gsk3) (cmgc group III) | 0.0195 | 0.242 | 0.1658 |
Brugia malayi | serine/threonine-protein kinase 6 | 0.0339 | 0.5912 | 1 |
Trypanosoma cruzi | cyclin 6, putative | 0.0161 | 0.1615 | 0.1403 |
Plasmodium vivax | glycogen synthase kinase 3, putative | 0.0195 | 0.242 | 0.3014 |
Echinococcus multilocularis | G2:mitotic specific cyclin B3 | 0.0308 | 0.5176 | 0.4692 |
Echinococcus granulosus | G2:mitotic specific cyclin B3 | 0.0308 | 0.5176 | 0.4692 |
Trichomonas vaginalis | AGC family protein kinase | 0.0339 | 0.5912 | 1 |
Trypanosoma cruzi | aurora B kinase, putative | 0.0339 | 0.5912 | 1 |
Trypanosoma cruzi | cyclin, putative | 0.0161 | 0.1615 | 0.1403 |
Giardia lamblia | Kinase, CMGC GSK | 0.0195 | 0.242 | 0.3014 |
Trichomonas vaginalis | CMGC family protein kinase | 0.0132 | 0.0913 | 0.1545 |
Loa Loa (eye worm) | hypothetical protein | 0.0161 | 0.1615 | 0.0915 |
Echinococcus granulosus | cyclin B | 0.0161 | 0.1615 | 0.0772 |
Schistosoma mansoni | cyclin B3 | 0.0308 | 0.5176 | 0.4692 |
Loa Loa (eye worm) | CMGC/GSK protein kinase | 0.0195 | 0.242 | 0.1788 |
Trypanosoma brucei | aurora B kinase | 0.0339 | 0.5912 | 1 |
Trypanosoma cruzi | CYC2-like cyclin, putative | 0.0161 | 0.1615 | 0.1403 |
Echinococcus granulosus | aurora kinase A | 0.0339 | 0.5912 | 0.5501 |
Schistosoma mansoni | cyclin-dependent kinase 5 activator | 0.0507 | 1 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0243 | 0.3589 | 0.3055 |
Entamoeba histolytica | protein kinase domain containing protein | 0.0195 | 0.242 | 0.3014 |
Toxoplasma gondii | aurora kinase | 0.0339 | 0.5912 | 1 |
Loa Loa (eye worm) | AUR protein kinase | 0.0339 | 0.5912 | 0.5572 |
Entamoeba histolytica | protein kinase, putative | 0.0339 | 0.5912 | 1 |
Trichomonas vaginalis | cyclin B, putative | 0.0161 | 0.1615 | 0.2731 |
Entamoeba histolytica | serine/threonine- protein kinase 6, putative | 0.0339 | 0.5912 | 1 |
Brugia malayi | Cyclin, N-terminal domain containing protein | 0.0308 | 0.5176 | 0.8528 |
Loa Loa (eye worm) | CMGC/GSK protein kinase | 0.0195 | 0.242 | 0.1788 |
Entamoeba histolytica | protein kinase , putative | 0.0339 | 0.5912 | 1 |
Echinococcus multilocularis | protein kinase shaggy | 0.0195 | 0.242 | 0.1658 |
Brugia malayi | intracellular kinase | 0.0195 | 0.242 | 0.3014 |
Giardia lamblia | G2/mitotic-specific cyclin B | 0.0161 | 0.1615 | 0.1403 |
Entamoeba histolytica | serine/threonine protein kinase 6, putative | 0.0339 | 0.5912 | 1 |
Echinococcus granulosus | protein kinase shaggy | 0.0195 | 0.242 | 0.1658 |
Echinococcus multilocularis | serine:threonine protein kinase 12 B | 0.0339 | 0.5912 | 0.5501 |
Schistosoma mansoni | cyclin B | 0.0161 | 0.1615 | 0.0772 |
Giardia lamblia | Aurora kinase | 0.0339 | 0.5912 | 1 |
Trichomonas vaginalis | cyclins, putative | 0.0161 | 0.1615 | 0.2731 |
Brugia malayi | serine/threonine protein kinase 6 | 0.0339 | 0.5912 | 1 |
Trichomonas vaginalis | cyclin B, putative | 0.0161 | 0.1615 | 0.2731 |
Brugia malayi | Cyclin, N-terminal domain containing protein | 0.0161 | 0.1615 | 0.1403 |
Trichomonas vaginalis | cyclin A, putative | 0.0161 | 0.1615 | 0.2731 |
Entamoeba histolytica | protein kinase, putative | 0.0195 | 0.242 | 0.3014 |
Onchocerca volvulus | 0.0195 | 0.242 | 1 | |
Echinococcus multilocularis | aurora kinase A | 0.0339 | 0.5912 | 0.5501 |
Loa Loa (eye worm) | CMGC/CDK/CDC2 protein kinase | 0.0132 | 0.0913 | 0.0156 |
Entamoeba histolytica | protein kinase, putative | 0.0339 | 0.5912 | 1 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
Potency (functional) | 28.1838 uM | PubChem BioAssay. qHTS of GLP-1 Receptor Inverse Agonists (Inhibition Mode). (Class of assay: confirmatory) | ChEMBL. | No reference |
Potency (functional) | 89.1251 uM | PUBCHEM_BIOASSAY: qHTS for Inhibitors of Polymerase Iota. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID588623] | ChEMBL. | No reference |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.