Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Trichomonas vaginalis | bromodomain-containing protein, putative | 0.0242 | 0.2237 | 0.4061 |
Schistosoma mansoni | CREB-binding protein 1 (SmCBP1) | 0.0158 | 0.1315 | 0.2386 |
Trypanosoma brucei | Bromodomain, putative | 0.0038 | 0 | 0.5 |
Trichomonas vaginalis | bromodomain-containing protein, putative | 0.0242 | 0.2237 | 0.4061 |
Trichomonas vaginalis | bromodomain-containing protein, putative | 0.0242 | 0.2237 | 0.4061 |
Plasmodium vivax | histone acetyltransferase GCN5, putative | 0.0038 | 0 | 0.5 |
Trypanosoma cruzi | Bromodomain factor 1 | 0.0038 | 0 | 0.5 |
Leishmania major | hypothetical protein, conserved,predicted bromodomain protein | 0.0038 | 0 | 0.5 |
Trichomonas vaginalis | bromodomain-containing protein, putative | 0.0242 | 0.2237 | 0.4061 |
Trichomonas vaginalis | bromodomain-containing protein, putative | 0.0242 | 0.2237 | 0.4061 |
Giardia lamblia | Kinase, putative | 0.0242 | 0.2237 | 1 |
Schistosoma mansoni | CREB-binding protein 2 | 0.0158 | 0.1315 | 0.2386 |
Trichomonas vaginalis | bromodomain-containing protein, putative | 0.0242 | 0.2237 | 0.4061 |
Trichomonas vaginalis | bromodomain containing protein, putative | 0.0336 | 0.3273 | 0.5939 |
Trichomonas vaginalis | conserved hypothetical protein | 0.0336 | 0.3273 | 0.5939 |
Trichomonas vaginalis | bromodomain-containing protein, putative | 0.054 | 0.551 | 1 |
Plasmodium vivax | bromodomain protein, putative | 0.0038 | 0 | 0.5 |
Echinococcus granulosus | CREB binding protein | 0.0111 | 0.0802 | 0.1455 |
Trichomonas vaginalis | bromodomain-containing protein, putative | 0.0242 | 0.2237 | 0.4061 |
Trichomonas vaginalis | bromodomain-containing protein, putative | 0.0242 | 0.2237 | 0.4061 |
Trichomonas vaginalis | bromodomain-containing protein, putative | 0.0336 | 0.3273 | 0.5939 |
Leishmania major | DNA-binding protein, putative,predicted bromodomain protein | 0.0038 | 0 | 0.5 |
Trypanosoma brucei | Bromodomain, putative | 0.0038 | 0 | 0.5 |
Trichomonas vaginalis | conserved hypothetical protein | 0.0242 | 0.2237 | 0.4061 |
Brugia malayi | hypothetical protein | 0.0613 | 0.6312 | 0.6312 |
Entamoeba histolytica | bromodomain-containing protein | 0.0242 | 0.2237 | 1 |
Trichomonas vaginalis | histone acetyltransferase gcn5, putative | 0.0242 | 0.2237 | 0.4061 |
Trichomonas vaginalis | bromodomain-containing protein, putative | 0.0242 | 0.2237 | 0.4061 |
Trichomonas vaginalis | bromodomain-containing protein, putative | 0.0336 | 0.3273 | 0.5939 |
Schistosoma mansoni | bromodomain-containing protein 3 brd3 | 0.054 | 0.551 | 1 |
Trichomonas vaginalis | bromodomain-containing protein, putative | 0.0242 | 0.2237 | 0.4061 |
Trypanosoma brucei | Bromodomain factor 1 | 0.0038 | 0 | 0.5 |
Trypanosoma cruzi | hypothetical protein, conserved | 0.0038 | 0 | 0.5 |
Trichomonas vaginalis | bromodomain-containing protein, putative | 0.0242 | 0.2237 | 0.4061 |
Echinococcus granulosus | CREB binding protein | 0.0158 | 0.1315 | 0.2386 |
Trypanosoma cruzi | Bromodomain, putative | 0.0038 | 0 | 0.5 |
Trichomonas vaginalis | bromodomain-containing protein, putative | 0.0242 | 0.2237 | 0.4061 |
Trichomonas vaginalis | bromodomain-containing protein, putative | 0.0242 | 0.2237 | 0.4061 |
Trypanosoma cruzi | Bromodomain, putative | 0.0038 | 0 | 0.5 |
Trypanosoma brucei | AAA ATPase, putative | 0.0038 | 0 | 0.5 |
Leishmania major | hypothetical protein, conserved | 0.0038 | 0 | 0.5 |
Trypanosoma brucei | bromodomain factor 2 protein, putative | 0.0038 | 0 | 0.5 |
Leishmania major | hypothetical protein, conserved | 0.0038 | 0 | 0.5 |
Trichomonas vaginalis | bromodomain containing protein, putative | 0.0242 | 0.2237 | 0.4061 |
Plasmodium vivax | hypothetical protein, conserved | 0.0038 | 0 | 0.5 |
Trichomonas vaginalis | bromodomain-containing protein, putative | 0.0242 | 0.2237 | 0.4061 |
Brugia malayi | Bromodomain containing protein | 0.054 | 0.551 | 0.551 |
Trypanosoma cruzi | bromodomain factor 2 protein | 0.0038 | 0 | 0.5 |
Trypanosoma cruzi | bromodomain-containing protein 3 | 0.0038 | 0 | 0.5 |
Brugia malayi | TAZ zinc finger family protein | 0.0158 | 0.1315 | 0.1315 |
Trypanosoma cruzi | Bromodomain, putative | 0.0038 | 0 | 0.5 |
Plasmodium vivax | bromodomain protein, putative | 0.0038 | 0 | 0.5 |
Entamoeba histolytica | bromodomain-containing protein | 0.0242 | 0.2237 | 1 |
Echinococcus multilocularis | Bromodomain containing protein | 0.0242 | 0.2237 | 0.4061 |
Loa Loa (eye worm) | bromodomain containing protein | 0.0242 | 0.2237 | 0.2237 |
Plasmodium falciparum | bromodomain protein 1 | 0.0038 | 0 | 0.5 |
Toxoplasma gondii | bromodomain-containing protein | 0.0242 | 0.2237 | 1 |
Trichomonas vaginalis | bromodomain-containing protein, putative | 0.0242 | 0.2237 | 0.4061 |
Trichomonas vaginalis | bromodomain-containing protein, putative | 0.0336 | 0.3273 | 0.5939 |
Trichomonas vaginalis | bromodomain-containing protein, putative | 0.0242 | 0.2237 | 0.4061 |
Plasmodium vivax | conserved Plasmodium protein, unknown function | 0.0038 | 0 | 0.5 |
Echinococcus granulosus | bromodomain containing 2 | 0.054 | 0.551 | 1 |
Trichomonas vaginalis | bromodomain-containing protein, putative | 0.0242 | 0.2237 | 0.4061 |
Loa Loa (eye worm) | CBP-B | 0.012 | 0.0906 | 0.0906 |
Trichomonas vaginalis | bromodomain-containing protein, putative | 0.054 | 0.551 | 1 |
Plasmodium vivax | bromodomain protein, putative | 0.0038 | 0 | 0.5 |
Trichomonas vaginalis | bromodomain-containing protein, putative | 0.0242 | 0.2237 | 0.4061 |
Trichomonas vaginalis | bromodomain-containing protein, putative | 0.0242 | 0.2237 | 0.4061 |
Trypanosoma cruzi | Bromodomain, putative | 0.0038 | 0 | 0.5 |
Onchocerca volvulus | 0.0242 | 0.2237 | 1 | |
Trichomonas vaginalis | bromodomain-containing protein 4, brd4, putative | 0.0242 | 0.2237 | 0.4061 |
Loa Loa (eye worm) | hypothetical protein | 0.0057 | 0.0213 | 0.0213 |
Echinococcus multilocularis | bromodomain containing 2 | 0.054 | 0.551 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0949 | 1 | 1 |
Trypanosoma brucei | Bromodomain, putative | 0.0038 | 0 | 0.5 |
Trypanosoma cruzi | Bromodomain, putative | 0.0038 | 0 | 0.5 |
Trichomonas vaginalis | conserved hypothetical protein | 0.0298 | 0.2857 | 0.5185 |
Echinococcus multilocularis | CREB binding protein | 0.0119 | 0.0894 | 0.1623 |
Entamoeba histolytica | bromodomain-containing protein | 0.0242 | 0.2237 | 1 |
Plasmodium falciparum | bromodomain protein 2, putative | 0.0038 | 0 | 0.5 |
Plasmodium vivax | SET domain containing protein | 0.0038 | 0 | 0.5 |
Plasmodium falciparum | bromodomain protein, putative | 0.0038 | 0 | 0.5 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
Activity (functional) | = 83.37 % | Growth inhibition of human MDA-MB-468 cells assessed as cell growth at 10 uM after 48 hrs by sulforhodamine B assay | ChEMBL. | 23732996 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.