Species | Target name | Source | Bibliographic reference |
---|---|---|---|
Homo sapiens | renin | Starlite/ChEMBL | References |
Species | Potential target | Known druggable target | Length | Alignment span | Identity |
---|---|---|---|---|---|
Plasmodium falciparum | plasmepsin X | renin | 406 aa | 352 aa | 26.4 % |
Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Echinococcus multilocularis | casein kinase I delta | 0.1475 | 1 | 1 |
Echinococcus multilocularis | casein kinase i | 0.1475 | 1 | 1 |
Loa Loa (eye worm) | CK1/CK1/CK1-A protein kinase | 0.1475 | 1 | 1 |
Trypanosoma cruzi | casein kinase, delta isoform, putative | 0.1475 | 1 | 1 |
Echinococcus granulosus | casein kinase I delta | 0.1475 | 1 | 1 |
Trypanosoma cruzi | casein kinase, putative | 0.1475 | 1 | 1 |
Echinococcus multilocularis | casein kinase I alpha | 0.1475 | 1 | 1 |
Schistosoma mansoni | serine/threonine protein kinase | 0.1475 | 1 | 1 |
Trichomonas vaginalis | CK1 family protein kinase | 0.1475 | 1 | 1 |
Toxoplasma gondii | casein kinase I | 0.1475 | 1 | 1 |
Echinococcus granulosus | casein kinase I alpha | 0.1475 | 1 | 1 |
Onchocerca volvulus | 0.1475 | 1 | 1 | |
Plasmodium falciparum | casein kinase 1 | 0.1475 | 1 | 1 |
Echinococcus multilocularis | casein kinase I alpha | 0.1475 | 1 | 1 |
Schistosoma mansoni | cathepsin D (A01 family) | 0.0174 | 0.0812 | 0.0812 |
Giardia lamblia | Kinase, CK1 Casein kinase | 0.1475 | 1 | 0.5 |
Brugia malayi | casein kinase I | 0.1475 | 1 | 0.5 |
Trypanosoma cruzi | casein kinase, putative | 0.1475 | 1 | 1 |
Echinococcus granulosus | casein kinase I alpha | 0.1475 | 1 | 1 |
Trypanosoma cruzi | casein kinase, putative | 0.1475 | 1 | 1 |
Echinococcus multilocularis | casein kinase I delta | 0.1475 | 1 | 1 |
Plasmodium vivax | casein kinase 1, putative | 0.1475 | 1 | 1 |
Trichomonas vaginalis | CK1 family protein kinase | 0.1475 | 1 | 1 |
Trypanosoma cruzi | casein kinase, putative | 0.1475 | 1 | 1 |
Leishmania major | casein kinase, putative | 0.1475 | 1 | 0.5 |
Echinococcus granulosus | casein kinase I alpha | 0.1475 | 1 | 1 |
Schistosoma mansoni | protein kinase | 0.1475 | 1 | 1 |
Trypanosoma brucei | casein kinase I, isoform 2 | 0.1475 | 1 | 0.5 |
Loa Loa (eye worm) | CK1/CK1/CK1-D protein kinase | 0.1475 | 1 | 1 |
Entamoeba histolytica | casein kinase, putative | 0.1475 | 1 | 0.5 |
Entamoeba histolytica | casein kinase 1, putative | 0.1475 | 1 | 0.5 |
Echinococcus granulosus | casein kinase I delta | 0.1475 | 1 | 1 |
Trichomonas vaginalis | CK1 family protein kinase | 0.1475 | 1 | 1 |
Echinococcus granulosus | casein kinase i | 0.1475 | 1 | 1 |
Loa Loa (eye worm) | CK1/CK1/CK1-A protein kinase | 0.1475 | 1 | 1 |
Trypanosoma cruzi | casein kinase, putative | 0.1475 | 1 | 1 |
Schistosoma mansoni | cathepsin D (A01 family) | 0.0174 | 0.0812 | 0.0812 |
Echinococcus multilocularis | casein kinase I alpha | 0.1475 | 1 | 1 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
IC50 (binding) | = 0.57 nM | Inhibition of human plasma renin | ChEMBL. | 3531517 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.