Species | Target name | Source | Bibliographic reference |
---|---|---|---|
Plasmodium falciparum | dihydroorotate dehydrogenase | Curated by TDR Targets | No references |
Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Loa Loa (eye worm) | acetyltransferase | 0.0151 | 0.7333 | 1 |
Trypanosoma cruzi | dihydroorotate dehydrogenase, putative | 0.02 | 1 | 1 |
Trichomonas vaginalis | dihydroorotate dehydrogenase, putative | 0.0078 | 0.3406 | 1 |
Echinococcus multilocularis | aldehyde dehydrogenase, mitochondrial | 0.0061 | 0.2476 | 0.3348 |
Echinococcus granulosus | lamin | 0.0033 | 0.0943 | 0.1288 |
Echinococcus multilocularis | musashi | 0.0033 | 0.0943 | 0.1248 |
Echinococcus granulosus | dihydropyrimidine dehydrogenase NADP | 0.0078 | 0.3406 | 0.4771 |
Schistosoma mansoni | aldehyde dehydrogenase | 0.0061 | 0.2476 | 0.1693 |
Echinococcus granulosus | jun protein | 0.0101 | 0.4665 | 0.6551 |
Schistosoma mansoni | dihydroorotate dehydrogenase | 0.02 | 1 | 1 |
Plasmodium falciparum | dihydroorotate dehydrogenase | 0.02 | 1 | 1 |
Toxoplasma gondii | dihydroorotate dehydrogenase reveal, putative | 0.02 | 1 | 1 |
Giardia lamblia | Histone acetyltransferase GCN5 | 0.0041 | 0.138 | 0.5 |
Echinococcus multilocularis | dihydropyrimidine dehydrogenase (NADP+) | 0.0078 | 0.3406 | 0.4622 |
Loa Loa (eye worm) | intermediate filament protein | 0.0033 | 0.0943 | 0.1286 |
Loa Loa (eye worm) | CYP4Cod1 | 0.002 | 0.0272 | 0.0371 |
Brugia malayi | Dihydroorotate dehydrogenase, mitochondrial precursor, putative | 0.02 | 1 | 1 |
Schistosoma mansoni | hypothetical protein | 0.0082 | 0.3638 | 0.2976 |
Toxoplasma gondii | aldehyde dehydrogenase | 0.0061 | 0.2476 | 0.1065 |
Brugia malayi | bZIP transcription factor family protein | 0.0101 | 0.4665 | 0.4597 |
Echinococcus granulosus | dihydropyrimidine dehydrogenase NADP | 0.0078 | 0.3406 | 0.4771 |
Mycobacterium leprae | Probable dihydroorotate dehydrogenase PyrD | 0.02 | 1 | 0.5 |
Schistosoma mansoni | jun-related protein | 0.0082 | 0.3638 | 0.2976 |
Echinococcus granulosus | Basic leucine zipper bZIP transcription factor | 0.0101 | 0.4665 | 0.6551 |
Echinococcus granulosus | lamin dm0 | 0.0033 | 0.0943 | 0.1288 |
Echinococcus granulosus | histone acetyltransferase KAT2B | 0.0147 | 0.7105 | 1 |
Echinococcus multilocularis | lamin | 0.0033 | 0.0943 | 0.1248 |
Echinococcus granulosus | histone acetyltransferase KAT2B | 0.0044 | 0.1579 | 0.2188 |
Mycobacterium tuberculosis | Probable dihydroorotate dehydrogenase PyrD | 0.02 | 1 | 1 |
Trypanosoma cruzi | dihydroorotate dehydrogenase, putative | 0.0078 | 0.3406 | 0.3222 |
Echinococcus multilocularis | gcn5proteinral control of amino acid synthesis | 0.0151 | 0.7333 | 1 |
Trichomonas vaginalis | dihydropyrimidine dehydrogenase, putative | 0.0078 | 0.3406 | 1 |
Brugia malayi | hypothetical protein | 0.008 | 0.3488 | 0.3405 |
Loa Loa (eye worm) | hypothetical protein | 0.0099 | 0.4515 | 0.6157 |
Trichomonas vaginalis | dihydroorotate dehydrogenase, putative | 0.0078 | 0.3406 | 1 |
Entamoeba histolytica | dihydropyrimidine dehydrogenase, putative | 0.0078 | 0.3406 | 1 |
Trypanosoma cruzi | dihydroorotate dehydrogenase (fumarate), putative | 0.02 | 1 | 1 |
Brugia malayi | Cytochrome P450 family protein | 0.002 | 0.0272 | 0.0148 |
Loa Loa (eye worm) | hypothetical protein | 0.0032 | 0.0911 | 0.1242 |
Mycobacterium ulcerans | aldehyde dehydrogenase | 0.0061 | 0.2476 | 0.2266 |
Brugia malayi | intermediate filament protein | 0.0033 | 0.0943 | 0.0828 |
Loa Loa (eye worm) | intermediate filament tail domain-containing protein | 0.0033 | 0.0943 | 0.1286 |
Trypanosoma cruzi | dihydroorotate dehydrogenase, putative | 0.02 | 1 | 1 |
Mycobacterium ulcerans | aldehyde dehydrogenase | 0.0061 | 0.2476 | 0.2266 |
Brugia malayi | Cytochrome P450 family protein | 0.002 | 0.0272 | 0.0148 |
Loa Loa (eye worm) | cytochrome P450 family protein | 0.002 | 0.0272 | 0.0371 |
Schistosoma mansoni | aldehyde dehydrogenase | 0.0061 | 0.2476 | 0.1693 |
Schistosoma mansoni | gcn5proteinral control of amino-acid synthesis 5-like 2 gcnl2 | 0.0151 | 0.7333 | 0.7056 |
Echinococcus multilocularis | lamin dm0 | 0.0033 | 0.0943 | 0.1248 |
Brugia malayi | acetyltransferase, GNAT family protein | 0.0151 | 0.7333 | 0.7299 |
Mycobacterium ulcerans | dihydroorotate dehydrogenase 2 | 0.02 | 1 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0016 | 0.0032 | 0.0044 |
Wolbachia endosymbiont of Brugia malayi | dihydroorotate dehydrogenase 2 | 0.02 | 1 | 0.5 |
Trichomonas vaginalis | dihydroorotate dehydrogenase, putative | 0.0078 | 0.3406 | 1 |
Loa Loa (eye worm) | cytochrome P450 family protein | 0.002 | 0.0272 | 0.0371 |
Loa Loa (eye worm) | cytoplasmic intermediate filament protein | 0.0017 | 0.0126 | 0.0171 |
Trichomonas vaginalis | dihydroorotate dehydrogenase, putative | 0.0078 | 0.3406 | 1 |
Echinococcus multilocularis | jun protein | 0.0101 | 0.4665 | 0.6346 |
Echinococcus granulosus | aldehyde dehydrogenase mitochondrial | 0.0061 | 0.2476 | 0.3456 |
Echinococcus multilocularis | dihydropyrimidine dehydrogenase (NADP+) | 0.0078 | 0.3406 | 0.4622 |
Loa Loa (eye worm) | hypothetical protein | 0.0033 | 0.0943 | 0.1286 |
Trichomonas vaginalis | dihydroorotate dehydrogenase, putative | 0.0078 | 0.3406 | 1 |
Leishmania major | dihydroorotate dehydrogenase | 0.02 | 1 | 1 |
Brugia malayi | Zinc finger, C2H2 type family protein | 0.0078 | 0.3406 | 0.3323 |
Leishmania major | aldehyde dehydrogenase, mitochondrial precursor | 0.0061 | 0.2476 | 0.2266 |
Plasmodium vivax | dihydroorotate dehydrogenase, mitochondrial precursor, putative | 0.02 | 1 | 1 |
Onchocerca volvulus | 0.008 | 0.3488 | 1 | |
Brugia malayi | Intermediate filament tail domain containing protein | 0.0033 | 0.0943 | 0.0828 |
Trypanosoma brucei | dihydroorotate dehydrogenase (fumarate) | 0.02 | 1 | 1 |
Echinococcus multilocularis | Basic leucine zipper (bZIP) transcription factor | 0.0101 | 0.4665 | 0.6346 |
Brugia malayi | Cytochrome P450 family protein | 0.0051 | 0.1926 | 0.1823 |
Loa Loa (eye worm) | cytochrome P450 family protein | 0.0051 | 0.1926 | 0.2626 |
Mycobacterium ulcerans | aldehyde dehydrogenase | 0.0061 | 0.2476 | 0.2266 |
Echinococcus granulosus | intermediate filament protein | 0.0033 | 0.0943 | 0.1288 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
59 literature references were collected for this gene.